JP2008545699A - 選択的エストロゲン受容体モジュレーターとしてのシクロアルキリデン化合物 - Google Patents
選択的エストロゲン受容体モジュレーターとしてのシクロアルキリデン化合物 Download PDFInfo
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- JP2008545699A JP2008545699A JP2008513693A JP2008513693A JP2008545699A JP 2008545699 A JP2008545699 A JP 2008545699A JP 2008513693 A JP2008513693 A JP 2008513693A JP 2008513693 A JP2008513693 A JP 2008513693A JP 2008545699 A JP2008545699 A JP 2008545699A
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- phenyl
- methyl
- tetramethylcyclohexylidene
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- disease
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- 208000025421 tumor of uterus Diseases 0.000 description 1
- 229940070710 valerate Drugs 0.000 description 1
- NQPDZGIKBAWPEJ-UHFFFAOYSA-N valeric acid Chemical compound CCCCC(O)=O NQPDZGIKBAWPEJ-UHFFFAOYSA-N 0.000 description 1
- 125000000391 vinyl group Chemical group [H]C([*])=C([H])[H] 0.000 description 1
- 229920002554 vinyl polymer Polymers 0.000 description 1
- 230000003612 virological effect Effects 0.000 description 1
- 239000011782 vitamin Substances 0.000 description 1
- 235000013343 vitamin Nutrition 0.000 description 1
- 229940088594 vitamin Drugs 0.000 description 1
- 229930003231 vitamin Natural products 0.000 description 1
- 239000007762 w/o emulsion Substances 0.000 description 1
- 239000008215 water for injection Substances 0.000 description 1
- 235000010493 xanthan gum Nutrition 0.000 description 1
- 239000000230 xanthan gum Substances 0.000 description 1
- 229920001285 xanthan gum Polymers 0.000 description 1
- 229940082509 xanthan gum Drugs 0.000 description 1
- 229930195724 β-lactose Natural products 0.000 description 1
Classifications
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- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/18—Systems containing only non-condensed rings with a ring being at least seven-membered
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US68443305P | 2005-05-25 | 2005-05-25 | |
| PCT/US2006/020185 WO2006127871A2 (en) | 2005-05-25 | 2006-05-24 | Cycloalkylidene compounds as selective estrogen receptor modulators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008545699A true JP2008545699A (ja) | 2008-12-18 |
| JP2008545699A5 JP2008545699A5 (https=) | 2009-05-14 |
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ID=37309167
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008513693A Pending JP2008545699A (ja) | 2005-05-25 | 2006-05-24 | 選択的エストロゲン受容体モジュレーターとしてのシクロアルキリデン化合物 |
Country Status (7)
| Country | Link |
|---|---|
| US (2) | US7723393B2 (https=) |
| EP (1) | EP1891026B1 (https=) |
| JP (1) | JP2008545699A (https=) |
| AT (1) | ATE473968T1 (https=) |
| DE (1) | DE602006015465D1 (https=) |
| ES (1) | ES2348838T3 (https=) |
| WO (1) | WO2006127871A2 (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007500705A (ja) * | 2003-07-28 | 2007-01-18 | スミスクライン ビーチャム コーポレーション | 化合物 |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5193196B2 (ja) | 2006-06-02 | 2013-05-08 | ペア ツリー ウーマンズ ヘルス ケア | 萎縮性膣炎の治療の方法 |
| CN102786394B (zh) * | 2012-07-30 | 2017-03-01 | 中国医学科学院医药生物技术研究所 | 取代双芳基亚甲基环烷基衍生物及其制备方法和应用 |
| AT514594B1 (de) | 2013-09-06 | 2015-02-15 | Durst Phototech Digital Tech | Photoinitiator |
| US9750716B2 (en) * | 2015-03-19 | 2017-09-05 | Wendy Anne Epstein | Compounds and forms of treatment for female sexual disorders |
| JP6545746B2 (ja) * | 2017-05-09 | 2019-07-17 | 山田化学工業株式会社 | 色素化合物 |
| WO2024245169A1 (zh) * | 2023-05-26 | 2024-12-05 | 北京盛诺基医药科技股份有限公司 | 一种靶向雌激素受体的protac化合物及其制备方法和用途 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007500705A (ja) * | 2003-07-28 | 2007-01-18 | スミスクライン ビーチャム コーポレーション | 化合物 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2000072612A (ja) * | 1998-06-17 | 2000-03-07 | Nonogawa Shoji Kk | 皮膚外用剤 |
-
2006
- 2006-05-24 US US11/915,436 patent/US7723393B2/en not_active Expired - Fee Related
- 2006-05-24 WO PCT/US2006/020185 patent/WO2006127871A2/en not_active Ceased
- 2006-05-24 ES ES06760363T patent/ES2348838T3/es active Active
- 2006-05-24 JP JP2008513693A patent/JP2008545699A/ja active Pending
- 2006-05-24 DE DE602006015465T patent/DE602006015465D1/de active Active
- 2006-05-24 AT AT06760363T patent/ATE473968T1/de not_active IP Right Cessation
- 2006-05-24 EP EP06760363A patent/EP1891026B1/en active Active
-
2010
- 2010-05-24 US US12/785,788 patent/US20100261772A1/en not_active Abandoned
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007500705A (ja) * | 2003-07-28 | 2007-01-18 | スミスクライン ビーチャム コーポレーション | 化合物 |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007500705A (ja) * | 2003-07-28 | 2007-01-18 | スミスクライン ビーチャム コーポレーション | 化合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| ES2348838T3 (es) | 2010-12-15 |
| DE602006015465D1 (de) | 2010-08-26 |
| EP1891026B1 (en) | 2010-07-14 |
| WO2006127871A3 (en) | 2007-02-01 |
| ATE473968T1 (de) | 2010-07-15 |
| WO2006127871A2 (en) | 2006-11-30 |
| US20080167360A1 (en) | 2008-07-10 |
| US20100261772A1 (en) | 2010-10-14 |
| EP1891026A2 (en) | 2008-02-27 |
| US7723393B2 (en) | 2010-05-25 |
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