JP2009519974A5 - - Google Patents

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Publication number
JP2009519974A5
JP2009519974A5 JP2008545979A JP2008545979A JP2009519974A5 JP 2009519974 A5 JP2009519974 A5 JP 2009519974A5 JP 2008545979 A JP2008545979 A JP 2008545979A JP 2008545979 A JP2008545979 A JP 2008545979A JP 2009519974 A5 JP2009519974 A5 JP 2009519974A5
Authority
JP
Japan
Prior art keywords
compound
medicament
effective amount
aurora kinase
mammal
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2008545979A
Other languages
English (en)
Japanese (ja)
Other versions
JP2009519974A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2006/062112 external-priority patent/WO2007120333A2/en
Publication of JP2009519974A publication Critical patent/JP2009519974A/ja
Publication of JP2009519974A5 publication Critical patent/JP2009519974A5/ja
Pending legal-status Critical Current

Links

JP2008545979A 2005-12-16 2006-12-14 四環系キナーゼ阻害剤 Pending JP2009519974A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US75123405P 2005-12-16 2005-12-16
PCT/US2006/062112 WO2007120333A2 (en) 2005-12-16 2006-12-14 Tetracyclic kinase inhibitors

Publications (2)

Publication Number Publication Date
JP2009519974A JP2009519974A (ja) 2009-05-21
JP2009519974A5 true JP2009519974A5 (https=) 2010-02-04

Family

ID=38610005

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008545979A Pending JP2009519974A (ja) 2005-12-16 2006-12-14 四環系キナーゼ阻害剤

Country Status (6)

Country Link
US (1) US20090131407A1 (https=)
EP (1) EP1968581A4 (https=)
JP (1) JP2009519974A (https=)
AU (1) AU2006342024A1 (https=)
CA (1) CA2631871A1 (https=)
WO (1) WO2007120333A2 (https=)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090203671A1 (en) * 2007-11-27 2009-08-13 Abbott Laboratories Method of treating cancer
US8716308B2 (en) 2008-01-11 2014-05-06 Albany Molecular Research, Inc. (1-azinone)-substituted pyridoindoles
MX2010008700A (es) 2008-02-22 2010-08-30 Hoffmann La Roche Moduladores de beta-amiloide.
WO2010039187A2 (en) * 2008-09-23 2010-04-08 University Of Maryland, Baltimore County Fused diimidazodiazepine compounds and methods of use and manufacture thereof
ES2429517T3 (es) 2008-10-09 2013-11-15 F. Hoffmann-La Roche Ag Moduladores para la beta amiloide
CN102209537A (zh) 2008-11-10 2011-10-05 弗·哈夫曼-拉罗切有限公司 杂环γ分泌酶调节剂
US8629158B2 (en) 2009-07-01 2014-01-14 Albany Molecular Research, Inc. Azabicycloalkane-indole and azabicycloalkane-pyrrolo-pyridine MCH-1 antagonists, methods of making, and use thereof
WO2011003012A1 (en) 2009-07-01 2011-01-06 Albany Molecular Research, Inc. Azinone-substituted azapolycycle mch-1 antagonists, methods of making, and use thereof
US9073925B2 (en) 2009-07-01 2015-07-07 Albany Molecular Research, Inc. Azinone-substituted azabicycloalkane-indole and azabicycloalkane-pyrrolo-pyridine MCH-1 antagonists, methods of making, and use thereof
US8637501B2 (en) 2009-07-01 2014-01-28 Albany Molecular Research, Inc. Azinone-substituted azepino[b]indole and pyrido-pyrrolo-azepine MCH-1 antagonists, methods of making, and use thereof
US8486967B2 (en) 2010-02-17 2013-07-16 Hoffmann-La Roche Inc. Heteroaryl substituted piperidines
WO2012088038A2 (en) 2010-12-21 2012-06-28 Albany Molecular Research, Inc. Piperazinone-substituted tetrahydro-carboline mch-1 antagonists, methods of making, and uses thereof
US8993765B2 (en) 2010-12-21 2015-03-31 Albany Molecular Research, Inc. Tetrahydro-azacarboline MCH-1 antagonists, methods of making, and uses thereof
CN106674081A (zh) * 2016-12-18 2017-05-17 南京理工大学 一种3‑甲硫基吲哚衍生物合成方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3772325A (en) * 1972-03-24 1973-11-13 American Cyanamid Co Novel hexahydro cyclohept(b)indoles
EP1127051A2 (en) * 1998-11-06 2001-08-29 Basf Aktiengesellschaft Tricyclic pyrazole derivatives
BRPI0407544A (pt) * 2003-02-17 2006-02-14 Pharmacia Italia Spa derivados de pirazol tetracìclicos como inibidores da cinase, processo para a sua preparação e composições farmacêuticas que os compreendem
US20050032869A1 (en) * 2003-07-08 2005-02-10 Pharmacia Italia S.P.A. Pyrazolyl-indole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
US20070254877A1 (en) * 2004-06-02 2007-11-01 Takada Pharmaceutical Company Limited Indole Derivative and Use for Treatment of Cancer

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