JP2007538027A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2007538027A5 JP2007538027A5 JP2007517048A JP2007517048A JP2007538027A5 JP 2007538027 A5 JP2007538027 A5 JP 2007538027A5 JP 2007517048 A JP2007517048 A JP 2007517048A JP 2007517048 A JP2007517048 A JP 2007517048A JP 2007538027 A5 JP2007538027 A5 JP 2007538027A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- substituted
- unsubstituted
- alkyl
- groups
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 125000004435 hydrogen atoms Chemical group [H]* 0.000 claims 5
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 claims 3
- 125000003118 aryl group Chemical group 0.000 claims 3
- 125000002619 bicyclic group Chemical group 0.000 claims 3
- 125000005843 halogen group Chemical group 0.000 claims 3
- 125000002560 nitrile group Chemical group 0.000 claims 3
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 3
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 2
- 125000002950 monocyclic group Chemical group 0.000 claims 2
- 125000004469 siloxy group Chemical group [SiH3]O* 0.000 claims 2
- 150000003431 steroids Chemical class 0.000 claims 2
- PROQIPRRNZUXQM-ZXXIGWHRSA-N Estriol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@H]([C@H](O)C4)O)[C@@H]4[C@@H]3CCC2=C1 PROQIPRRNZUXQM-ZXXIGWHRSA-N 0.000 claims 1
- 229960001348 Estriol Drugs 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- 239000000651 prodrug Substances 0.000 claims 1
- 229940002612 prodrugs Drugs 0.000 claims 1
- 150000003839 salts Chemical class 0.000 claims 1
- 239000011780 sodium chloride Substances 0.000 claims 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims 1
- 0 CC(CC(O)=O)c1c(*)c(*)c(*)c(*)c1* Chemical compound CC(CC(O)=O)c1c(*)c(*)c(*)c(*)c1* 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004025985A DE102004025985A1 (de) | 2004-05-21 | 2004-05-21 | Estriol- und Estetrol-Prodrugs |
| PCT/EP2005/005258 WO2005113576A1 (de) | 2004-05-21 | 2005-05-10 | Aminosulfonyl- oder aminosulfonylamino-substituierte phenyl-ester als estriol-und estetrol-prodrugs |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2007538027A JP2007538027A (ja) | 2007-12-27 |
| JP2007538027A5 true JP2007538027A5 (ru) | 2008-06-26 |
Family
ID=34969311
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007517048A Pending JP2007538027A (ja) | 2004-05-21 | 2005-05-10 | エストリオール及びエステトロールプロドラッグ類 |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP1747231A1 (ru) |
| JP (1) | JP2007538027A (ru) |
| AR (1) | AR049108A1 (ru) |
| DE (1) | DE102004025985A1 (ru) |
| GT (1) | GT200500120A (ru) |
| PA (1) | PA8633801A1 (ru) |
| PE (1) | PE20060314A1 (ru) |
| SV (1) | SV2006002122A (ru) |
| TW (1) | TW200612962A (ru) |
| UY (1) | UY28910A1 (ru) |
| WO (1) | WO2005113576A1 (ru) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10027887A1 (de) | 2000-05-31 | 2001-12-13 | Jenapharm Gmbh | Verbindungen mit einer Sulfonamidgruppe und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen |
| US7534780B2 (en) | 2004-05-21 | 2009-05-19 | Bayer Schering Pharma Aktiengesellschaft | Estradiol prodrugs |
| DE102004025966A1 (de) * | 2004-05-21 | 2005-12-15 | Schering Ag | Estradiol-Prodrugs |
| DE102005057224A1 (de) * | 2005-11-29 | 2007-05-31 | Bayer Schering Pharma Ag | Prodrugs ERß-selektiver Substanzen, Verfahren zu deren Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen |
| DE102005057408A1 (de) * | 2005-11-30 | 2007-05-31 | Bayer Schering Pharma Ag | Sulfamoylsulfonat-Prodrugs |
| CN100396693C (zh) * | 2006-11-08 | 2008-06-25 | 浙江大学 | 1,4-孕二烯-16β-甲基-17α,21-二羟基物的制备方法 |
| CN102079771B (zh) * | 2010-12-10 | 2012-10-03 | 郑州大学 | 具有抗肿瘤活性的雌甾氨基酸酯化合物及其合成方法 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1238739A (fr) * | 1958-08-04 | 1960-08-19 | Chimiotherapie Lab Franc | Procédé de préparation de dérivés hydrosolubles de testostérone |
| FR8290M (ru) * | 1968-12-31 | 1970-11-09 | Rech Chimiques Et Ind Mar Lab | |
| US5001234A (en) * | 1987-04-16 | 1991-03-19 | The Upjohn Company | Cyclic hydrocarbons with an aminoalkyl sidechain |
| US5116828A (en) * | 1989-10-26 | 1992-05-26 | Nippon Zoki Pharmaceutical Co., Ltd. | Pharmaceutical composition for treatment of osteoporosis |
| US5571933A (en) * | 1994-11-17 | 1996-11-05 | Duquesne University Of The Holy Ghost | Derivatives of estra 1,3,5(10)triene-17-one, 3-amino compounds and their use |
| DE19712488A1 (de) * | 1997-03-25 | 1998-10-01 | Knoell Hans Forschung Ev | Steroidsulfamate, Verfahren zu ihrer Herstellung und Anwendung derselben |
| EP1284272A4 (en) * | 2000-04-24 | 2003-09-10 | Kyowa Hakko Kogyo Kk | Estra-1,3,5 (10) -triene |
| DE10027887A1 (de) * | 2000-05-31 | 2001-12-13 | Jenapharm Gmbh | Verbindungen mit einer Sulfonamidgruppe und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen |
| GB0015876D0 (en) * | 2000-06-28 | 2000-08-23 | Novartis Ag | Organic compounds |
| GB0316290D0 (en) * | 2003-07-11 | 2003-08-13 | Glaxo Group Ltd | Novel compounds |
| TWI331154B (en) * | 2003-11-12 | 2010-10-01 | Solvay Pharm Gmbh | Novel 17-hydroxysteroid dehydrogenase type i inhibitors |
| DE102004025966A1 (de) * | 2004-05-21 | 2005-12-15 | Schering Ag | Estradiol-Prodrugs |
-
2004
- 2004-05-21 DE DE102004025985A patent/DE102004025985A1/de not_active Ceased
-
2005
- 2005-05-10 EP EP05747926A patent/EP1747231A1/de not_active Withdrawn
- 2005-05-10 WO PCT/EP2005/005258 patent/WO2005113576A1/de active Application Filing
- 2005-05-10 JP JP2007517048A patent/JP2007538027A/ja active Pending
- 2005-05-19 UY UY28910A patent/UY28910A1/es not_active Application Discontinuation
- 2005-05-20 AR ARP050102085A patent/AR049108A1/es unknown
- 2005-05-20 PE PE2005000555A patent/PE20060314A1/es not_active Application Discontinuation
- 2005-05-20 PA PA20058633801A patent/PA8633801A1/es unknown
- 2005-05-20 GT GT200500120A patent/GT200500120A/es unknown
- 2005-05-20 TW TW094116505A patent/TW200612962A/zh unknown
- 2005-05-23 SV SV2005002122A patent/SV2006002122A/es not_active Application Discontinuation
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2007538027A5 (ru) | ||
| JP2007538025A5 (ru) | ||
| JP2004131511A5 (ru) | ||
| JP2005511536A5 (ru) | ||
| JP2005533804A5 (ru) | ||
| JP2007523139A5 (ru) | ||
| JP2002542342A5 (ru) | ||
| RS51044B (sr) | 2-(piridin-2-ilamino)-pirido(2,3-d)pirimidin-7-oni | |
| JP2009511649A5 (ru) | ||
| JP2009515872A5 (ru) | ||
| EP1591832A3 (en) | Photosensitive composition, compound used in the same, and patterning method using the same | |
| RS20050182A (en) | Derivatives of dioxane-2-alkyl carbamates,preparation method thereof and application of same in therapeutics | |
| TW574626B (en) | Positive resist composition | |
| JP2008538381A5 (ru) | ||
| JP2010525122A5 (ru) | ||
| JP2004533444A5 (ru) | ||
| JP2008521811A5 (ru) | ||
| EP1849836A3 (en) | Compound having polymethine-chain structure, image forming material, planographic printing plate precursor, and image forming method using the same, method of making planographic printing plate, and planographic printing method | |
| EA200500240A1 (ru) | Новый способ синтеза соединений 1,3,4,5-тетрагидро-2h-3-бензазепин-2-она и применение при синтезе ивабрадина и его солей присоединения с фармацевтически приемлемой кислотой | |
| JP2004529953A5 (ru) | ||
| JP2005537219A5 (ru) | ||
| JP2009184932A5 (ru) | ||
| JP2004531479A5 (ru) | ||
| JP2004502755A5 (ru) | ||
| JP2004529172A5 (ru) |