JP2005516946A5 - - Google Patents
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- Publication number
- JP2005516946A5 JP2005516946A5 JP2003554189A JP2003554189A JP2005516946A5 JP 2005516946 A5 JP2005516946 A5 JP 2005516946A5 JP 2003554189 A JP2003554189 A JP 2003554189A JP 2003554189 A JP2003554189 A JP 2003554189A JP 2005516946 A5 JP2005516946 A5 JP 2005516946A5
- Authority
- JP
- Japan
- Prior art keywords
- present
- tegaserod
- granulation
- formulations
- minutes
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000000203 mixture Substances 0.000 description 2
- 229960002876 Tegaserod Drugs 0.000 description 1
- 238000004090 dissolution Methods 0.000 description 1
- 238000001035 drying Methods 0.000 description 1
- 238000005469 granulation Methods 0.000 description 1
- 230000003179 granulation Effects 0.000 description 1
- IKBKZGMPCYNSLU-RGVLZGJSSA-N tegaserod Chemical compound C1=C(OC)C=C2C(/C=N/NC(=N)NCCCCC)=CNC2=C1 IKBKZGMPCYNSLU-RGVLZGJSSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP01403339A EP1321142A1 (en) | 2001-12-21 | 2001-12-21 | Solid pharmaceutical composition for oral administration of Tegaserod |
| EP01403339.3 | 2001-12-21 | ||
| PCT/EP2002/014674 WO2003053432A1 (en) | 2001-12-21 | 2002-12-20 | 5ht4 partial agonist pharmaceutical compositions |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005516946A JP2005516946A (ja) | 2005-06-09 |
| JP2005516946A5 true JP2005516946A5 (pt) | 2006-01-19 |
| JP4718776B2 JP4718776B2 (ja) | 2011-07-06 |
Family
ID=8183045
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003554189A Expired - Fee Related JP4718776B2 (ja) | 2001-12-21 | 2002-12-20 | ５ｈｔ４部分アゴニスト医薬組成物 |
Country Status (31)
| Country | Link |
|---|---|
| US (2) | US20050106236A1 (pt) |
| EP (2) | EP1321142A1 (pt) |
| JP (1) | JP4718776B2 (pt) |
| KR (1) | KR100980144B1 (pt) |
| CN (1) | CN100464749C (pt) |
| AR (1) | AR037937A1 (pt) |
| AT (1) | ATE320807T1 (pt) |
| AU (1) | AU2002361198B2 (pt) |
| BR (1) | BR0215148A (pt) |
| CA (1) | CA2470668C (pt) |
| CO (1) | CO5640102A2 (pt) |
| CY (1) | CY1105559T1 (pt) |
| DE (1) | DE60210139T2 (pt) |
| DK (1) | DK1458377T3 (pt) |
| EC (1) | ECSP105163A (pt) |
| EG (1) | EG24194A (pt) |
| ES (1) | ES2258171T3 (pt) |
| HU (1) | HU226589B1 (pt) |
| IL (2) | IL162451A0 (pt) |
| MX (1) | MXPA04006157A (pt) |
| MY (1) | MY139546A (pt) |
| NO (1) | NO20042779L (pt) |
| NZ (1) | NZ533585A (pt) |
| PE (1) | PE20030872A1 (pt) |
| PL (1) | PL369509A1 (pt) |
| PT (1) | PT1458377E (pt) |
| RU (1) | RU2322978C2 (pt) |
| SI (1) | SI1458377T1 (pt) |
| TW (1) | TWI260221B (pt) |
| WO (1) | WO2003053432A1 (pt) |
| ZA (1) | ZA200404467B (pt) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL141236A0 (en) * | 1998-08-21 | 2002-03-10 | Novartis Ag | New oral formulations for 5-ht4 agonists or antagonists |
| SG192300A1 (en) | 2003-01-28 | 2013-08-30 | Ironwood Pharmaceuticals Inc | Methods and compositions for the treatment of gastrointestinal disorders |
| US7772188B2 (en) | 2003-01-28 | 2010-08-10 | Ironwood Pharmaceuticals, Inc. | Methods and compositions for the treatment of gastrointestinal disorders |
| AU2003222439A1 (en) * | 2003-03-25 | 2004-10-18 | Hetero Drugs Limited | Novel crystalline forms of tegaserod maleate |
| WO2004104577A2 (en) * | 2003-05-21 | 2004-12-02 | Bayer Healthcare Ag | Diagnostics and therapeutics for diseases associated with 5-hydroxytryptamine (serotonin) receptor 4 (5-ht4) |
| PE20050253A1 (es) * | 2003-07-24 | 2005-06-03 | Novartis Ag | Modificaciones estables de maleato de hidrogeno de tegaserod |
| DK1663182T4 (da) | 2003-09-12 | 2020-02-17 | Amgen Inc | Hurtigt opløsende formulering af cinacalcet HCI |
| JP2007514000A (ja) * | 2003-12-16 | 2007-05-31 | テバ ファーマシューティカル インダストリーズ リミティド | テガセロッド塩基及びその塩の多形現象形 |
| CZ298399B6 (cs) * | 2005-05-02 | 2007-09-19 | Zentiva, A. S. | Zpusob prípravy 2-[(5-methoxy-1 H-indol-3-yl) methylen]-N-pentylkarbazimidamidu (tegaserodu) |
| US20070259052A1 (en) | 2006-05-05 | 2007-11-08 | Shire International Licensing B.V. | Assay for lanthanum hydroxycarbonate |
| US8969514B2 (en) | 2007-06-04 | 2015-03-03 | Synergy Pharmaceuticals, Inc. | Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases |
| MX354786B (es) | 2007-06-04 | 2018-03-21 | Synergy Pharmaceuticals Inc | Agonistas de guanilato ciclasa utiles para el tratamiento de trastornos gastrointestinales, inflamacion, cancer y otros trastornos. |
| CA2726917C (en) | 2008-06-04 | 2018-06-26 | Synergy Pharmaceuticals Inc. | Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders |
| WO2010009319A2 (en) | 2008-07-16 | 2010-01-21 | Synergy Pharmaceuticals Inc. | Agonists of guanylate cyclase useful for the treatment of gastrointestinal, inflammation, cancer and other disorders |
| WO2010078449A2 (en) | 2008-12-31 | 2010-07-08 | Ardelyx, Inc. | Compounds and methods for inhibiting nhe-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders |
| WO2018129556A1 (en) | 2017-01-09 | 2018-07-12 | Ardelyx, Inc. | Compounds and methods for inhibiting nhe-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders |
| US10376481B2 (en) | 2012-08-21 | 2019-08-13 | Ardelyx, Inc. | Compounds and methods for inhibiting NHE-mediated antiport in the treatment of disorders associated with fluid retention or salt overload and gastrointestinal tract disorders |
| CN104902930A (zh) | 2012-08-21 | 2015-09-09 | 阿德利克斯公司 | 在治疗与液体潴留或盐分过载相关的疾病和胃肠道疾病中用于抑制nhe-介导的反向转运的化合物和方法 |
| EP2970384A1 (en) | 2013-03-15 | 2016-01-20 | Synergy Pharmaceuticals Inc. | Agonists of guanylate cyclase and their uses |
| WO2014151200A2 (en) | 2013-03-15 | 2014-09-25 | Synergy Pharmaceuticals Inc. | Compositions useful for the treatment of gastrointestinal disorders |
| HUE044550T2 (hu) | 2013-04-12 | 2019-11-28 | Ardelyx Inc | NHE-3 megkötõ vegyületek és foszfát transzport gátlási módszerek |
| CN104922083B (zh) * | 2015-04-15 | 2017-12-22 | 湖南尔康湘药制药有限公司 | 磺胺嘧啶片及其制备方法 |
| EA036204B1 (ru) * | 2015-10-16 | 2020-10-14 | Нобел Илач Санайи Ве Тиджарет А.Ш. | Фармацевтические композиции нилотиниба гидрохлорида |
| CN110267944B (zh) | 2017-01-09 | 2024-03-08 | 阿德利克斯股份有限公司 | 可用于治疗胃肠道病症的化合物 |
| JP2020505333A (ja) | 2017-01-09 | 2020-02-20 | アルデリックス， インコーポレイテッド | Ｎｈｅ媒介性アンチポートの阻害薬 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH0820586A (ja) * | 1994-07-05 | 1996-01-23 | Sanwa Kagaku Kenkyusho Co Ltd | １−アザビシクロ［３．３．０］オクタン誘導体、その塩及び製法並びに用途 |
| IL117438A (en) * | 1995-03-16 | 2001-12-23 | Lilly Co Eli | Indazolecarboxamides, their preparation and pharmaceutical compositions containing them |
| JPH09194374A (ja) * | 1995-11-14 | 1997-07-29 | Taisho Pharmaceut Co Ltd | 消化器疾患治療剤 |
| DE69713948D1 (de) * | 1996-04-23 | 2002-08-22 | Janssen Pharmaceutica Nv | Rasch-freisetzende pH-unabhängige feste Dosisformen enthaltend Cisaprid |
| US5739151A (en) * | 1996-07-19 | 1998-04-14 | Sepracor Inc. | Method for treating emesis and central nervous system disorders using optically pure (+) norcisapride |
| IL141236A0 (en) * | 1998-08-21 | 2002-03-10 | Novartis Ag | New oral formulations for 5-ht4 agonists or antagonists |
| US6465502B1 (en) * | 1998-12-23 | 2002-10-15 | Novartis Ag | Additional therapeutic use |
| WO2000057857A1 (en) * | 1999-03-25 | 2000-10-05 | Yuhan Corporation | Rapidly disintegrable tablet for oral administration |
| ES2435816T3 (es) * | 1999-08-03 | 2013-12-23 | Icos Corporation | Formulación farmacéutica que comprende una Beta-carbolina y su uso para el tratamiento de la disfunción sexual |
-
2001
- 2001-12-21 EP EP01403339A patent/EP1321142A1/en not_active Withdrawn
-
2002
- 2002-12-17 EG EG2002121358A patent/EG24194A/xx active
- 2002-12-19 TW TW091136675A patent/TWI260221B/zh not_active IP Right Cessation
- 2002-12-19 AR ARP020105024A patent/AR037937A1/es not_active Application Discontinuation
- 2002-12-20 NZ NZ533585A patent/NZ533585A/en not_active IP Right Cessation
- 2002-12-20 CA CA2470668A patent/CA2470668C/en not_active Expired - Fee Related
- 2002-12-20 US US10/499,721 patent/US20050106236A1/en not_active Abandoned
- 2002-12-20 RU RU2004122631/15A patent/RU2322978C2/ru not_active IP Right Cessation
- 2002-12-20 SI SI200230334T patent/SI1458377T1/sl unknown
- 2002-12-20 WO PCT/EP2002/014674 patent/WO2003053432A1/en active IP Right Grant
- 2002-12-20 PT PT02796711T patent/PT1458377E/pt unknown
- 2002-12-20 MX MXPA04006157A patent/MXPA04006157A/es active IP Right Grant
- 2002-12-20 MY MYPI20024825A patent/MY139546A/en unknown
- 2002-12-20 DE DE60210139T patent/DE60210139T2/de not_active Expired - Lifetime
- 2002-12-20 CN CNB028255321A patent/CN100464749C/zh not_active Expired - Fee Related
- 2002-12-20 DK DK02796711T patent/DK1458377T3/da active
- 2002-12-20 PL PL02369509A patent/PL369509A1/xx not_active Application Discontinuation
- 2002-12-20 KR KR1020047009594A patent/KR100980144B1/ko not_active IP Right Cessation
- 2002-12-20 AT AT02796711T patent/ATE320807T1/de active
- 2002-12-20 BR BR0215148-0A patent/BR0215148A/pt not_active IP Right Cessation
- 2002-12-20 JP JP2003554189A patent/JP4718776B2/ja not_active Expired - Fee Related
- 2002-12-20 ES ES02796711T patent/ES2258171T3/es not_active Expired - Lifetime
- 2002-12-20 AU AU2002361198A patent/AU2002361198B2/en not_active Ceased
- 2002-12-20 EP EP02796711A patent/EP1458377B1/en not_active Expired - Lifetime
- 2002-12-20 IL IL16245102A patent/IL162451A0/xx active IP Right Grant
- 2002-12-20 HU HU0402492A patent/HU226589B1/hu not_active IP Right Cessation
-
2003
- 2003-01-06 PE PE2003000004A patent/PE20030872A1/es not_active Application Discontinuation
-
2004
- 2004-06-07 ZA ZA200404467A patent/ZA200404467B/en unknown
- 2004-06-10 IL IL162451A patent/IL162451A/en not_active IP Right Cessation
- 2004-07-01 NO NO20042779A patent/NO20042779L/no not_active Application Discontinuation
- 2004-07-15 CO CO04067463A patent/CO5640102A2/es not_active Application Discontinuation
-
2006
- 2006-05-04 CY CY20061100579T patent/CY1105559T1/el unknown
-
2008
- 2008-10-07 US US12/287,232 patent/US20090104263A1/en not_active Abandoned
-
2010
- 2010-06-16 EC EC2010005163A patent/ECSP105163A/es unknown
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