JP2008533065A - アミノカルボニル置換８−ｎ−ベンゾイミダゾール、その製造方法及びその医薬としての使用 - Google Patents
アミノカルボニル置換８−ｎ−ベンゾイミダゾール、その製造方法及びその医薬としての使用 Download PDFInfo
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- JP2008533065A JP2008533065A JP2008501195A JP2008501195A JP2008533065A JP 2008533065 A JP2008533065 A JP 2008533065A JP 2008501195 A JP2008501195 A JP 2008501195A JP 2008501195 A JP2008501195 A JP 2008501195A JP 2008533065 A JP2008533065 A JP 2008533065A
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- Prior art keywords
- alkyl
- aryl
- alkylene
- heterocyclyl
- cycloalkyl
- Prior art date
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- Abandoned
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| DE102005012873A DE102005012873B4 (de) | 2005-03-19 | 2005-03-19 | Aminocarbonyl substituierte 8-N-Benzimidazole, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| PCT/EP2006/002056 WO2006099941A1 (de) | 2005-03-19 | 2006-03-07 | Aminocarbonyl substituierte 8-n-benzimidazole, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
Publications (2)
| Publication Number | Publication Date |
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| JP2008533065A true JP2008533065A (ja) | 2008-08-21 |
| JP2008533065A5 JP2008533065A5 (cg-RX-API-DMAC7.html) | 2009-04-23 |
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| JP2008501195A Abandoned JP2008533065A (ja) | 2005-03-19 | 2006-03-07 | アミノカルボニル置換８−ｎ−ベンゾイミダゾール、その製造方法及びその医薬としての使用 |
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| US (1) | US8138207B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP1863789B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP2008533065A (cg-RX-API-DMAC7.html) |
| AU (1) | AU2006226638A1 (cg-RX-API-DMAC7.html) |
| BR (1) | BRPI0608454A2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2602233A1 (cg-RX-API-DMAC7.html) |
| DE (1) | DE102005012873B4 (cg-RX-API-DMAC7.html) |
| IL (1) | IL185804A0 (cg-RX-API-DMAC7.html) |
| MX (1) | MX2007010837A (cg-RX-API-DMAC7.html) |
| WO (1) | WO2006099941A1 (cg-RX-API-DMAC7.html) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| CA2666193A1 (en) | 2006-08-08 | 2008-02-14 | Sanofi-Aventis | Arylaminoaryl-alkyl-substituted imidazolidine-2,4-diones, process for preparing them, medicaments comprising these compounds, and their use |
| DE102007005045B4 (de) | 2007-01-26 | 2008-12-18 | Sanofi-Aventis | Phenothiazin Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| AR072707A1 (es) | 2008-07-09 | 2010-09-15 | Sanofi Aventis | Compuestos heterociclicos, procesos para su preparacion, medicamentos que comprenden estos compuestos y el uso de los mismos |
| WO2010068601A1 (en) | 2008-12-08 | 2010-06-17 | Sanofi-Aventis | A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof |
| AU2010288523A1 (en) | 2009-08-26 | 2012-03-15 | Sanofi | Novel crystalline heteroaromatic fluoroglycoside hydrates, pharmaceuticals comprising these compounds and their use |
| WO2011107494A1 (de) | 2010-03-03 | 2011-09-09 | Sanofi | Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
| US8933024B2 (en) | 2010-06-18 | 2015-01-13 | Sanofi | Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases |
| US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
| TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
| TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
| TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
| US8809325B2 (en) | 2011-03-08 | 2014-08-19 | Sanofi | Benzyl-oxathiazine derivatives substituted with adamantane and noradamantane, medicaments containing said compounds and use thereof |
| EP2683701B1 (de) | 2011-03-08 | 2014-12-24 | Sanofi | Mit benzyl- oder heteromethylengruppen substituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| EP2683700B1 (de) | 2011-03-08 | 2015-02-18 | Sanofi | Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| US8828994B2 (en) | 2011-03-08 | 2014-09-09 | Sanofi | Di- and tri-substituted oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof |
| EP2683699B1 (de) | 2011-03-08 | 2015-06-24 | Sanofi | Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| WO2012120057A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| EP2766349B1 (de) | 2011-03-08 | 2016-06-01 | Sanofi | Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| EP2683702B1 (de) | 2011-03-08 | 2014-12-24 | Sanofi | Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| US8828995B2 (en) | 2011-03-08 | 2014-09-09 | Sanofi | Branched oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof |
| WO2013037390A1 (en) | 2011-09-12 | 2013-03-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| WO2013045413A1 (en) | 2011-09-27 | 2013-04-04 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
| CN105142621A (zh) | 2012-10-24 | 2015-12-09 | 国家健康科学研究所 | 用于预防或治疗糖尿病和促进β-细胞存活的TPL2激酶抑制剂 |
| EP3273981B1 (en) | 2015-03-24 | 2020-04-29 | INSERM - Institut National de la Santé et de la Recherche Médicale | Method and pharmaceutical composition for use in the treatment of diabetes |
| HUE066335T2 (hu) | 2018-10-05 | 2024-07-28 | Annapurna Bio Inc | Vegyületek és készítmények APJ receptor aktivitáshoz kapcsolódó állapotok kezelésére |
| WO2023107705A1 (en) | 2021-12-10 | 2023-06-15 | Incyte Corporation | Bicyclic amines as cdk12 inhibitors |
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| IL113472A0 (en) * | 1994-04-29 | 1995-07-31 | Lilly Co Eli | Non-peptidyl tachykinin receptor antogonists |
| US6025372A (en) * | 1997-04-04 | 2000-02-15 | Merck & Co., Inc. | Somatostatin agonists |
| AUPP150098A0 (en) * | 1998-01-27 | 1998-02-19 | Fujisawa Pharmaceutical Co., Ltd. | Benzamide derivatives |
| US6340681B1 (en) * | 1999-07-16 | 2002-01-22 | Pfizer Inc | 2-benzimidazolylamine compounds as ORL-1-receptor agonists |
| WO2002046168A1 (en) * | 2000-12-07 | 2002-06-13 | Astrazeneca Ab | Therapeutic benzimidazole compounds |
| WO2004011440A1 (ja) * | 2002-07-30 | 2004-02-05 | Banyu Pharmaceutical Co., Ltd. | ベンズイミダゾール誘導体を有効成分とするメラニン凝集ホルモン受容体拮抗剤 |
| WO2007069053A1 (en) * | 2005-12-14 | 2007-06-21 | Pfizer Products Inc. | Benzimidazole antagonists of the h-3 receptor |
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2005
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2006
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- 2006-03-07 WO PCT/EP2006/002056 patent/WO2006099941A1/de not_active Ceased
- 2006-03-07 BR BRPI0608454-0A patent/BRPI0608454A2/pt not_active Application Discontinuation
- 2006-03-07 AU AU2006226638A patent/AU2006226638A1/en not_active Abandoned
- 2006-03-07 JP JP2008501195A patent/JP2008533065A/ja not_active Abandoned
- 2006-03-07 EP EP06723255.3A patent/EP1863789B1/de not_active Not-in-force
- 2006-03-07 MX MX2007010837A patent/MX2007010837A/es not_active Application Discontinuation
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2007
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Also Published As
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| EP1863789B1 (de) | 2014-08-20 |
| IL185804A0 (en) | 2008-01-06 |
| AU2006226638A1 (en) | 2006-09-28 |
| WO2006099941A1 (de) | 2006-09-28 |
| BRPI0608454A2 (pt) | 2010-01-05 |
| DE102005012873A1 (de) | 2006-09-28 |
| CA2602233A1 (en) | 2006-09-28 |
| EP1863789A1 (de) | 2007-12-12 |
| WO2006099941A8 (de) | 2006-11-09 |
| US8138207B2 (en) | 2012-03-20 |
| DE102005012873B4 (de) | 2007-05-03 |
| MX2007010837A (es) | 2007-11-09 |
| US20080090869A1 (en) | 2008-04-17 |
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