JP2008519794A5 - - Google Patents

Download PDF

Info

Publication number
JP2008519794A5
JP2008519794A5 JP2007540588A JP2007540588A JP2008519794A5 JP 2008519794 A5 JP2008519794 A5 JP 2008519794A5 JP 2007540588 A JP2007540588 A JP 2007540588A JP 2007540588 A JP2007540588 A JP 2007540588A JP 2008519794 A5 JP2008519794 A5 JP 2008519794A5
Authority
JP
Japan
Prior art keywords
pyrimidine
benzo
furo
chloro
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2007540588A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008519794A (ja
Filing date
Publication date
Priority claimed from GB0424972A external-priority patent/GB0424972D0/en
Priority claimed from EP05022665A external-priority patent/EP1776982A1/en
Application filed filed Critical
Priority claimed from PCT/EP2005/012087 external-priority patent/WO2006050965A1/en
Publication of JP2008519794A publication Critical patent/JP2008519794A/ja
Publication of JP2008519794A5 publication Critical patent/JP2008519794A5/ja
Withdrawn legal-status Critical Current

Links

JP2007540588A 2004-11-11 2005-11-11 ピリミジン化合物 Withdrawn JP2008519794A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0424972A GB0424972D0 (en) 2004-11-11 2004-11-11 Pyrimidine compounds
EP05022665A EP1776982A1 (en) 2005-10-18 2005-10-18 Pyrimidine compounds as histamine modulators
PCT/EP2005/012087 WO2006050965A1 (en) 2004-11-11 2005-11-11 Pyrimidine compounds as histamine modulators

Publications (2)

Publication Number Publication Date
JP2008519794A JP2008519794A (ja) 2008-06-12
JP2008519794A5 true JP2008519794A5 (https=) 2008-12-25

Family

ID=35658998

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007540588A Withdrawn JP2008519794A (ja) 2004-11-11 2005-11-11 ピリミジン化合物

Country Status (6)

Country Link
US (1) US20080269239A1 (https=)
EP (1) EP1812113A1 (https=)
JP (1) JP2008519794A (https=)
AU (1) AU2005303893A1 (https=)
CA (1) CA2586316A1 (https=)
WO (1) WO2006050965A1 (https=)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009514969A (ja) 2005-11-09 2009-04-09 コンビナトアールエックス インコーポレーティッド 医学的状態を治療するための方法、組成物、およびキット
GB0525068D0 (en) 2005-12-08 2006-01-18 Novartis Ag Organic compounds
EP1860109A1 (en) * 2006-05-24 2007-11-28 Cellzome (UK) Ltd. Azetidine amino pyrimidine compounds for the treatment of inflammatory disorders
WO2007090854A1 (en) * 2006-02-10 2007-08-16 Cellzome (Uk) Ltd. Azetidine amino pyrimidine compounds for the treatment of inflammatory disorders
TW200815054A (en) * 2006-06-19 2008-04-01 Otsuka Pharma Co Ltd Methods of using a thiazole derivative
KR20090028819A (ko) * 2006-07-11 2009-03-19 얀센 파마슈티카 엔.브이. 히스타민 h4 수용체의 벤조푸로- 및 벤조티에노피리미딘 조절제
US8735411B2 (en) 2006-10-02 2014-05-27 Abbvie Inc. Macrocyclic benzofused pyrimidine derivatives
US7985745B2 (en) 2006-10-02 2011-07-26 Abbott Laboratories Method for pain treatment
CA2705719C (en) 2007-09-14 2016-10-11 Janssen Pharmaceutica N.V. Thieno-and furo-pyrimidine modulators of the histamine h4 receptor
PE20090978A1 (es) * 2007-10-30 2009-07-13 Palau Pharma Sa DERIVADOS DE FURO {3,2-d} PIRIMIDINA
AR069869A1 (es) * 2007-12-21 2010-02-24 Exelixis Inc Derivados de benzofuro[3,2-d]pirimidinas inhibidores de proteinquinasas,composiciones farmaceuticas que los comprenden y usos de los mismos en el tratamiento del cancer.
EP2077263A1 (en) 2008-01-02 2009-07-08 Vereniging voor christelijk hoger onderwijs, wetenschappelijk onderzoek en patiëntenzorg Quinazolines and related heterocyclic compounds and their therapeutic use
US8278313B2 (en) 2008-03-11 2012-10-02 Abbott Laboratories Macrocyclic spiro pyrimidine derivatives
WO2009115496A1 (en) * 2008-03-17 2009-09-24 Palau Pharma, S. A. Furo [3, 2-d] pyrimidine derivatives as h4 receptor antagonists
US8546410B2 (en) 2008-05-05 2013-10-01 Abbvie Inc. Heteroaryl-fused macrocyclic pyrimidine derivatives
MX2010013726A (es) 2008-06-12 2011-01-14 Janssen Pharmaceutica Nv Moduladores de diamino-piridina, pirimidina, y piridazina del receptor h4 de histamina.
EP2201982A1 (en) 2008-12-24 2010-06-30 INSERM (Institut National de la Santé et de la Recherche Médicale) Histamine H4 receptor antagonists for the treatment of vestibular disorders
US8349852B2 (en) 2009-01-13 2013-01-08 Novartis Ag Quinazolinone derivatives useful as vanilloid antagonists
AR080056A1 (es) 2010-02-01 2012-03-07 Novartis Ag Derivados de ciclohexil-amida como antagonistas de los receptores de crf
JP2013518085A (ja) 2010-02-01 2013-05-20 ノバルティス アーゲー CRF−1受容体アンタゴニストとしてのピラゾロ[5,1b]オキサゾール誘導体
JP5748777B2 (ja) 2010-02-02 2015-07-15 ノバルティス アーゲー Crf受容体アンタゴニストとしてのシクロヘキシルアミド誘導体
TW201500358A (zh) 2010-12-16 2015-01-01 赫夫門羅氏藥廠股份有限公司 三環pi3k抑制劑化合物及其使用方法
UY34094A (es) 2011-05-27 2013-01-03 Novartis Ag Derivados de la piperidina 3-espirocíclica como agonistas de receptores de la ghrelina
CA2867043A1 (en) 2012-05-03 2013-11-07 Novartis Ag L-malate salt of 2,7-diaza-spiro[4.5]dec-7-yle derivatives and crystalline forms thereof as ghrelin receptor agonists
HUE039713T2 (hu) 2012-06-08 2019-02-28 Sensorion H4 receptor inhibitorok tinnitus kezelésére
CN105103327B (zh) * 2013-03-26 2018-09-07 株式会社半导体能源研究所 发光元件、化合物、有机化合物、显示模块、照明模块、发光装置、显示装置、照明装置以及电子设备
KR102287012B1 (ko) * 2014-05-28 2021-08-09 덕산네오룩스 주식회사 유기전기 소자용 화합물, 이를 이용한 유기전기소자 및 그 전자 장치
KR20250065420A (ko) 2015-12-25 2025-05-12 가부시키가이샤 한도오따이 에네루기 켄큐쇼 화합물, 발광 소자, 표시 장치, 전자 기기, 및 조명 장치
CA3023867A1 (en) * 2016-05-09 2017-11-16 Biogaia Ab Selection of bacterial strains useful in allergy treatment
CN115275032B (zh) 2016-12-28 2025-12-23 株式会社半导体能源研究所 发光元件、有机化合物、发光装置、电子设备及照明装置
JP2019006763A (ja) 2017-06-22 2019-01-17 株式会社半導体エネルギー研究所 有機化合物、発光素子、発光装置、電子機器、および照明装置
CA3125625A1 (en) * 2019-01-04 2020-07-09 Bellbrook Labs, Llc Inhibitors of cgas activity as therapeutic agents
US20240059712A1 (en) * 2022-03-09 2024-02-22 Risen (Suzhou) Pharma Tech Co., Ltd. Bifunctional compounds and pharmaceutical uses thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3755583A (en) * 1970-06-05 1973-08-28 Chas0!nhx
JPH06220059A (ja) * 1993-01-28 1994-08-09 Tanabe Seiyaku Co Ltd 縮合ピリミジン誘導体及びその製法
EP1373204B1 (en) * 2001-03-09 2016-10-26 Janssen Pharmaceuticals, Inc. Heterocyclic compounds
EP1543011B1 (en) * 2002-09-06 2006-05-03 Janssen Pharmaceutica N.V. Thienopyrrolyl and furanopyrrolyl compounds and their use as histamine h4 receptor ligands
JP4845736B2 (ja) * 2003-10-14 2011-12-28 アリゾナ ボード オブ リージェンツ オン ビハーフ ザ ユニバーシティー オブ アリゾナ プロテインキナーゼ阻害剤

Similar Documents

Publication Publication Date Title
JP2008519794A5 (https=)
HRP20201539T1 (hr) Pozitivni alosterni modulatori muskarinskog m1 receptora
JP2005508932A5 (https=)
US20120053168A1 (en) Fused benzoazepines as neuronal nicotinic acetylcholine receptor ligands
HRP20151250T1 (hr) Derivati izoksazolo-piridina
JP2013515729A5 (https=)
JP2010523556A5 (https=)
CN106573006A (zh) 作为药物的rip1激酶抑制剂杂环酰胺
JP2011521963A5 (https=)
HRP20161708T1 (hr) Supstituirani 4-fenil-piridini za terapiju bolesti povezanih sa nk-1 receptorom
JP2014505735A5 (https=)
JP2011500621A5 (https=)
JP2009529047A5 (https=)
JP2005516067A5 (https=)
EA201401150A1 (ru) Аминоиндолилзамещенные имидазолпиримидины и их применение в качестве лекарственных средств
RS52526B2 (sr) Derivati oksadiazola i njihovo korišćenje kao potencijatora metabotropnih glutamatnih receptora-842
HRP20140599T1 (hr) Derivati kiinazolin-4(3h)-ona koji se koriste kao inhibitori pi3 kinaze
JP2009510044A5 (https=)
JP2015522018A5 (https=)
JP2016503785A5 (https=)
JP2015512888A5 (https=)
JP2016028076A5 (https=)
JP2019505529A5 (https=)
JP2017526724A5 (https=)
JP2013507426A5 (https=)