JP2006503056A5 - - Google Patents
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- Publication number
- JP2006503056A5 JP2006503056A5 JP2004537671A JP2004537671A JP2006503056A5 JP 2006503056 A5 JP2006503056 A5 JP 2006503056A5 JP 2004537671 A JP2004537671 A JP 2004537671A JP 2004537671 A JP2004537671 A JP 2004537671A JP 2006503056 A5 JP2006503056 A5 JP 2006503056A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- phenyl
- halogens
- och
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 claims 6
- -1 N-piperidinyl Chemical group 0.000 claims 6
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 claims 5
- 229910052736 halogen Inorganic materials 0.000 claims 5
- 150000002367 halogens Chemical class 0.000 claims 4
- 150000001875 compounds Chemical class 0.000 claims 2
- 150000003839 salts Chemical class 0.000 claims 2
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 claims 1
- 125000005037 alkyl phenyl group Chemical group 0.000 claims 1
- 239000004305 biphenyl Substances 0.000 claims 1
- 239000003937 drug carrier Substances 0.000 claims 1
- 125000005843 halogen group Chemical group 0.000 claims 1
- 239000008194 pharmaceutical composition Substances 0.000 claims 1
- 239000012453 solvate Substances 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41162502P | 2002-09-18 | 2002-09-18 | |
| PCT/US2003/025860 WO2004026837A2 (en) | 2002-09-18 | 2003-09-12 | Histamine h3 receptor antagonists, preparaton and therapeutic uses |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2006503056A JP2006503056A (ja) | 2006-01-26 |
| JP2006503056A5 true JP2006503056A5 (https=) | 2006-10-19 |
Family
ID=32030698
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004537671A Pending JP2006503056A (ja) | 2002-09-18 | 2003-09-12 | ヒスタミンｈ３受容体アンタゴニスト、その製造および治療用使用 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20060167046A1 (https=) |
| EP (1) | EP1585731A2 (https=) |
| JP (1) | JP2006503056A (https=) |
| AU (1) | AU2003268117A1 (https=) |
| WO (1) | WO2004026837A2 (https=) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR048134A1 (es) * | 2003-12-15 | 2006-04-05 | Lundbeck & Co As H | La combinacion de un inhibidor de la recaptacion de serotonina y un antagonista del receptor de la histamina 3, el agonista inverso o el agonista parcial |
| US20060069087A1 (en) * | 2004-09-27 | 2006-03-30 | Pfizer Inc | Histamine-3 receptor antagonists |
| BRPI0613430A2 (pt) | 2005-07-13 | 2011-01-11 | Hoffmann La Roche | compostos derivados de benzimidazol, uso dos mesmos, método para a preparação destes e composição farmacêutica |
| ES2351940T3 (es) * | 2005-11-18 | 2011-02-14 | F. Hoffmann-La Roche Ag | Derivados de azaindol-2-carboxamida. |
| JP2009518351A (ja) * | 2005-12-09 | 2009-05-07 | エフ．ホフマン−ラ ロシュ アーゲー | 肥満症の処置に有用な三環性アミド誘導体 |
| CA2646023A1 (en) | 2006-03-10 | 2007-09-20 | Neurogen Corporation | Piperazinyl oxoalkyl tetrahydroisoquinolines and related analogues |
| JPWO2007129745A1 (ja) | 2006-05-09 | 2009-09-17 | 第一三共株式会社 | ヘテロアリールアミド低級カルボン酸誘導体 |
| RU2009136330A (ru) | 2007-03-01 | 2011-04-10 | Янссен Фармацевтика Н.В. (Be) | Тетрагидроизохинолиновые соединения в качестве модуляторов гистаминового н3 рецептора |
| WO2008126886A1 (ja) * | 2007-04-12 | 2008-10-23 | Taisho Pharmaceutical Co., Ltd. | インドール又はインドリン誘導体 |
| TW201039822A (en) * | 2009-02-06 | 2010-11-16 | Taisho Pharmaceutical Co Ltd | Dihydroquinolinone derivatives |
| WO2013151982A1 (en) | 2012-04-03 | 2013-10-10 | Arena Pharmaceuticals, Inc. | Methods and compounds useful in treating pruritus, and methods for identifying such compounds |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5310986B2 (https=) * | 1974-02-05 | 1978-04-18 | ||
| JPS5310989B2 (https=) * | 1974-04-25 | 1978-04-18 | ||
| JPS533534A (en) * | 1976-06-30 | 1978-01-13 | Otsuka Pharmaceut Co Ltd | Local anesthetics |
| JPS5780322A (en) * | 1980-11-05 | 1982-05-19 | Otsuka Pharmaceut Co Ltd | Cardiotonic agent |
| JPS63290821A (ja) * | 1987-05-25 | 1988-11-28 | Otsuka Pharmaceut Co Ltd | 抗不整脈剤 |
| EP1268484A1 (en) * | 2000-03-17 | 2003-01-02 | Novo Nordisk A/S | Condensed imidazoles as histamine h3 receptor ligands |
| GB0019950D0 (en) * | 2000-08-12 | 2000-09-27 | Smithkline Beecham Plc | Compounds |
| ATE283853T1 (de) * | 2000-09-20 | 2004-12-15 | Schering Corp | Substituierte imidazole als duale histamine h1 und h3 agonisten oder antagonisten |
| TW593278B (en) * | 2001-01-23 | 2004-06-21 | Wyeth Corp | 1-aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands |
-
2003
- 2003-09-12 AU AU2003268117A patent/AU2003268117A1/en not_active Abandoned
- 2003-09-12 US US10/525,315 patent/US20060167046A1/en not_active Abandoned
- 2003-09-12 WO PCT/US2003/025860 patent/WO2004026837A2/en not_active Ceased
- 2003-09-12 EP EP03749068A patent/EP1585731A2/en not_active Withdrawn
- 2003-09-12 JP JP2004537671A patent/JP2006503056A/ja active Pending
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