JP2008540685A5 - - Google Patents

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Publication number
JP2008540685A5
JP2008540685A5 JP2008512588A JP2008512588A JP2008540685A5 JP 2008540685 A5 JP2008540685 A5 JP 2008540685A5 JP 2008512588 A JP2008512588 A JP 2008512588A JP 2008512588 A JP2008512588 A JP 2008512588A JP 2008540685 A5 JP2008540685 A5 JP 2008540685A5
Authority
JP
Japan
Prior art keywords
oxolan
hydroxymethyl
purin
dihydroxy
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2008512588A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008540685A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2006/019694 external-priority patent/WO2006125211A1/en
Publication of JP2008540685A publication Critical patent/JP2008540685A/ja
Publication of JP2008540685A5 publication Critical patent/JP2008540685A5/ja
Pending legal-status Critical Current

Links

JP2008512588A 2005-05-19 2006-05-19 A1アデノシンレセプターアゴニスト Pending JP2008540685A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68350505P 2005-05-19 2005-05-19
PCT/US2006/019694 WO2006125211A1 (en) 2005-05-19 2006-05-19 A1 adenosine receptor agonists

Publications (2)

Publication Number Publication Date
JP2008540685A JP2008540685A (ja) 2008-11-20
JP2008540685A5 true JP2008540685A5 (https=) 2009-07-02

Family

ID=36950224

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008512588A Pending JP2008540685A (ja) 2005-05-19 2006-05-19 A1アデノシンレセプターアゴニスト

Country Status (5)

Country Link
US (2) US7514417B2 (https=)
EP (1) EP1881991A1 (https=)
JP (1) JP2008540685A (https=)
CA (1) CA2609117A1 (https=)
WO (1) WO2006125211A1 (https=)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008000743A2 (en) * 2006-06-27 2008-01-03 Biovitrum Ab (Publ) Novel 2',3'-methylidene acetyl adenosine prodrugs for use as prodrugs for adenosine receptor agonists
EP2132208A1 (en) 2007-03-28 2009-12-16 NeuroSearch AS Purinyl derivatives and their use as potassium channel modulators
JP2010522719A (ja) * 2007-03-28 2010-07-08 ノイロサーチ アクティーゼルスカブ プリニル誘導体及びカリウムチャネルモジュレーターとしてのそれらの使用
EP2268641B1 (en) * 2008-03-26 2014-09-03 Advinus Therapeutics Pvt. Ltd. Heterocyclic compounds as adenosine receptor antagonist
WO2010034707A1 (en) 2008-09-26 2010-04-01 Neurosearch A/S Substituted purinyl-pyrazol derivatives and their use as potassium channel modulators
CA2876780A1 (en) 2012-06-26 2014-01-03 Saniona Aps A phenyl triazole derivative and its use for modulating the gabaa receptor complex
JO3215B1 (ar) 2012-08-09 2018-03-08 Phenex Pharmaceuticals Ag حلقات غير متجانسة بها 5 ذرات تحتوي على النيتروجين بها استبدال بكربوكساميد أو سلفوناميد كمعدلات لمستقبل نووي غير محمي RORy
US9422267B2 (en) 2012-12-26 2016-08-23 Medivation Technologies, Inc. Fused pyrimidine compounds and use thereof
WO2022143740A1 (zh) * 2020-12-29 2022-07-07 浙江春禾医药科技有限公司 A3腺苷受体激动剂及其制备方法和用途
JP2026500305A (ja) 2022-12-16 2026-01-06 アストラゼネカ・アクチエボラーグ 2,6,9三置換プリン

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030078232A1 (en) * 2001-08-08 2003-04-24 Elfatih Elzein Adenosine receptor A3 agonists
US7262176B2 (en) * 2001-08-08 2007-08-28 Cv Therapeutics, Inc. Adenosine A3 receptor agonists

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