JP2007509184A - 尿失禁の処置におけるニューロキニンアンタゴニストの使用 - Google Patents
尿失禁の処置におけるニューロキニンアンタゴニストの使用 Download PDFInfo
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- JP2007509184A JP2007509184A JP2006537162A JP2006537162A JP2007509184A JP 2007509184 A JP2007509184 A JP 2007509184A JP 2006537162 A JP2006537162 A JP 2006537162A JP 2006537162 A JP2006537162 A JP 2006537162A JP 2007509184 A JP2007509184 A JP 2007509184A
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- Prior art keywords
- phenyl
- hydrogen
- methyl
- formula
- alkyl
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Landscapes
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- Veterinary Medicine (AREA)
- Public Health (AREA)
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- Biomedical Technology (AREA)
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- Other In-Based Heterocyclic Compounds (AREA)
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| US51479103P | 2003-10-27 | 2003-10-27 | |
| PCT/EP2004/012081 WO2005039563A2 (en) | 2003-10-27 | 2004-10-26 | Use of neurokinin antagonists in the treatment of urinary incontinence |
Publications (2)
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| JP2007509184A true JP2007509184A (ja) | 2007-04-12 |
| JP2007509184A5 JP2007509184A5 (enExample) | 2007-12-06 |
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| EP (2) | EP1686985A2 (enExample) |
| JP (1) | JP2007509184A (enExample) |
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| CA (1) | CA2543552A1 (enExample) |
| MX (1) | MXPA06004688A (enExample) |
| WO (1) | WO2005039563A2 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2010513356A (ja) * | 2006-12-22 | 2010-04-30 | ノバルティス アーゲー | ニューロキニンアンタゴニストを含む製剤 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2001503387A (ja) * | 1996-08-22 | 2001-03-13 | ノバルティス アクチエンゲゼルシャフト | Ｎｋ１およびｎｋ２アンタゴニストとしてのアシルアミノアルケニレン―アミド誘導体 |
| WO2002051440A1 (en) * | 2000-12-22 | 2002-07-04 | Takeda Chemical Industries, Ltd. | Combination drugs |
| WO2003066062A1 (en) * | 2002-02-08 | 2003-08-14 | Novartis Ag | Use of acylaminoalkenylene-amide derivatives in functional motility disorders of the viscera |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0593559A1 (en) * | 1991-07-05 | 1994-04-27 | MERCK SHARP & DOHME LTD. | Aromatic compounds, pharmaceutical compositions containing them and their use in therapy |
| FR2700472B1 (fr) * | 1993-01-19 | 1995-02-17 | Rhone Poulenc Rorer Sa | Association synergisante ayant un effet antagoniste des récepteurs NK1 et NK2. |
| GB0015246D0 (en) * | 2000-06-22 | 2000-08-16 | Astrazeneca Ab | Method for the treatment of urinary incontinence |
| US6664253B2 (en) * | 2000-10-17 | 2003-12-16 | Boehringer Ingelheim Pharma Kg | Neurokinin antagonists |
| KR20030081520A (ko) | 2001-03-14 | 2003-10-17 | 오노 야꾸힝 고교 가부시키가이샤 | Ｅｐ１ 안타고니스트를 유효 성분으로서 함유하는 울병의치료제 |
| WO2003062245A1 (en) * | 2002-01-18 | 2003-07-31 | Kyorin Pharmaceutical Co., Ltd. | Fused bicyclic pyrimidine derivatives |
| WO2003080626A1 (en) * | 2002-03-26 | 2003-10-02 | Kyorin Pharmaceutical Co., Ltd. | Fused bicyclic pyridine derivative as tachykinin receptor antagonist |
| DE60315626T2 (de) * | 2002-03-26 | 2008-06-05 | Kyorin Pharmaceutical Co., Ltd. | Kondensierte bicyclische pyrimidinderivate |
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2004
- 2004-10-26 MX MXPA06004688A patent/MXPA06004688A/es active IP Right Grant
- 2004-10-26 US US10/576,052 patent/US7776851B2/en not_active Expired - Fee Related
- 2004-10-26 CN CNA2004800316761A patent/CN1874766A/zh active Pending
- 2004-10-26 BR BRPI0415923-3A patent/BRPI0415923A/pt not_active IP Right Cessation
- 2004-10-26 JP JP2006537162A patent/JP2007509184A/ja active Pending
- 2004-10-26 EP EP04790864A patent/EP1686985A2/en not_active Ceased
- 2004-10-26 EP EP09013092A patent/EP2158910A1/en not_active Withdrawn
- 2004-10-26 WO PCT/EP2004/012081 patent/WO2005039563A2/en not_active Ceased
- 2004-10-26 AU AU2004283038A patent/AU2004283038B9/en not_active Ceased
- 2004-10-26 CA CA002543552A patent/CA2543552A1/en not_active Abandoned
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2001503387A (ja) * | 1996-08-22 | 2001-03-13 | ノバルティス アクチエンゲゼルシャフト | Ｎｋ１およびｎｋ２アンタゴニストとしてのアシルアミノアルケニレン―アミド誘導体 |
| WO2002051440A1 (en) * | 2000-12-22 | 2002-07-04 | Takeda Chemical Industries, Ltd. | Combination drugs |
| WO2003066062A1 (en) * | 2002-02-08 | 2003-08-14 | Novartis Ag | Use of acylaminoalkenylene-amide derivatives in functional motility disorders of the viscera |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2010513356A (ja) * | 2006-12-22 | 2010-04-30 | ノバルティス アーゲー | ニューロキニンアンタゴニストを含む製剤 |
Also Published As
| Publication number | Publication date |
|---|---|
| US7776851B2 (en) | 2010-08-17 |
| WO2005039563A3 (en) | 2005-06-30 |
| BRPI0415923A (pt) | 2006-12-26 |
| AU2004283038B2 (en) | 2008-01-31 |
| WO2005039563A2 (en) | 2005-05-06 |
| MXPA06004688A (es) | 2006-07-05 |
| US20070149504A1 (en) | 2007-06-28 |
| EP1686985A2 (en) | 2006-08-09 |
| AU2004283038A1 (en) | 2005-05-06 |
| CN1874766A (zh) | 2006-12-06 |
| AU2004283038B9 (en) | 2008-04-24 |
| EP2158910A1 (en) | 2010-03-03 |
| CA2543552A1 (en) | 2005-05-06 |
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