JP2005529923A - 肥満および糖尿病の治療におけるメラニン凝集ホルモンアンタゴニストとして使用するための多環式化合物 - Google Patents

肥満および糖尿病の治療におけるメラニン凝集ホルモンアンタゴニストとして使用するための多環式化合物 Download PDF

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JP2005529923A
JP2005529923A JP2004505046A JP2004505046A JP2005529923A JP 2005529923 A JP2005529923 A JP 2005529923A JP 2004505046 A JP2004505046 A JP 2004505046A JP 2004505046 A JP2004505046 A JP 2004505046A JP 2005529923 A JP2005529923 A JP 2005529923A
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phenoxy
oxadiazol
ethylsulfanylmethyl
phenyl
mmol
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JP2005529923A5 (OSRAM
Inventor
ヨッヘン・アンメン
ジェイムズ・ロナルド・ジリグ
ローレンス・ジョゼフ・ハインツ
フィリップ・アーサー・ヒップスカインド
マイケル・ディーン・キニック
ライ・イェン−シ
ジョン・マイケル・モリン・ジュニア
ジェイムズ・アーサー・ニクソン
カルステン・オット
ケネス・アレン・セイビン
テオ・ショッテン
ローレンス・ジョン・スリーカー
ナンシー・ジューン・スナイダー
マイケル・アラン・ロバートソン
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Eli Lilly and Co
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Eli Lilly and Co
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  • Organic Chemistry (AREA)
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  • Obesity (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
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JP2004505046A 2002-05-13 2003-05-06 肥満および糖尿病の治療におけるメラニン凝集ホルモンアンタゴニストとして使用するための多環式化合物 Pending JP2005529923A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38035102P 2002-05-13 2002-05-13
PCT/US2003/012123 WO2003097047A1 (en) 2002-05-13 2003-05-06 Multicyclic compounds for use as melanin concentrating hormone antagonists in the treatment of obesity and diabetes

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JP2005529923A true JP2005529923A (ja) 2005-10-06
JP2005529923A5 JP2005529923A5 (OSRAM) 2006-06-29

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JP2004505046A Pending JP2005529923A (ja) 2002-05-13 2003-05-06 肥満および糖尿病の治療におけるメラニン凝集ホルモンアンタゴニストとして使用するための多環式化合物

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US (1) US7229987B2 (OSRAM)
EP (1) EP1505968A1 (OSRAM)
JP (1) JP2005529923A (OSRAM)
AU (1) AU2003222648A1 (OSRAM)
CA (1) CA2484233A1 (OSRAM)
WO (1) WO2003097047A1 (OSRAM)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007043400A1 (ja) * 2005-10-07 2007-04-19 Kissei Pharmaceutical Co., Ltd. 含窒素芳香族複素環化合物およびそれを含有する医薬組成物
JP2007510629A (ja) * 2003-10-22 2007-04-26 イーライ リリー アンド カンパニー 新規ｍｃｈ受容体アンタゴニスト
JP2009108028A (ja) * 2007-08-30 2009-05-21 National Sun Yat-Sen Univ イオウ含有化合物、その調製方法および薬学的使用
JP2010504320A (ja) * 2006-09-21 2010-02-12 アクテリオン ファーマシューティカルズ リミテッド フェニル誘導体及びそれらの免疫調節薬としての使用
JP2010538001A (ja) * 2007-08-27 2010-12-09 ヘリコン・セラピューティクス・インコーポレーテッド 治療用イソオキサゾール化合物
JP2014205687A (ja) * 2008-05-30 2014-10-30 株式会社アールテック・ウエノ ベンゼンまたはチオフェン誘導体およびｖａｐ−１阻害剤としてのその使用

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Publication number Priority date Publication date Assignee Title
AU2002352878B2 (en) 2001-11-27 2007-11-22 Merck Sharp & Dohme Corp. 2-Aminoquinoline compounds
JPWO2004069798A1 (ja) 2003-02-10 2006-05-25 萬有製薬株式会社 ピペリジン誘導体を有効成分とするメラニン凝集ホルモン受容体拮抗剤
EP1706384A1 (en) * 2004-01-07 2006-10-04 AstraZeneca AB Therapeutic agents i
US7550602B1 (en) * 2004-01-14 2009-06-23 Palatin Technologies, Inc. Small molecule compositions for sexual dysfunction
US7319108B2 (en) 2004-01-25 2008-01-15 Sanofi-Aventis Deutschland Gmbh Aryl-substituted heterocycles, process for their preparation and their use as medicaments
US7241787B2 (en) 2004-01-25 2007-07-10 Sanofi-Aventis Deutschland Gmbh Substituted N-cycloexylimidazolinones, process for their preparation and their use as medicaments
DE102004003812A1 (de) * 2004-01-25 2005-08-11 Aventis Pharma Deutschland Gmbh Arylsubstituierte Heterozyklen, Verfahren ihrer Herstellung und ihre Verwendung als Arzneimittel
DE102004017932A1 (de) * 2004-04-14 2005-11-03 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Alkin-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel
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