JP2008534653A - 新規エナンチオマー及びモノアミン神経伝達物質再取り込み阻害剤としてのそれらの使用 - Google Patents

新規エナンチオマー及びモノアミン神経伝達物質再取り込み阻害剤としてのそれらの使用 Download PDF

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JP2008534653A
JP2008534653A JP2008504765A JP2008504765A JP2008534653A JP 2008534653 A JP2008534653 A JP 2008534653A JP 2008504765 A JP2008504765 A JP 2008504765A JP 2008504765 A JP2008504765 A JP 2008504765A JP 2008534653 A JP2008534653 A JP 2008534653A
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oct
ene
disorder
enantiopure
azabicyclo
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JP2008534653A5 (enExample
Inventor
ペーターズ、ダン
ダール、ビョルン、エイチ.
オルセン、ドルセ、フィルテンベルイ
ニールセン、エルセベット、オステルガード
オルセン、グンナー、エム.
レッドローブ、ジョン、ポール
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ノイロサーチ アクティーゼルスカブ
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Publication of JP2008534653A5 publication Critical patent/JP2008534653A5/ja
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
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  • Ophthalmology & Optometry (AREA)
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  • Hospice & Palliative Care (AREA)
JP2008504765A 2005-04-08 2006-04-06 新規エナンチオマー及びモノアミン神経伝達物質再取り込み阻害剤としてのそれらの使用 Abandoned JP2008534653A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
DKPA200500505 2005-04-08
US66991805P 2005-04-11 2005-04-11
DKPA200501572 2005-11-11
US73633105P 2005-11-15 2005-11-15
PCT/EP2006/061363 WO2006108789A1 (en) 2005-04-08 2006-04-06 Novel enantiomers and their use as monoamine neurotransmitter re-uptake inhibitors

Publications (2)

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JP2008534653A true JP2008534653A (ja) 2008-08-28
JP2008534653A5 JP2008534653A5 (enExample) 2009-05-28

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JP2008504765A Abandoned JP2008534653A (ja) 2005-04-08 2006-04-06 新規エナンチオマー及びモノアミン神経伝達物質再取り込み阻害剤としてのそれらの使用

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US (1) US20090137625A1 (enExample)
EP (2) EP2272847A1 (enExample)
JP (1) JP2008534653A (enExample)
WO (1) WO2006108789A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI415850B (zh) * 2007-07-20 2013-11-21 Theravance Inc 製備mu類鴉片受體拮抗劑之中間物的方法
DE102007063210A1 (de) * 2007-12-20 2009-06-25 Eberhard-Karls-Universität Tübingen Universitätsklinikum Arzneimittel zur Behandlung von Phantomphänomenen

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2233541C (en) * 1995-10-13 2002-04-30 Neurosearch A/S 8-azabicyclo[3.2.1]oct-2-ene derivatives, their preparation and use
CZ285571B6 (cs) 1995-11-02 1999-09-15 Neurosearch A/S Kondenzované tropanové deriváty, způsob jejich výroby, farmaceutické prostředky, které je obsahují a jejich použití k léčení
TR199801641T2 (xx) 1996-02-22 1998-11-23 Neurosearch A/S Tropan t�revleri bunlar�n haz�rlanmas� ve kullan�m�
WO2000032600A1 (en) * 1998-11-27 2000-06-08 Neurosearch A/S 8-azabicyclo[3.2.1]oct-2-ene and -octane derivatives

Also Published As

Publication number Publication date
WO2006108789A1 (en) 2006-10-19
EP1869033A1 (en) 2007-12-26
EP2272847A1 (en) 2011-01-12
US20090137625A1 (en) 2009-05-28

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