JP2007506703A5 - - Google Patents

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Publication number
JP2007506703A5
JP2007506703A5 JP2006527374A JP2006527374A JP2007506703A5 JP 2007506703 A5 JP2007506703 A5 JP 2007506703A5 JP 2006527374 A JP2006527374 A JP 2006527374A JP 2006527374 A JP2006527374 A JP 2006527374A JP 2007506703 A5 JP2007506703 A5 JP 2007506703A5
Authority
JP
Japan
Prior art keywords
alkyl
optionally substituted
quinolinecarboxamide
hydrogen
alkoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2006527374A
Other languages
English (en)
Japanese (ja)
Other versions
JP2007506703A (ja
Filing date
Publication date
Priority claimed from GBGB0322722.0A external-priority patent/GB0322722D0/en
Application filed filed Critical
Publication of JP2007506703A publication Critical patent/JP2007506703A/ja
Publication of JP2007506703A5 publication Critical patent/JP2007506703A5/ja
Pending legal-status Critical Current

Links

JP2006527374A 2003-09-27 2004-09-23 Pde4阻害剤としての4−アミノキノリン−3−カルボキサミド誘導体 Pending JP2007506703A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0322722.0A GB0322722D0 (en) 2003-09-27 2003-09-27 Compounds
PCT/EP2004/010844 WO2005030212A1 (en) 2003-09-27 2004-09-23 4-aminoquinoline-3-carboxamide derivatives as pde4 inhibitors

Publications (2)

Publication Number Publication Date
JP2007506703A JP2007506703A (ja) 2007-03-22
JP2007506703A5 true JP2007506703A5 (OSRAM) 2007-09-20

Family

ID=29287002

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006527374A Pending JP2007506703A (ja) 2003-09-27 2004-09-23 Pde4阻害剤としての4−アミノキノリン−3−カルボキサミド誘導体

Country Status (10)

Country Link
US (1) US20080096884A1 (OSRAM)
EP (1) EP1673086B1 (OSRAM)
JP (1) JP2007506703A (OSRAM)
AR (1) AR045824A1 (OSRAM)
AT (1) ATE384530T1 (OSRAM)
DE (1) DE602004011548T2 (OSRAM)
ES (1) ES2298806T3 (OSRAM)
GB (1) GB0322722D0 (OSRAM)
TW (1) TW200526584A (OSRAM)
WO (1) WO2005030212A1 (OSRAM)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI328009B (en) * 2003-05-21 2010-08-01 Glaxo Group Ltd Quinoline derivatives as phosphodiesterase inhibitors
GB0601951D0 (en) 2006-01-31 2006-03-15 Novartis Ag Organic compounds
GB0605462D0 (en) * 2006-03-17 2006-04-26 Glaxo Group Ltd Novel compounds
WO2008052734A1 (en) 2006-10-30 2008-05-08 Novartis Ag Heterocyclic compounds as antiinflammatory agents
JP5584138B2 (ja) 2008-01-11 2014-09-03 ノバルティス アーゲー キナーゼ阻害剤としてのピリミジン類
EP2379076B1 (en) * 2008-12-23 2014-11-12 The Trustees of Columbia University in the City of New York Phosphodiesterase inhibitors and uses thereof
WO2010097248A1 (en) 2009-01-13 2010-09-02 Glaxo Group Limited Pyrimidinecarboxamide derivatives as inhibitors of syk kinase
US8367829B2 (en) 2010-05-10 2013-02-05 Gilead Sciences, Inc. Bi-functional pyrazolopyridine compounds
US8394829B2 (en) 2010-05-10 2013-03-12 Gilead Sciences, Inc. Bi-functional quinoline analogs
UY33597A (es) 2010-09-09 2012-04-30 Irm Llc Compuestos y composiciones como inhibidores de la trk
WO2012034095A1 (en) 2010-09-09 2012-03-15 Irm Llc Compounds and compositions as trk inhibitors
CA2828219A1 (en) 2011-02-25 2012-08-30 Irm Llc Pyrazolo [1,5-a] pyridines as trk inhibitors
BR112015019276A2 (pt) 2013-02-19 2017-07-18 Pfizer compostos de azabenzimidazol como inibidores de isoenzimas de pde4 para o tratamento de distúrbios do snc e outros distúrbios
US10131669B2 (en) 2014-07-24 2018-11-20 Pfizer Inc. Pyrazolopyrimidine compounds
EA031201B1 (ru) 2014-08-06 2018-11-30 Пфайзер Инк. Соединения имидазопиридазина
MA41140A (fr) 2014-12-12 2017-10-17 Cancer Research Tech Ltd Dérivés de 2,4-dioxo-quinazoline-6-sulfonamide en tant qu'inhibiteurs de la parg
MA41179A (fr) 2014-12-19 2017-10-24 Cancer Research Tech Ltd Composés inhibiteurs de parg
BR112018006873A2 (pt) 2015-10-05 2018-11-06 The Trustees Of Columbia University In The City Of New York ativadores do fluxo autofágico e fosfolipase d e depuração de agregados de proteína incluindo tau e tratamento de proteinopatias
TW202345809A (zh) 2022-03-23 2023-12-01 美商愛德亞生物科學公司 作為parg抑制劑之經哌取代的吲唑化合物
TW202430172A (zh) * 2023-01-17 2024-08-01 大陸商瑞石生物醫藥有限公司 Pde4抑制劑、其製備方法及其在醫藥上的應用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR920701162A (ko) * 1990-03-28 1992-08-11 오츠카 아끼히코 퀴놀린 유도체, 당해 유도체를 함유하는 항궤양제 및 당해 유도체의 제조방법
AU722662B2 (en) * 1996-05-20 2000-08-10 Darwin Discovery Limited Quinoline sulfonamides as TNF inhibitors and as PDE-IV inhibitors
ATE303993T1 (de) * 1997-12-22 2005-09-15 Pharmacia & Upjohn Co Llc 4-hydroxychinolin-3-carboxamide und hydrazide als antivirale wirkstoffe
US6576644B2 (en) * 2000-09-06 2003-06-10 Bristol-Myers Squibb Co. Quinoline inhibitors of cGMP phosphodiesterase
SE0101675D0 (sv) * 2001-05-11 2001-05-11 Astrazeneca Ab Novel composition
JO2311B1 (en) * 2001-08-29 2005-09-12 ميرك فروست كندا ليمتد Alkyl inhibitors Ariel phosphodiesterase-4

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