JP2007509055A - ［２−（８，９−ジオキソ−２，６−ジアザビシクロ［５．２．０］ノナ−１（７）−エン−２−イル）アルキル］ホスホン酸および誘導体の経口投与 - Google Patents
［２−（８，９−ジオキソ−２，６−ジアザビシクロ［５．２．０］ノナ−１（７）−エン−２−イル）アルキル］ホスホン酸および誘導体の経口投与 Download PDFInfo
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- JP2007509055A JP2007509055A JP2006535354A JP2006535354A JP2007509055A JP 2007509055 A JP2007509055 A JP 2007509055A JP 2006535354 A JP2006535354 A JP 2006535354A JP 2006535354 A JP2006535354 A JP 2006535354A JP 2007509055 A JP2007509055 A JP 2007509055A
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Public Health (AREA)
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- Animal Behavior & Ethology (AREA)
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- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Addiction (AREA)
- Psychology (AREA)
- Ophthalmology & Optometry (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
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- Orthopedic Medicine & Surgery (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US51156003P | 2003-10-15 | 2003-10-15 | |
| US10/961,871 US20050142192A1 (en) | 2003-10-15 | 2004-10-08 | Oral administration of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)alkyl] phosphonic acid and derivatives |
| PCT/US2004/034113 WO2005037287A1 (en) | 2003-10-15 | 2004-10-14 | Oral administration of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7) en-2-yl)alkyl]phosphonic acid and derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2007509055A true JP2007509055A (ja) | 2007-04-12 |
| JP2007509055A5 JP2007509055A5 (https=) | 2007-12-06 |
Family
ID=34704145
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006535354A Pending JP2007509055A (ja) | 2003-10-15 | 2004-10-14 | ［２−（８，９−ジオキソ−２，６−ジアザビシクロ［５．２．０］ノナ−１（７）−エン−２−イル）アルキル］ホスホン酸および誘導体の経口投与 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20050142192A1 (https=) |
| EP (1) | EP1682151A1 (https=) |
| JP (1) | JP2007509055A (https=) |
| KR (1) | KR20070029114A (https=) |
| AU (1) | AU2004281806A1 (https=) |
| BR (1) | BRPI0415432A (https=) |
| CA (1) | CA2541402A1 (https=) |
| CO (1) | CO5690561A2 (https=) |
| MX (1) | MXPA06003982A (https=) |
| PA (1) | PA8614901A1 (https=) |
| PE (1) | PE20050480A1 (https=) |
| TW (1) | TW200528113A (https=) |
| WO (1) | WO2005037287A1 (https=) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2006523694A (ja) * | 2003-04-09 | 2006-10-19 | ワイス | ［２−（８，９−ジオキソ−２，６−ジアザビシクロ［５．２．０］ノナ−１（７）−エン−２−イル）アルキル］ホスホン酸の誘導体およびｎ−メチル−ｄ−アスパルテート（ｎｍｄａ）受容体アンタゴニストとしてのその使用 |
| WO2009101940A1 (ja) * | 2008-02-11 | 2009-08-20 | Dainippon Sumitomo Pharma Co., Ltd. | 溶出性の改善された錠剤 |
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| EP1622625A1 (en) * | 2003-04-09 | 2006-02-08 | Wyeth | Pharmaceutical compositions for intranasal administration of [2-(8,9-dioxo-2,6-diazabicyclo [5.2.o] non-1 (7)-en-2-yl )alkyl] phosphonic acid and derivatives and methods of use thereof |
| GT200400213A (es) * | 2003-10-22 | 2007-09-05 | Metodos para la preparacion del acido {2-[(8,9)-dioxo-2,6-diaza-biciclo[5.2.0]-non-1(7)-en-2-il]etil} fosfonico y esteres del mismo | |
| US20050244365A1 (en) * | 2004-05-03 | 2005-11-03 | Novaflux Biosciences, Inc. | Methods, compositions, formulations, and uses of cellulose and acrylic-based polymers |
| ES2364495T3 (es) | 2005-02-03 | 2011-09-05 | The General Hospital Corporation | Método para tratar cáncer resistente a gefitinib. |
| JP2009514870A (ja) | 2005-11-04 | 2009-04-09 | ワイス | ｍＴＯＲインヒビター、ハーセプチン、および／またはＨＫＩ−２７２の抗悪性腫瘍性組み合わせ |
| EP2195031A1 (en) * | 2007-08-27 | 2010-06-16 | Wyeth a Corporation of the State of Delaware | Compositions and methods employing nmda antagonists for achieving an anesthetic-sparing effect |
| US8022216B2 (en) | 2007-10-17 | 2011-09-20 | Wyeth Llc | Maleate salts of (E)-N-{4-[3-chloro-4-(2-pyridinylmethoxy)anilino]-3-cyano-7-ethoxy-6-quinolinyl}-4-(dimethylamino)-2-butenamide and crystalline forms thereof |
| ES2692769T3 (es) | 2008-06-17 | 2018-12-05 | Wyeth Llc | Combinaciones antineoplásicas que contienen HKI-272 y vinorelbina |
| CN105147713A (zh) | 2008-08-04 | 2015-12-16 | 惠氏有限责任公司 | 4-苯胺基-3-氰基喹啉和卡培他滨的抗肿瘤组合 |
| US8778398B2 (en) * | 2008-11-04 | 2014-07-15 | Jazz Pharmaceuticals, Inc. | Immediate release formulations and dosage forms of gamma-hydroxybutyrate |
| US8771735B2 (en) * | 2008-11-04 | 2014-07-08 | Jazz Pharmaceuticals, Inc. | Immediate release dosage forms of sodium oxybate |
| SG174382A1 (en) | 2009-04-06 | 2011-11-28 | Wyeth Llc | Treatment regimen utilizing neratinib for breast cancer |
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| AU2010316683B2 (en) * | 2009-11-09 | 2015-10-08 | Wyeth Llc | Tablet formulations of neratinib maleate |
| MX391660B (es) | 2010-03-24 | 2025-03-21 | Jazz Pharmaceuticals Inc | Formas de dosis de liberacion controlada para substancias de farmaco de alta dosis, solubles en agua e higroscopicas |
| SMT201800657T1 (it) * | 2013-03-13 | 2019-01-11 | Sage Therapeutics Inc | Steroidi neuroattivi e loro metodi di utilizzo |
| US10398662B1 (en) | 2015-02-18 | 2019-09-03 | Jazz Pharma Ireland Limited | GHB formulation and method for its manufacture |
| PL3319611T3 (pl) | 2015-07-06 | 2021-07-12 | Sage Therapeutics, Inc. | Oksysterole i sposoby ich stosowania |
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| CA3041088C (en) | 2016-10-18 | 2024-05-21 | Sage Therapeutics, Inc. | Oxysterols and methods of use thereof |
| US20180263936A1 (en) | 2017-03-17 | 2018-09-20 | Jazz Pharmaceuticals Ireland Limited | Gamma-hydroxybutyrate compositions and their use for the treatment of disorders |
| BR112021006027A2 (pt) | 2018-11-19 | 2021-06-29 | Jazz Pharmaceuticals Ireland Limited | formulações de fármaco resistente a álcool |
| CN113473980A (zh) | 2019-03-01 | 2021-10-01 | 弗拉梅尔爱尔兰有限公司 | 在进食状态下具有改善的药代动力学的γ-羟基丁酸酯组合物 |
| TW202139986A (zh) | 2020-02-21 | 2021-11-01 | 愛爾蘭商爵士製藥愛爾蘭有限責任公司 | 治療原發性嗜睡症之方法 |
| US12582622B2 (en) | 2020-10-08 | 2026-03-24 | Jazz Pharmaceuticals Ireland Limited | Sodium oxybate to treat idiopathic hypersomnia |
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| JPH04321654A (ja) * | 1991-01-22 | 1992-11-11 | American Home Prod Corp | ［［２−（アミノ−３，４−ジオキソ−１−シクロブテン−１−イル）アミノ］アルキル］酸誘導体 |
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| JP2003286163A (ja) * | 2002-03-27 | 2003-10-07 | Nippon Zoki Pharmaceut Co Ltd | ジクロフェナクナトリウム経口製剤 |
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| US6225343B1 (en) * | 1999-06-16 | 2001-05-01 | Nastech Pharmaceutical Company, Inc. | Compositions and methods comprising morphine gluconate |
| US6468559B1 (en) * | 2000-04-28 | 2002-10-22 | Lipocine, Inc. | Enteric coated formulation of bishosphonic acid compounds and associated therapeutic methods |
| US6555581B1 (en) * | 2001-02-15 | 2003-04-29 | Jones Pharma, Inc. | Levothyroxine compositions and methods |
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| EP1622625A1 (en) * | 2003-04-09 | 2006-02-08 | Wyeth | Pharmaceutical compositions for intranasal administration of [2-(8,9-dioxo-2,6-diazabicyclo [5.2.o] non-1 (7)-en-2-yl )alkyl] phosphonic acid and derivatives and methods of use thereof |
-
2004
- 2004-10-08 US US10/961,871 patent/US20050142192A1/en not_active Abandoned
- 2004-10-13 TW TW093131004A patent/TW200528113A/zh unknown
- 2004-10-14 CA CA002541402A patent/CA2541402A1/en not_active Abandoned
- 2004-10-14 WO PCT/US2004/034113 patent/WO2005037287A1/en not_active Ceased
- 2004-10-14 JP JP2006535354A patent/JP2007509055A/ja active Pending
- 2004-10-14 AU AU2004281806A patent/AU2004281806A1/en not_active Abandoned
- 2004-10-14 BR BRPI0415432-0A patent/BRPI0415432A/pt not_active IP Right Cessation
- 2004-10-14 KR KR1020067007283A patent/KR20070029114A/ko not_active Withdrawn
- 2004-10-14 MX MXPA06003982A patent/MXPA06003982A/es unknown
- 2004-10-14 PA PA20048614901A patent/PA8614901A1/es unknown
- 2004-10-14 EP EP04795300A patent/EP1682151A1/en not_active Withdrawn
- 2004-10-15 PE PE2004001002A patent/PE20050480A1/es not_active Application Discontinuation
-
2006
- 2006-04-19 CO CO06037154A patent/CO5690561A2/es not_active Application Discontinuation
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| JPH04321654A (ja) * | 1991-01-22 | 1992-11-11 | American Home Prod Corp | ［［２−（アミノ−３，４−ジオキソ−１−シクロブテン−１−イル）アミノ］アルキル］酸誘導体 |
| WO2002067903A2 (en) * | 2001-02-27 | 2002-09-06 | Cephalon, Inc. | Compositions and methods of manufacture for oral dissolvable dosage forms |
| WO2003031416A2 (en) * | 2001-10-10 | 2003-04-17 | Wyeth | [[2-(amino-3,4-dioxo-1cyclobuten-1-yl)amino]alkyl]-acid derivatives for the treatment of pain |
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Cited By (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2006523694A (ja) * | 2003-04-09 | 2006-10-19 | ワイス | ［２−（８，９−ジオキソ−２，６−ジアザビシクロ［５．２．０］ノナ−１（７）−エン−２−イル）アルキル］ホスホン酸の誘導体およびｎ−メチル−ｄ−アスパルテート（ｎｍｄａ）受容体アンタゴニストとしてのその使用 |
| WO2009101940A1 (ja) * | 2008-02-11 | 2009-08-20 | Dainippon Sumitomo Pharma Co., Ltd. | 溶出性の改善された錠剤 |
| JPWO2009101940A1 (ja) * | 2008-02-11 | 2011-06-09 | 大日本住友製薬株式会社 | 溶出性の改善された錠剤 |
| US8673353B2 (en) | 2008-02-11 | 2014-03-18 | Dainippon Sumitomo Pharma Co., Ltd | Tablet having improved elution properties |
| US9463164B2 (en) | 2008-02-11 | 2016-10-11 | Sumitomo Dainippon Pharma Co., Ltd. | Tablet having improved elution properties |
Also Published As
| Publication number | Publication date |
|---|---|
| KR20070029114A (ko) | 2007-03-13 |
| BRPI0415432A (pt) | 2006-12-05 |
| CO5690561A2 (es) | 2006-10-31 |
| MXPA06003982A (es) | 2006-07-05 |
| EP1682151A1 (en) | 2006-07-26 |
| WO2005037287A1 (en) | 2005-04-28 |
| PE20050480A1 (es) | 2005-10-24 |
| PA8614901A1 (es) | 2006-05-16 |
| WO2005037287A8 (en) | 2005-06-30 |
| AU2004281806A1 (en) | 2005-04-28 |
| CA2541402A1 (en) | 2005-04-28 |
| TW200528113A (en) | 2005-09-01 |
| US20050142192A1 (en) | 2005-06-30 |
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