JP2008247753A - ４−アミノ−５−クロロ−２−エトキシ−ｎ−［［４−（４−フルオロベンジル）−２−モルホリニル］メチル］ベンズアミドの製造方法 - Google Patents

４−アミノ−５−クロロ−２−エトキシ−ｎ−［［４−（４−フルオロベンジル）−２−モルホリニル］メチル］ベンズアミドの製造方法 Download PDF

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Publication number
JP2008247753A
JP2008247753A JP2007087739A JP2007087739A JP2008247753A JP 2008247753 A JP2008247753 A JP 2008247753A JP 2007087739 A JP2007087739 A JP 2007087739A JP 2007087739 A JP2007087739 A JP 2007087739A JP 2008247753 A JP2008247753 A JP 2008247753A
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Japan
Prior art keywords
chloro
amino
fluorobenzyl
compound
acid
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JP2007087739A
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Japanese (ja)
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JP2008247753A5 (https=
Inventor
Tsutomu Ishikura
勉 石倉
Takayuki Hirose
隆幸 廣▲瀬▼
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Sumitomo Pharma Co Ltd
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Sumitomo Dainippon Pharma Co Ltd
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Priority to JP2007087739A priority Critical patent/JP2008247753A/ja
Publication of JP2008247753A publication Critical patent/JP2008247753A/ja
Publication of JP2008247753A5 publication Critical patent/JP2008247753A5/ja
Pending legal-status Critical Current

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  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
JP2007087739A 2007-03-29 2007-03-29 ４−アミノ−５−クロロ−２−エトキシ−ｎ−［［４−（４−フルオロベンジル）−２−モルホリニル］メチル］ベンズアミドの製造方法 Pending JP2008247753A (ja)

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JP2007087739A JP2008247753A (ja) 2007-03-29 2007-03-29 ４−アミノ−５−クロロ−２−エトキシ−ｎ−［［４−（４−フルオロベンジル）−２−モルホリニル］メチル］ベンズアミドの製造方法

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JP2007087739A JP2008247753A (ja) 2007-03-29 2007-03-29 ４−アミノ−５−クロロ−２−エトキシ−ｎ−［［４−（４−フルオロベンジル）−２−モルホリニル］メチル］ベンズアミドの製造方法

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JP2008247753A true JP2008247753A (ja) 2008-10-16
JP2008247753A5 JP2008247753A5 (https=) 2009-08-20

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Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100953527B1 (ko) * 2009-05-13 2010-04-21 주식회사 파마코스텍 모사프리드의 신규 제조방법
JP2011068611A (ja) * 2009-09-28 2011-04-07 Tokuyama Corp ４−アミノ−５−クロロ−２−エトキシ−ｎ−〔［４−（４−フルオロベンジル）−２−モルホリニル］メチル〕ベンズアミドの精製方法
WO2011107903A1 (en) 2010-03-04 2011-09-09 Ranbaxy Laboratories Limited Highly pure mosapride citrate dihydrate and processes for its preparation
KR101123281B1 (ko) * 2008-10-17 2012-03-19 주식회사 엘지생명과학 치환된 벤즈아미드 유도체 및 그의 약제학상 허용되는 염의제조방법
JP2012072070A (ja) * 2010-09-28 2012-04-12 Tokuyama Corp ４−アミノ−５−クロロ−２−エトキシ−ｎ−〔［４−（４−フルオロベンジル）−２−モルホリニル］メチル〕ベンズアミドクエン酸塩２水和物の製造方法

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH08268988A (ja) * 1995-03-31 1996-10-15 Dai Ichi Seiyaku Co Ltd アミノベンズアミド化合物とその製法
WO2003106440A2 (en) * 2002-06-13 2003-12-24 Richter Gedeon Vegyészeti Gyár Rt. Process for the synthesis of a benzamide derivative

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH08268988A (ja) * 1995-03-31 1996-10-15 Dai Ichi Seiyaku Co Ltd アミノベンズアミド化合物とその製法
WO2003106440A2 (en) * 2002-06-13 2003-12-24 Richter Gedeon Vegyészeti Gyár Rt. Process for the synthesis of a benzamide derivative

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101123281B1 (ko) * 2008-10-17 2012-03-19 주식회사 엘지생명과학 치환된 벤즈아미드 유도체 및 그의 약제학상 허용되는 염의제조방법
KR100953527B1 (ko) * 2009-05-13 2010-04-21 주식회사 파마코스텍 모사프리드의 신규 제조방법
JP2011068611A (ja) * 2009-09-28 2011-04-07 Tokuyama Corp ４−アミノ−５−クロロ−２−エトキシ−ｎ−〔［４−（４−フルオロベンジル）−２−モルホリニル］メチル〕ベンズアミドの精製方法
WO2011107903A1 (en) 2010-03-04 2011-09-09 Ranbaxy Laboratories Limited Highly pure mosapride citrate dihydrate and processes for its preparation
JP2012072070A (ja) * 2010-09-28 2012-04-12 Tokuyama Corp ４−アミノ−５−クロロ−２−エトキシ−ｎ−〔［４−（４−フルオロベンジル）−２−モルホリニル］メチル〕ベンズアミドクエン酸塩２水和物の製造方法

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