JP2005507878A5 - - Google Patents

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Publication number
JP2005507878A5
JP2005507878A5 JP2003526920A JP2003526920A JP2005507878A5 JP 2005507878 A5 JP2005507878 A5 JP 2005507878A5 JP 2003526920 A JP2003526920 A JP 2003526920A JP 2003526920 A JP2003526920 A JP 2003526920A JP 2005507878 A5 JP2005507878 A5 JP 2005507878A5
Authority
JP
Japan
Prior art keywords
cyclopentylamino
pyrimidinyl
pyridin
cyclopentyl
amine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003526920A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005507878A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2002/027251 external-priority patent/WO2003022845A1/en
Publication of JP2005507878A publication Critical patent/JP2005507878A/ja
Publication of JP2005507878A5 publication Critical patent/JP2005507878A5/ja
Pending legal-status Critical Current

Links

JP2003526920A 2001-09-07 2002-08-27 ヘルペス感染症を治療するためのピラゾロ−ピリジン類 Pending JP2005507878A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31820301P 2001-09-07 2001-09-07
PCT/US2002/027251 WO2003022845A1 (en) 2001-09-07 2002-08-27 Pyrazolo-pyridines for the treatment of herpes infections

Publications (2)

Publication Number Publication Date
JP2005507878A JP2005507878A (ja) 2005-03-24
JP2005507878A5 true JP2005507878A5 (enExample) 2005-11-17

Family

ID=23237109

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003526920A Pending JP2005507878A (ja) 2001-09-07 2002-08-27 ヘルペス感染症を治療するためのピラゾロ−ピリジン類

Country Status (7)

Country Link
US (1) US20040214834A1 (enExample)
EP (1) EP1423389B1 (enExample)
JP (1) JP2005507878A (enExample)
AT (1) ATE364043T1 (enExample)
DE (1) DE60220525T2 (enExample)
ES (1) ES2286272T3 (enExample)
WO (1) WO2003022845A1 (enExample)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2245772T3 (es) 2002-03-07 2006-01-16 Smithkline Beecham Corporation Derivados de pirazolopirimidina y pirazolotriazina y composiciones farmaceuticas que los contienen.
US20070155738A1 (en) 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
UA103319C2 (en) 2008-05-06 2013-10-10 Глаксосмитклайн Ллк Thiazole- and oxazole-benzene sulfonamide compounds
EP2402336A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazolopyridine compounds
EP2402335A1 (en) 2010-06-29 2012-01-04 Basf Se Pyrazolopyridine compounds
EP3365340B1 (en) 2015-10-19 2022-08-10 Incyte Corporation Heterocyclic compounds as immunomodulators
HUE060680T2 (hu) 2015-11-19 2023-04-28 Incyte Corp Heterociklusos vegyületek mint immunmodulátorok
MA44075A (fr) 2015-12-17 2021-05-19 Incyte Corp Dérivés de n-phényl-pyridine-2-carboxamide et leur utilisation en tant que modulateurs des interactions protéine/protéine pd-1/pd-l1
ES2844374T3 (es) 2015-12-22 2021-07-22 Incyte Corp Compuestos heterocíclicos como inmunomoduladores
ES2906460T3 (es) 2016-05-06 2022-04-18 Incyte Corp Compuestos heterocíclicos como inmunomoduladores
WO2017205464A1 (en) 2016-05-26 2017-11-30 Incyte Corporation Heterocyclic compounds as immunomodulators
HUE060256T2 (hu) 2016-06-20 2023-02-28 Incyte Corp Heterociklusos vegyületek mint immunmodulátorok
EP3484866B1 (en) 2016-07-14 2022-09-07 Incyte Corporation Heterocyclic compounds as immunomodulators
MA46045A (fr) 2016-08-29 2021-04-28 Incyte Corp Composés hétérocycliques utilisés comme immunomodulateurs
UA127785C2 (uk) 2016-12-22 2024-01-03 Інсайт Корпорейшн ПОХІДНІ ТЕТРАГІДРОІМІДАЗО[4,5-c]ПІРИДИНУ, ЯКІ ВИКЛИКАЮТЬ ІНТЕРНАЛІЗАЦІЮ PD-L1
WO2018119236A1 (en) 2016-12-22 2018-06-28 Incyte Corporation Triazolo[1,5-a]pyridine derivatives as immunomodulators
GEP20227428B (en) 2016-12-22 2022-10-25 Incyte Corp Heterocyclic compounds as immunomodulators
ES2899402T3 (es) 2016-12-22 2022-03-11 Incyte Corp Derivados de piridina como inmunomoduladores
WO2018119286A1 (en) 2016-12-22 2018-06-28 Incyte Corporation Bicyclic heteroaromatic compounds as immunomodulators
FI4212529T3 (fi) 2018-03-30 2025-04-23 Incyte Corp Heterosyklisiä yhdisteitä immunomodulaattoreina
SMT202300127T1 (it) 2018-05-11 2023-05-12 Incyte Corp Derivati di tetraidro-imidazo[4,5-c]piridina come immunomodulatori di pd-l1
US11753406B2 (en) 2019-08-09 2023-09-12 Incyte Corporation Salts of a PD-1/PD-L1 inhibitor
KR20220075382A (ko) 2019-09-30 2022-06-08 인사이트 코포레이션 면역조절제로서의 피리도[3,2-d]피리미딘 화합물
KR20220101664A (ko) 2019-11-11 2022-07-19 인사이트 코포레이션 Pd-1/pd-l1 억제제의 염 및 결정질 형태
WO2022099075A1 (en) 2020-11-06 2022-05-12 Incyte Corporation Crystalline form of a pd-1/pd-l1 inhibitor
US11780836B2 (en) 2020-11-06 2023-10-10 Incyte Corporation Process of preparing a PD-1/PD-L1 inhibitor
IL302590A (en) 2020-11-06 2023-07-01 Incyte Corp Process for preparing PD-1/PD-L1 inhibitor and salts and crystalline forms thereof

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0151962A3 (en) * 1984-01-25 1985-10-02 Beecham Group Plc Pyrazolopyridine derivatives
GB8404584D0 (en) * 1984-02-22 1984-03-28 Beecham Group Plc Compounds
GB8404586D0 (en) * 1984-02-22 1984-03-28 Beecham Group Plc Compounds
US4925849A (en) * 1987-06-15 1990-05-15 Fujisawa Pharmaceutical Company, Ltd. Pharmaceutically useful pyrazolopyridines
US5155114A (en) * 1989-01-23 1992-10-13 Fujisawa Pharmaceutical Company, Ltd. Method of treatment using pyrazolopyridine compound
GB8901423D0 (en) * 1989-01-23 1989-03-15 Fujisawa Pharmaceutical Co Pyrazolopyridine compound and processes for preparation thereof
AU622330B2 (en) * 1989-06-23 1992-04-02 Takeda Chemical Industries Ltd. Condensed heterocyclic compounds having a nitrogen atom in the bridgehead for use as fungicides
GB9015764D0 (en) * 1990-07-18 1990-09-05 Fujisawa Pharmaceutical Co Pyrazolopyridine compound and processes for preparation thereof
GB9107513D0 (en) * 1991-04-10 1991-05-29 Fujisawa Pharmaceutical Co Pyrazolopyridine compound and processes for preparation thereof
US5300478A (en) * 1993-01-28 1994-04-05 Zeneca Limited Substituted fused pyrazolo compounds
US5552422A (en) * 1995-01-11 1996-09-03 Merck Frosst Canada, Inc. Aryl substituted 5,5 fused aromatic nitrogen compounds as anti-inflammatory agents
AU6111796A (en) * 1995-06-12 1997-01-09 G.D. Searle & Co. Compositions comprising a cyclooxygenase-2 inhibitor and a 5 -lipoxygenase inhibitor
US5700816A (en) * 1995-06-12 1997-12-23 Isakson; Peter C. Treatment of inflammation and inflammation-related disorders with a combination of a cyclooxygenase-2 inhibitor and a leukotriene A4 hydrolase inhibitor
FR2757166B1 (fr) * 1996-12-12 1999-01-29 Rhone Poulenc Rorer Sa Derives du pyrrole, leur preparation et les compositions pharmaceutiques qui les contiennent
WO1998056377A1 (en) * 1997-06-13 1998-12-17 Smithkline Beecham Corporation Novel pyrazole and pyrazoline substituted compounds
TR200101208T2 (tr) * 1998-11-03 2001-10-22 Glaxo Group Limited Seçici COX-2 inhibitörleri olarak pirazolopiridin türevleri
AU2661400A (en) * 1999-02-27 2000-09-21 Glaxo Group Limited Pyrazolopyridines
ATE301653T1 (de) * 2000-12-15 2005-08-15 Glaxo Group Ltd Pyrazolopyridine
DE60112330T2 (de) * 2000-12-15 2006-04-13 Glaxo Group Ltd., Greenford Pyrazolopyridinderivate
ATE274515T1 (de) * 2001-03-08 2004-09-15 Smithkline Beecham Corp Pyrazolopyridinderivate
JP2004525150A (ja) * 2001-03-30 2004-08-19 スミスクライン ビーチャム コーポレーション 治療用化合物としてのピラゾロピリジン類の使用
US7141569B2 (en) * 2001-04-10 2006-11-28 Smithkline Beecham Corporation Antiviral pyrazolopyridine compounds
WO2002088124A2 (en) * 2001-04-27 2002-11-07 Smithkline Beecham Corporation Pyrazolo'1,5-a!pyridine derivatives

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