JP2008530171A - 新規なジアザ二環系アリール誘導体及びそれらの医療上の使用 - Google Patents
新規なジアザ二環系アリール誘導体及びそれらの医療上の使用 Download PDFInfo
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- JP2008530171A JP2008530171A JP2007555581A JP2007555581A JP2008530171A JP 2008530171 A JP2008530171 A JP 2008530171A JP 2007555581 A JP2007555581 A JP 2007555581A JP 2007555581 A JP2007555581 A JP 2007555581A JP 2008530171 A JP2008530171 A JP 2008530171A
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Classifications
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200500229 | 2005-02-16 | ||
| US65351205P | 2005-02-17 | 2005-02-17 | |
| PCT/EP2006/050873 WO2006087305A1 (en) | 2005-02-16 | 2006-02-13 | Novel diazabicyclic aryl derivatives and their medical use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008530171A true JP2008530171A (ja) | 2008-08-07 |
| JP2008530171A5 JP2008530171A5 (enExample) | 2009-04-02 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007555581A Abandoned JP2008530171A (ja) | 2005-02-16 | 2006-02-13 | 新規なジアザ二環系アリール誘導体及びそれらの医療上の使用 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US7750011B2 (enExample) |
| EP (1) | EP1866314B1 (enExample) |
| JP (1) | JP2008530171A (enExample) |
| AT (1) | ATE481407T1 (enExample) |
| DE (1) | DE602006016926D1 (enExample) |
| WO (1) | WO2006087305A1 (enExample) |
Families Citing this family (22)
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| GB0220581D0 (en) * | 2002-09-04 | 2002-10-09 | Novartis Ag | Organic Compound |
| AR049401A1 (es) | 2004-06-18 | 2006-07-26 | Novartis Ag | Aza-biciclononanos |
| GB0415746D0 (en) | 2004-07-14 | 2004-08-18 | Novartis Ag | Organic compounds |
| GB0521508D0 (en) * | 2005-10-21 | 2005-11-30 | Novartis Ag | Organic compounds |
| GB0525673D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| GB0525672D0 (en) * | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| RS20090154A (sr) * | 2006-10-18 | 2010-10-31 | Pfizer Products Inc. | Jedinjenja biaril etra uree |
| US7994156B2 (en) * | 2007-11-30 | 2011-08-09 | Neurosearch A/S | Carboxylic acid 4-phenylazo-phenyl ester derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| JP5865397B2 (ja) | 2011-02-03 | 2016-02-17 | ルピン・リミテッドＬｕｐｉｎ Ｌｉｍｉｔｅｄ | α７ｎＡＣｈＲのモジュレータとして使用されるピロール誘導体 |
| HUE030659T2 (hu) | 2011-02-23 | 2017-05-29 | Lupin Ltd | Heteroaril származékok mint Alfa7 NACHR modulátorok |
| AU2012235779B2 (en) | 2011-03-31 | 2017-03-02 | Lupin Limited | Pyrrole derivatives as nicotinic acetylcholine receptor modulators for use in the treatment of neurodegenerative disorders such as Alzheimer's and Parkinson's disease |
| US8946432B2 (en) | 2011-07-05 | 2015-02-03 | Lupin Limited | Biaryl derivatives as nAChR modulators |
| SG11201405239WA (en) | 2012-03-06 | 2014-09-26 | Lupin Ltd | Thiazole derivatives as alpha 7 nachr modulators |
| WO2014072957A1 (en) | 2012-11-12 | 2014-05-15 | Lupin Limited | Thiazole derivatives as alpha 7 nachr modulators |
| EP2945941B1 (en) | 2013-01-16 | 2016-12-07 | Lupin Limited | Pyrrole derivatives as alpha 7 nachr modulators |
| AU2014229300A1 (en) | 2013-03-13 | 2015-06-11 | Lupin Limited | Pyrrole derivatives as alpha 7 nAChR modulators |
| TW201446243A (zh) | 2013-06-03 | 2014-12-16 | Lupin Ltd | 4-(5-(4-氯苯基)-2-(2-環丙基乙醯基)-1,4-二甲基-1氫-吡咯-3-基)苯磺醯胺作為α7尼古丁乙醯膽鹼受體調節劑 |
| AU2014282886A1 (en) | 2013-06-17 | 2015-12-17 | Lupin Limited | Pyrrole derivatives as alpha 7 nAChR modulators |
| CA3026784A1 (en) | 2016-06-07 | 2017-12-14 | Jacobio Pharmaceuticals Co., Ltd. | Heterocyclic pyrazine derivatives useful as shp2 inhibitors |
| MY200227A (en) | 2017-03-23 | 2023-12-15 | Jacobio Pharmaceuticals Co Ltd | Novel heterocyclic derivatives useful as shp2 inhibitors |
| US20210393623A1 (en) | 2018-09-26 | 2021-12-23 | Jacobio Pharmaceuticals Co., Ltd. | Novel Heterocyclic Derivatives Useful as SHP2 Inhibitors |
| CN114409669B (zh) * | 2022-01-24 | 2023-06-23 | 云南民族大学 | 一种氧杂降冰片烯环上c-5位炔基取代的斑蝥素衍生物及其制备方法与应用 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5478939A (en) * | 1994-07-20 | 1995-12-26 | American Cyanamid Company | (R,R) and (S,S) 2,5-diazabicyclo [2,2,1]heptane derivatives |
| GB9803411D0 (en) | 1998-02-18 | 1998-04-15 | Smithkline Beecham Plc | Novel compounds |
| FR2786769B1 (fr) | 1998-12-04 | 2002-10-25 | Synthelabo | Derives de 2,5-diazabicyclo[2.2.1]heptane, leur preparation et leur application en therapeutique |
| NZ512884A (en) | 1999-01-29 | 2004-03-26 | Abbott Lab | Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands |
| DK1506200T3 (da) | 2002-05-07 | 2007-04-10 | Neurosearch As | Diazabicykliske biarylderivater |
| ATE353899T1 (de) | 2002-09-30 | 2007-03-15 | Neurosearch As | Neue 1,4-diazabicycloalkanderivate, deren herstellung und verwendung |
| WO2004043960A1 (en) | 2002-11-11 | 2004-05-27 | Neurosearch A/S | 1,4-diazabicyclo (3,2,2)nonane derivatives, preparation and therapeutical use thereof |
| BRPI0413059A (pt) | 2003-07-29 | 2006-10-31 | Xenon Pharmaceuticals Inc | derivados de piridila e seu uso como agentes terapêuticos |
| BRPI0412348A (pt) * | 2003-07-30 | 2006-09-05 | Xenon Pharmaceuticals Inc | derivados de piperazina e seu uso como agentes terapêuticos |
| DE602005018020D1 (de) | 2004-02-04 | 2010-01-14 | Neurosearch As | Diazabicyclische aryl-derivate als cholinerge rezeptor-modulatoren |
-
2006
- 2006-02-13 JP JP2007555581A patent/JP2008530171A/ja not_active Abandoned
- 2006-02-13 EP EP06708215A patent/EP1866314B1/en not_active Not-in-force
- 2006-02-13 AT AT06708215T patent/ATE481407T1/de not_active IP Right Cessation
- 2006-02-13 WO PCT/EP2006/050873 patent/WO2006087305A1/en not_active Ceased
- 2006-02-13 DE DE602006016926T patent/DE602006016926D1/de active Active
- 2006-02-13 US US11/884,345 patent/US7750011B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US20080161314A1 (en) | 2008-07-03 |
| WO2006087305A1 (en) | 2006-08-24 |
| EP1866314B1 (en) | 2010-09-15 |
| EP1866314A1 (en) | 2007-12-19 |
| DE602006016926D1 (de) | 2010-10-28 |
| US7750011B2 (en) | 2010-07-06 |
| ATE481407T1 (de) | 2010-10-15 |
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