JP2008525358A5 - Ｍ３ムスカリン受容体としてのピロリジニウム誘導体 - Google Patents
Ｍ３ムスカリン受容体としてのピロリジニウム誘導体 Download PDFInfo
- Publication number
- JP2008525358A5 JP2008525358A5 JP2007547367A JP2007547367A JP2008525358A5 JP 2008525358 A5 JP2008525358 A5 JP 2008525358A5 JP 2007547367 A JP2007547367 A JP 2007547367A JP 2007547367 A JP2007547367 A JP 2007547367A JP 2008525358 A5 JP2008525358 A5 JP 2008525358A5
- Authority
- JP
- Japan
- Prior art keywords
- muscarinic receptors
- pyrrolidinium derivatives
- pyrrolidinium
- derivatives
- muscarinic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 102000014415 Muscarinic acetylcholine receptor family Human genes 0.000 title 1
- 108050003473 Muscarinic acetylcholine receptor family Proteins 0.000 title 1
- RWRDLPDLKQPQOW-UHFFFAOYSA-O pyrrolidinium Chemical class C1CC[NH2+]C1 RWRDLPDLKQPQOW-UHFFFAOYSA-O 0.000 title 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0428416.2A GB0428416D0 (en) | 2004-12-24 | 2004-12-24 | Organic compounds |
| PCT/EP2005/013896 WO2006066928A1 (en) | 2004-12-24 | 2005-12-22 | Pyrrolinidium derivatives as m3 muscarinic receptors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008525358A JP2008525358A (ja) | 2008-07-17 |
| JP2008525358A5 true JP2008525358A5 (ja) | 2009-02-12 |
Family
ID=34130966
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007547367A Pending JP2008525358A (ja) | 2004-12-24 | 2005-12-22 | Ｍ３ムスカリン受容体としてのピロリニジウム誘導体 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US8383625B2 (ja) |
| EP (1) | EP1831202B1 (ja) |
| JP (1) | JP2008525358A (ja) |
| KR (1) | KR101256242B1 (ja) |
| CN (1) | CN101087777B (ja) |
| AT (1) | ATE541839T1 (ja) |
| AU (1) | AU2005318423B2 (ja) |
| BR (1) | BRPI0519208A2 (ja) |
| CA (1) | CA2589744C (ja) |
| ES (1) | ES2377486T3 (ja) |
| GB (1) | GB0428416D0 (ja) |
| MX (1) | MX2007007720A (ja) |
| PL (1) | PL1831202T3 (ja) |
| PT (1) | PT1831202E (ja) |
| RU (1) | RU2412183C2 (ja) |
| WO (1) | WO2006066928A1 (ja) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1957451B1 (en) | 2005-11-10 | 2011-10-19 | Nicholas S. Bodor | Soft anticholinergic zwitterions |
| CA2627982C (en) | 2005-11-10 | 2013-09-10 | Nicholas S. Bodor | Soft anticholinergic esters |
| TW200825084A (en) | 2006-11-14 | 2008-06-16 | Astrazeneca Ab | New compounds 521 |
| WO2008103426A1 (en) | 2007-02-23 | 2008-08-28 | Theravance, Inc. | Quaternary ammonium diphenylmethyl compounds useful as muscarinic receptor antagonists |
| SI2197841T1 (sl) | 2007-09-07 | 2012-02-29 | Theravance Inc | Spojine, ki vsebujejo gvanidin, uporabne kot antagonisti muskarinskih receptorjev |
| JP2011506477A (ja) | 2007-12-14 | 2011-03-03 | セラヴァンス， インコーポレーテッド | ムスカリン受容体拮抗薬として有用なアミジン含有化合物 |
| EP2300464A1 (en) | 2008-05-13 | 2011-03-30 | AstraZeneca AB | Quinuclidine derivatives as muscarinic m3 receptor antagonists |
| WO2014097151A2 (en) | 2012-12-19 | 2014-06-26 | Novartis Ag | Autotaxin inhibitors |
| US9220707B2 (en) | 2013-03-15 | 2015-12-29 | Bodor Laboratories, Inc. | Method of dosing and use of soft anticholinergic esters |
| US20150259283A1 (en) | 2014-03-13 | 2015-09-17 | Brickell Biotech, Inc. | Formulation for soft anticholinergic analogs |
| US20170037030A1 (en) | 2014-04-24 | 2017-02-09 | Novartis Ag | Autotaxin inhibitors |
| CN108137612A (zh) | 2015-07-21 | 2018-06-08 | 博多尔实验仪器公司 | 软性抗胆碱能药类似物的制剂 |
| TWI767507B (zh) | 2016-07-21 | 2022-06-11 | 美商波德實驗股份有限公司 | 軟性抗膽鹼類似物之製劑 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL195520B1 (pl) * | 1996-11-11 | 2007-09-28 | Meda Pharma Gmbh & Co Kg | Enancjomerycznie czyste estry, farmaceutycznie dopuszczalna sól, sposób wytwarzania, środek leczniczy i zastosowanie enancjomerycznie czystych estrów |
| CA2415468A1 (en) | 2000-07-11 | 2003-01-10 | Yoshio Ogino | Ester derivatives |
| ES2206021B1 (es) * | 2002-04-16 | 2005-08-01 | Almirall Prodesfarma, S.A. | Nuevos derivados de pirrolidinio. |
| AR044134A1 (es) * | 2003-05-02 | 2005-08-24 | Novartis Ag | Derivados de quinuclidina, metodo de preparacion y composiciones farmaceuticas. |
| AR044851A1 (es) | 2003-06-24 | 2005-10-05 | Novartis Ag | Compuestos heterociclicos, antagonistas del receptor m3 muscarinico |
| GB0428418D0 (en) | 2004-12-24 | 2005-02-02 | Novartis Ag | Organic compounds |
| EP2227234B1 (en) * | 2007-10-15 | 2014-05-07 | Can-Fite Biopharma Ltd. | Method for inducing hepatocyte proliferation and uses thereof |
-
2004
- 2004-12-24 GB GBGB0428416.2A patent/GB0428416D0/en not_active Ceased
-
2005
- 2005-12-22 ES ES05850334T patent/ES2377486T3/es active Active
- 2005-12-22 EP EP05850334A patent/EP1831202B1/en not_active Not-in-force
- 2005-12-22 US US11/721,058 patent/US8383625B2/en not_active Expired - Fee Related
- 2005-12-22 BR BRPI0519208-0A patent/BRPI0519208A2/pt not_active IP Right Cessation
- 2005-12-22 KR KR1020077014263A patent/KR101256242B1/ko not_active IP Right Cessation
- 2005-12-22 JP JP2007547367A patent/JP2008525358A/ja active Pending
- 2005-12-22 AU AU2005318423A patent/AU2005318423B2/en not_active Ceased
- 2005-12-22 WO PCT/EP2005/013896 patent/WO2006066928A1/en active Application Filing
- 2005-12-22 PL PL05850334T patent/PL1831202T3/pl unknown
- 2005-12-22 AT AT05850334T patent/ATE541839T1/de active
- 2005-12-22 CA CA2589744A patent/CA2589744C/en not_active Expired - Fee Related
- 2005-12-22 RU RU2007128080/04A patent/RU2412183C2/ru not_active IP Right Cessation
- 2005-12-22 CN CN2005800447368A patent/CN101087777B/zh not_active Expired - Fee Related
- 2005-12-22 MX MX2007007720A patent/MX2007007720A/es active IP Right Grant
- 2005-12-22 PT PT05850334T patent/PT1831202E/pt unknown
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