JP2005508983A5 - - Google Patents

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Publication number
JP2005508983A5
JP2005508983A5 JP2003541843A JP2003541843A JP2005508983A5 JP 2005508983 A5 JP2005508983 A5 JP 2005508983A5 JP 2003541843 A JP2003541843 A JP 2003541843A JP 2003541843 A JP2003541843 A JP 2003541843A JP 2005508983 A5 JP2005508983 A5 JP 2005508983A5
Authority
JP
Japan
Prior art keywords
methyl
drug
dione
rheumatic
dmard
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003541843A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005508983A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2002/012415 external-priority patent/WO2003039552A1/en
Publication of JP2005508983A publication Critical patent/JP2005508983A/ja
Publication of JP2005508983A5 publication Critical patent/JP2005508983A5/ja
Pending legal-status Critical Current

Links

JP2003541843A 2001-11-09 2002-11-07 Pde4又はpde3/4阻害剤及び抗リウマチ薬の複合薬 Pending JP2005508983A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01000607 2001-11-09
PCT/EP2002/012415 WO2003039552A1 (en) 2001-11-09 2002-11-07 Combination of pde4 or pde3/4 inhibitor and an anti-rheumatic drug

Publications (2)

Publication Number Publication Date
JP2005508983A JP2005508983A (ja) 2005-04-07
JP2005508983A5 true JP2005508983A5 (https=) 2006-01-05

Family

ID=8176085

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003541843A Pending JP2005508983A (ja) 2001-11-09 2002-11-07 Pde4又はpde3/4阻害剤及び抗リウマチ薬の複合薬

Country Status (6)

Country Link
US (2) US20030092706A1 (https=)
EP (1) EP1448202A1 (https=)
JP (1) JP2005508983A (https=)
AU (1) AU2002300754B2 (https=)
CA (1) CA2399840C (https=)
WO (1) WO2003039552A1 (https=)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7718644B2 (en) * 2004-01-22 2010-05-18 The Trustees Of Columbia University In The City Of New York Anti-arrhythmic and heart failure drugs that target the leak in the ryanodine receptor (RyR2) and uses thereof
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
ME00565A (en) * 2002-05-28 2011-12-20 Topically applicable pharmaceutical preparation
US6727272B1 (en) * 2002-07-15 2004-04-27 Unitech Pharmaceuticals, Inc. Leflunomide analogs for treating rheumatoid arthritis
UA82323C2 (uk) * 2002-08-09 2008-04-10 Меда Фарма Гмбх & Ко. Кг Нова комбінація глюкокортикоїду та pde-інгібітору для лікування респіраторних захворювань, алергічних захворювань, астми та хронічних обструктивних легеневих захворювань
PT1606261E (pt) 2003-03-10 2010-01-11 Nycomed Gmbh Novo processo para a preparação de roflumilast
EP1755595A1 (en) * 2004-05-10 2007-02-28 Altana Pharma AG Use of roflumilast for the prophylaxis or treatment of emphysema
EP1815867A4 (en) * 2004-11-02 2010-06-09 Dainippon Sumitomo Pharma Co COMBINATION PREPARATION FOR THE TREATMENT OF AUTOIMMUNE DISEASE
JP5385605B2 (ja) * 2005-03-11 2014-01-08 バーテックス ファーマシューティカルズ インコーポレイテッド Atp結合カセットトランスポーターのモジュレーター
US8663694B2 (en) * 2005-03-16 2014-03-04 Takeda Gmbh Taste masked dosage form containing roflumilast
KR100838702B1 (ko) * 2007-02-08 2008-06-16 한국화학연구원 1-[1-(3,4-디알콕시아릴)-피리딜메틸]-1h-피라졸 화합물의제조방법
US20100203146A1 (en) * 2009-02-09 2010-08-12 Callisto Pharmaceuticals, Inc. Intermittent dosing strategy for treating rheumatoid arthritis
EP2736489A4 (en) * 2011-07-28 2015-01-14 Cellworks Res India Private Ltd COMPOSITIONS, METHOD FOR THE PRODUCTION THEREOF, AND METHOD FOR THE TREATMENT OF INFLAMMATORY DISEASES
CN105121439A (zh) 2013-02-19 2015-12-02 辉瑞公司 作为pde4亚型抑制剂用于治疗cns和其他病症的氮杂苯并咪唑化合物
WO2016012896A1 (en) 2014-07-24 2016-01-28 Pfizer Inc. Pyrazolopyrimidine compounds
PL3177624T3 (pl) 2014-08-06 2019-09-30 Pfizer Inc. Związki imidazopirydazynowe
US11977085B1 (en) 2023-09-05 2024-05-07 Elan Ehrlich Date rape drug detection device and method of using same

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1161239E (pt) * 1999-03-10 2005-02-28 Altana Pharma Ag 3-ciclopropilmetoxi-4-difluorometoxi-n-(3,5-dicloropirid-4-il)-benzamida para o tratamento da esclerose multipla

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