JP2005536553A - 化合物、組成物および方法 - Google Patents

化合物、組成物および方法 Download PDF

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Publication number
JP2005536553A
JP2005536553A JP2004531141A JP2004531141A JP2005536553A JP 2005536553 A JP2005536553 A JP 2005536553A JP 2004531141 A JP2004531141 A JP 2004531141A JP 2004531141 A JP2004531141 A JP 2004531141A JP 2005536553 A JP2005536553 A JP 2005536553A
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optionally substituted
benzyl
tolyl
propyl
compound
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JP2004531141A
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Japanese (ja)
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JP2005536553A5 (https=
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ベルグネス,ギュスターヴ
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Cytokinetics Inc
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Cytokinetics Inc
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Publication of JP2005536553A publication Critical patent/JP2005536553A/ja
Publication of JP2005536553A5 publication Critical patent/JP2005536553A5/ja
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
JP2004531141A 2002-08-21 2003-08-20 化合物、組成物および方法 Pending JP2005536553A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40486402P 2002-08-21 2002-08-21
PCT/US2003/026093 WO2004018058A2 (en) 2002-08-21 2003-08-20 Compounds, compositions, and methods

Publications (2)

Publication Number Publication Date
JP2005536553A true JP2005536553A (ja) 2005-12-02
JP2005536553A5 JP2005536553A5 (https=) 2006-08-03

Family

ID=31946773

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004531141A Pending JP2005536553A (ja) 2002-08-21 2003-08-20 化合物、組成物および方法

Country Status (5)

Country Link
US (2) US20040048853A1 (https=)
EP (1) EP1539180A4 (https=)
JP (1) JP2005536553A (https=)
AU (1) AU2003262747A1 (https=)
WO (1) WO2004018058A2 (https=)

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JP2007524600A (ja) * 2003-03-25 2007-08-30 タケダ サン ディエゴ インコーポレイテッド ジペプチジルペプチダーゼインヒビター
JP2022509434A (ja) * 2018-10-31 2022-01-20 アコンディシオナミエント タルラセンス 疼痛に対して活性があるピペラジニル及びピペリジニルキナゾリン-4(3h)-オン誘導体
JP2022551156A (ja) * 2019-10-10 2022-12-07 エステベ ファーマシューティカルズ,ソシエダッド アノニマ 疼痛に対する多様な活性を有するホモピペラジニル及びホモピペリジニルキナゾリン-4(3h)-オン誘導体

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