JP2006501201A - 化合物、組成物および方法 - Google Patents
化合物、組成物および方法 Download PDFInfo
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- JP2006501201A JP2006501201A JP2004523405A JP2004523405A JP2006501201A JP 2006501201 A JP2006501201 A JP 2006501201A JP 2004523405 A JP2004523405 A JP 2004523405A JP 2004523405 A JP2004523405 A JP 2004523405A JP 2006501201 A JP2006501201 A JP 2006501201A
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- benzyl
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Classifications
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
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- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
- C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
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EP1556357A4 (en) * | 2002-06-14 | 2006-09-13 | Cytokinetics Inc | COMPOUNDS, COMPOSITIONS AND METHODS |
US20040092561A1 (en) * | 2002-11-07 | 2004-05-13 | Thomas Ruckle | Azolidinone-vinyl fused -benzene derivatives |
AU2003256805A1 (en) * | 2002-07-23 | 2004-02-09 | Cytokinetics, Inc. | Compounds compositions and methods |
US20040048853A1 (en) * | 2002-08-21 | 2004-03-11 | Gustave Bergnes | Compounds, compositions, and methods |
CA2536633A1 (en) * | 2003-09-10 | 2005-03-24 | Icagen, Inc. | Fused ring heterocycles as potassium channel modulators |
US20050152940A1 (en) * | 2003-12-23 | 2005-07-14 | Medtronic Vascular, Inc. | Medical devices to treat or inhibit restenosis |
-
2003
- 2003-07-23 AU AU2003256805A patent/AU2003256805A1/en not_active Abandoned
- 2003-07-23 EP EP03766028A patent/EP1537089A4/en not_active Withdrawn
- 2003-07-23 JP JP2004523405A patent/JP2006501201A/ja active Pending
- 2003-07-23 WO PCT/US2003/023319 patent/WO2004009036A2/en active Application Filing
- 2003-07-23 US US10/626,012 patent/US7211580B2/en not_active Expired - Fee Related
-
2007
- 2007-03-12 US US11/717,223 patent/US20080021050A1/en not_active Abandoned
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2010540525A (ja) * | 2007-09-26 | 2010-12-24 | セルジーン コーポレイション | 6、7又は8置換キナゾリノン誘導体並びにそれらを含有する組成物及びそれらを使用する方法 |
JP2013545744A (ja) * | 2010-11-10 | 2013-12-26 | アクテリオン ファーマシューティカルズ リミテッド | オレキシン受容体拮抗薬として有用なラクタム誘導体 |
Also Published As
Publication number | Publication date |
---|---|
US20080021050A1 (en) | 2008-01-24 |
AU2003256805A1 (en) | 2004-02-09 |
EP1537089A2 (en) | 2005-06-08 |
AU2003256805A8 (en) | 2004-02-09 |
US20040142949A1 (en) | 2004-07-22 |
EP1537089A4 (en) | 2008-04-16 |
WO2004009036A2 (en) | 2004-01-29 |
WO2004009036A3 (en) | 2004-08-19 |
US7211580B2 (en) | 2007-05-01 |
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