JP2008527028A5 - - Google Patents

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Publication number
JP2008527028A5
JP2008527028A5 JP2007551726A JP2007551726A JP2008527028A5 JP 2008527028 A5 JP2008527028 A5 JP 2008527028A5 JP 2007551726 A JP2007551726 A JP 2007551726A JP 2007551726 A JP2007551726 A JP 2007551726A JP 2008527028 A5 JP2008527028 A5 JP 2008527028A5
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JP
Japan
Prior art keywords
synthase
leukotriene
activating protein
mpges
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2007551726A
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English (en)
Japanese (ja)
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JP2008527028A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/GB2005/004980 external-priority patent/WO2006077365A1/en
Publication of JP2008527028A publication Critical patent/JP2008527028A/ja
Publication of JP2008527028A5 publication Critical patent/JP2008527028A5/ja
Withdrawn legal-status Critical Current

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JP2007551726A 2005-01-19 2005-12-22 炎症の治療に有用なインドール類 Withdrawn JP2008527028A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US64451905P 2005-01-19 2005-01-19
PCT/GB2005/004980 WO2006077365A1 (en) 2005-01-19 2005-12-22 Indoles useful in the treatment of inflammation

Publications (2)

Publication Number Publication Date
JP2008527028A JP2008527028A (ja) 2008-07-24
JP2008527028A5 true JP2008527028A5 (https=) 2009-02-19

Family

ID=34956617

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007551726A Withdrawn JP2008527028A (ja) 2005-01-19 2005-12-22 炎症の治療に有用なインドール類

Country Status (5)

Country Link
US (1) US20090042949A1 (https=)
EP (1) EP1838669A1 (https=)
JP (1) JP2008527028A (https=)
CA (1) CA2594773A1 (https=)
WO (1) WO2006077365A1 (https=)

Families Citing this family (29)

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US20080249091A1 (en) * 2005-01-19 2008-10-09 Benjamin Pelcman Indoles Useful in the Treatment of Inflammation
JP2008527030A (ja) * 2005-01-19 2008-07-24 バイオリポックス エービー 炎症の治療に有用なインドール類
BRPI0519774A2 (pt) * 2005-01-19 2009-02-10 Biolipox Ab composto ou um sal farmaceuticamente aceitÁvel do mesmo, formulaÇço farmacÊutica, uso de um composto ou um sal farmaceuticamente aceitÁvel do mesmo, mÉtodo de tratamento de uma doenÇa em que inibiÇço da atividade de um membro da famÍlia mapeg É desejada e/ou necessÁria, produto combinado, e, processo para a preparaÇço de um composto
EP1854011A2 (en) * 2005-02-15 2007-11-14 Koninklijke Philips Electronics N.V. Enhancing performance of a memory unit of a data processing device by separating reading and fetching functionalities
US7977359B2 (en) 2005-11-04 2011-07-12 Amira Pharmaceuticals, Inc. 5-lipdxygenase-activating protein (FLAP) inhibitors
US8399666B2 (en) 2005-11-04 2013-03-19 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein (FLAP) inhibitors
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TW200920369A (en) 2007-10-26 2009-05-16 Amira Pharmaceuticals Inc 5-lipoxygenase activating protein (flap) inhibitor
JP5791500B2 (ja) 2008-05-23 2015-10-07 パンミラ ファーマシューティカルズ，エルエルシー． ５−リポキシゲナーゼ活性化タンパク質阻害剤
US8546431B2 (en) 2008-10-01 2013-10-01 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein (FLAP) inhibitors
US20120029016A1 (en) 2008-12-30 2012-02-02 Biolipox Ab Indoles Useful in the Treatment of Inflammation
EA201200046A1 (ru) 2009-06-24 2012-08-30 Бёрингер Ингельхайм Интернациональ Гмбх Новые соединения, фармацевтическая композиция и связанные с ними способы
US8481731B2 (en) 2009-06-24 2013-07-09 Boehringer Ingelheim International Gmbh Compounds, pharmaceutical composition and methods relating thereto
JP2012211085A (ja) * 2009-08-12 2012-11-01 Kyowa Hakko Kirin Co Ltd ヘッジホッグシグナル阻害剤
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WO2012145069A2 (en) * 2011-02-24 2012-10-26 The University Of Toledo Materials and methods useful to induce cell death via methuosis
JOP20130213B1 (ar) 2012-07-17 2021-08-17 Takeda Pharmaceuticals Co معارضات لمستقبلht3-5
CA2894536C (en) 2012-12-18 2020-07-28 Vertex Pharmaceuticals Incorporated Mannose derivatives for treating bacterial infections
MX2015012472A (es) 2013-03-12 2016-02-10 Vertex Pharma Derivados de manosa para el tratamiento de infecciones bacterianas.
JP7055017B2 (ja) 2014-09-29 2022-04-15 武田薬品工業株式会社 結晶形の１－（１－メチル－１ｈ－ピラゾール－４－イル）－ｎ－（（１ｒ，５ｓ，７ｓ）－９－メチル－３－オキサ－９－アザビシクロ［３．３．１］ノナン－７－イル）－１ｈ－インドール－３－カルボキサミド
DK3240785T3 (da) 2014-12-29 2021-09-27 Us Health Småmolekylede hæmmere af laktasedehydrogenase og fremgangsmåder til brug deraf
CN107098846B (zh) * 2016-02-26 2020-10-09 中国医学科学院药物研究所 N-酰基磺酰胺类FBPase抑制剂、其制备方法、药物组合物及用途
AU2017275657B2 (en) 2016-06-02 2021-08-19 Novartis Ag Potassium channel modulators
PL3571193T3 (pl) 2017-01-23 2022-04-25 Cadent Therapeutics, Inc. Modulatory kanału potasowego
ES2812698T3 (es) 2017-09-29 2021-03-18 Probiodrug Ag Inhibidores de glutaminil ciclasa
EP3870291A1 (en) 2018-10-22 2021-09-01 Cadent Therapeutics, Inc. Crystalline forms of potassium channel modulators
KR102711104B1 (ko) 2019-08-26 2024-09-27 국제약품 주식회사 인돌 카복사미드 유도체 및 그를 포함하는 약제학적 조성물
CN119950495A (zh) * 2020-07-24 2025-05-09 上海交通大学医学院附属瑞金医院 一种干扰整合素β3/Src相互作用的化合物的用途
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