JP2008518895A - 低用量のエストラジオールを含む経口固形製剤 - Google Patents
低用量のエストラジオールを含む経口固形製剤 Download PDFInfo
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- JP2008518895A JP2008518895A JP2007538360A JP2007538360A JP2008518895A JP 2008518895 A JP2008518895 A JP 2008518895A JP 2007538360 A JP2007538360 A JP 2007538360A JP 2007538360 A JP2007538360 A JP 2007538360A JP 2008518895 A JP2008518895 A JP 2008518895A
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- Prior art keywords
- estradiol
- formulation
- pharmaceutically acceptable
- hydrate
- salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Physical Education & Sports Medicine (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Endocrinology (AREA)
- Pain & Pain Management (AREA)
- Diabetes (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychiatry (AREA)
- Reproductive Health (AREA)
- Otolaryngology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04078014 | 2004-11-02 | ||
| PCT/EP2005/011726 WO2006048261A2 (en) | 2004-11-02 | 2005-11-01 | Oral solid dosage forms containing a low dose of estradiol |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008518895A true JP2008518895A (ja) | 2008-06-05 |
| JP2008518895A5 JP2008518895A5 (OSRAM) | 2008-12-25 |
Family
ID=34928627
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007538360A Pending JP2008518895A (ja) | 2004-11-02 | 2005-11-01 | 低用量のエストラジオールを含む経口固形製剤 |
Country Status (21)
| Country | Link |
|---|---|
| EP (1) | EP1814526A2 (OSRAM) |
| JP (1) | JP2008518895A (OSRAM) |
| KR (1) | KR20070085558A (OSRAM) |
| CN (1) | CN101094656A (OSRAM) |
| AR (1) | AR053650A1 (OSRAM) |
| AU (1) | AU2005300658A1 (OSRAM) |
| BR (1) | BRPI0517940A (OSRAM) |
| CA (1) | CA2585095A1 (OSRAM) |
| CR (1) | CR9112A (OSRAM) |
| CU (1) | CU20070094A7 (OSRAM) |
| EA (1) | EA013262B1 (OSRAM) |
| GT (1) | GT200500315A (OSRAM) |
| IL (1) | IL182635A0 (OSRAM) |
| MX (1) | MX2007005281A (OSRAM) |
| NO (1) | NO20072704L (OSRAM) |
| PA (1) | PA8651401A1 (OSRAM) |
| PE (1) | PE20061126A1 (OSRAM) |
| TW (1) | TW200621312A (OSRAM) |
| UY (1) | UY29185A1 (OSRAM) |
| WO (1) | WO2006048261A2 (OSRAM) |
| ZA (1) | ZA200705012B (OSRAM) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2024000555A (ja) * | 2022-06-21 | 2024-01-09 | 東ソー株式会社 | 紫外線抑制下でのエストラジオール測定試薬の製造方法 |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8022053B2 (en) | 2004-11-02 | 2011-09-20 | Bayer Schering Pharma Aktiengesellschaft | Oral solid dosage forms containing a low dose of estradiol |
| KR20080047959A (ko) * | 2006-11-27 | 2008-05-30 | 주식회사 엠디바이오알파 | 비만, 당뇨, 대사성 질환, 퇴행성 질환 및 미토콘드리아이상 질환의 치료 또는 예방을 위한 나프토퀴논계 약제조성물 |
| DE102009007771B4 (de) | 2009-02-05 | 2012-02-16 | Bayer Schering Pharma Aktiengesellschaft | Bukkales Applikationssystem, 17α-Estradiol enthaltend |
| ES2533584T3 (es) | 2010-04-15 | 2015-04-13 | Bayer Intellectual Property Gmbh | Formas de dosificación oral sólidas de dosis baja para TSH |
| MX356702B (es) | 2010-04-15 | 2018-06-11 | Bayer Ip Gmbh | Formas de dosificación sólidas orales con dosis muy bajas para la hrt. |
| CN112516149B (zh) * | 2020-07-21 | 2023-07-18 | 南方医科大学 | 苯甲酸雌二醇或其药物可接受盐在制备抗冠状病毒的药物中的应用 |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002509524A (ja) * | 1996-10-08 | 2002-03-26 | ラボラトアール、テラメックス | エストロゲン化合物とプロゲステロン様化合物よりなるホルモン組成物 |
| JP2003048836A (ja) * | 2001-07-10 | 2003-02-21 | Medical College Of Hampton Roads | 効能を保持し無月経を引き起こす超低用量の経口避妊薬 |
| JP2004512369A (ja) * | 2000-10-30 | 2004-04-22 | ユニバーシティ・オブ・チューリッヒ | 尿失禁の治療のためのｇｎｒｈアナログ |
| JP2004155779A (ja) * | 2002-10-16 | 2004-06-03 | Taisho Pharmaceut Co Ltd | 更年期症の予防・治療用経口組成物 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL125069C (OSRAM) * | 1963-12-24 | |||
| US4755386A (en) * | 1986-01-22 | 1988-07-05 | Schering Corporation | Buccal formulation |
| US5073374A (en) * | 1988-11-30 | 1991-12-17 | Schering Corporation | Fast dissolving buccal tablet |
| FR2739558B1 (fr) * | 1995-10-05 | 1997-11-28 | Innothera Lab Sa | Forme galenique unitaire pour hormonotherapie locale de la secheresse vaginale |
| US6326366B1 (en) * | 2000-08-22 | 2001-12-04 | Protein Technologies International | Hormone replacement therapy |
| EP1343508B1 (en) * | 2000-12-15 | 2011-11-09 | Novo Nordisk Femcare AG | Use of an oestrogen in the manufacture of a composition containing oestrogen for the treatment of atrophic vaginitis |
| FR2823976A1 (fr) * | 2001-04-25 | 2002-10-31 | Theramex | Nouvelle composition hormonale et son utilisation |
| US6962908B2 (en) * | 2001-12-21 | 2005-11-08 | Warner Chilcott Company Inc. | Oral pharmaceutical products containing 17 β-estradiol-3-lower alkanoate, method of administering the same and process of preparation |
-
2005
- 2005-10-31 GT GT200500315A patent/GT200500315A/es unknown
- 2005-10-31 UY UY29185A patent/UY29185A1/es not_active Application Discontinuation
- 2005-11-01 EP EP05800512A patent/EP1814526A2/en not_active Withdrawn
- 2005-11-01 CN CNA200580045694XA patent/CN101094656A/zh active Pending
- 2005-11-01 JP JP2007538360A patent/JP2008518895A/ja active Pending
- 2005-11-01 MX MX2007005281A patent/MX2007005281A/es not_active Application Discontinuation
- 2005-11-01 BR BRPI0517940-8A patent/BRPI0517940A/pt not_active IP Right Cessation
- 2005-11-01 CA CA002585095A patent/CA2585095A1/en not_active Abandoned
- 2005-11-01 AU AU2005300658A patent/AU2005300658A1/en not_active Abandoned
- 2005-11-01 TW TW094138264A patent/TW200621312A/zh unknown
- 2005-11-01 EA EA200700979A patent/EA013262B1/ru not_active IP Right Cessation
- 2005-11-01 WO PCT/EP2005/011726 patent/WO2006048261A2/en not_active Ceased
- 2005-11-01 KR KR1020077012174A patent/KR20070085558A/ko not_active Ceased
- 2005-11-02 PA PA20058651401A patent/PA8651401A1/es unknown
- 2005-11-02 PE PE2005001279A patent/PE20061126A1/es not_active Application Discontinuation
- 2005-11-02 AR ARP050104580A patent/AR053650A1/es unknown
-
2007
- 2007-04-18 IL IL182635A patent/IL182635A0/en unknown
- 2007-04-30 CU CU20070094A patent/CU20070094A7/es unknown
- 2007-05-09 CR CR9112A patent/CR9112A/es not_active Application Discontinuation
- 2007-05-29 NO NO20072704A patent/NO20072704L/no not_active Application Discontinuation
- 2007-06-01 ZA ZA200705012A patent/ZA200705012B/xx unknown
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002509524A (ja) * | 1996-10-08 | 2002-03-26 | ラボラトアール、テラメックス | エストロゲン化合物とプロゲステロン様化合物よりなるホルモン組成物 |
| JP2004512369A (ja) * | 2000-10-30 | 2004-04-22 | ユニバーシティ・オブ・チューリッヒ | 尿失禁の治療のためのｇｎｒｈアナログ |
| JP2003048836A (ja) * | 2001-07-10 | 2003-02-21 | Medical College Of Hampton Roads | 効能を保持し無月経を引き起こす超低用量の経口避妊薬 |
| JP2004155779A (ja) * | 2002-10-16 | 2004-06-03 | Taisho Pharmaceut Co Ltd | 更年期症の予防・治療用経口組成物 |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2024000555A (ja) * | 2022-06-21 | 2024-01-09 | 東ソー株式会社 | 紫外線抑制下でのエストラジオール測定試薬の製造方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| PA8651401A1 (es) | 2006-12-07 |
| EA200700979A1 (ru) | 2007-10-26 |
| MX2007005281A (es) | 2008-03-11 |
| EP1814526A2 (en) | 2007-08-08 |
| AU2005300658A1 (en) | 2006-05-11 |
| IL182635A0 (en) | 2007-07-24 |
| CN101094656A (zh) | 2007-12-26 |
| WO2006048261A3 (en) | 2006-09-21 |
| NO20072704L (no) | 2007-05-29 |
| CU20070094A7 (es) | 2009-09-08 |
| ZA200705012B (en) | 2008-10-29 |
| TW200621312A (en) | 2006-07-01 |
| WO2006048261A2 (en) | 2006-05-11 |
| GT200500315A (es) | 2006-06-06 |
| PE20061126A1 (es) | 2006-11-11 |
| BRPI0517940A (pt) | 2008-10-21 |
| KR20070085558A (ko) | 2007-08-27 |
| CR9112A (es) | 2007-11-23 |
| CA2585095A1 (en) | 2006-05-11 |
| AR053650A1 (es) | 2007-05-16 |
| EA013262B1 (ru) | 2010-04-30 |
| UY29185A1 (es) | 2006-05-31 |
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