JP2005507871A - シクロオキシゲナーゼ−２選択的阻害薬およびグルコサミンを含む、疼痛および炎症を治療および予防するための組成物 - Google Patents

シクロオキシゲナーゼ−２選択的阻害薬およびグルコサミンを含む、疼痛および炎症を治療および予防するための組成物 Download PDF

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JP2005507871A
JP2005507871A JP2003520756A JP2003520756A JP2005507871A JP 2005507871 A JP2005507871 A JP 2005507871A JP 2003520756 A JP2003520756 A JP 2003520756A JP 2003520756 A JP2003520756 A JP 2003520756A JP 2005507871 A JP2005507871 A JP 2005507871A
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trifluoromethyl
alkyl
phenyl
group
benzenesulfonamide
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JP2005507871A5 (OSRAM
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プラスキ，スティーヴン・ピー
クンデル，スーザン
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ファルマシア・コーポレーション
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Virology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Molecular Biology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biotechnology (AREA)
  • Reproductive Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
JP2003520756A 2001-08-14 2002-08-13 シクロオキシゲナーゼ−２選択的阻害薬およびグルコサミンを含む、疼痛および炎症を治療および予防するための組成物 Pending JP2005507871A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US31227201P 2001-08-14 2001-08-14
US10/215,816 US20030114418A1 (en) 2001-08-14 2002-08-09 Method for the treatment and prevention of pain and inflammation with glucosamine and a cyclooxygenase-2 selective inhibitor and compositions therefor
PCT/US2002/025674 WO2003015797A1 (en) 2001-08-14 2002-08-13 Compositions for the treatment and prevention of pain and inflammation with a cyclooxygenase-2 selective inhibitor and glucosamine

Publications (2)

Publication Number Publication Date
JP2005507871A true JP2005507871A (ja) 2005-03-24
JP2005507871A5 JP2005507871A5 (OSRAM) 2006-01-05

Family

ID=26910415

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003520756A Pending JP2005507871A (ja) 2001-08-14 2002-08-13 シクロオキシゲナーゼ−２選択的阻害薬およびグルコサミンを含む、疼痛および炎症を治療および予防するための組成物

Country Status (9)

Country Link
US (1) US20030114418A1 (OSRAM)
EP (1) EP1416940A1 (OSRAM)
JP (1) JP2005507871A (OSRAM)
AU (1) AU2002331076A2 (OSRAM)
BR (1) BR0211936A (OSRAM)
CA (1) CA2457453A1 (OSRAM)
MX (1) MXPA04001398A (OSRAM)
PL (1) PL368271A1 (OSRAM)
WO (1) WO2003015797A1 (OSRAM)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0209022D0 (en) * 2002-04-19 2002-05-29 Imp College Innovations Ltd Compounds
US20040127402A1 (en) * 2002-12-27 2004-07-01 Vad Vijay B. Injectible composition and method for treating degenerative animal joints
CN1232256C (zh) * 2003-03-27 2005-12-21 中国人民解放军第三军医大学 N－乙酰氨基葡萄糖在制备治疗自身免疫反应所致的局部损伤或全身症状的药物中的应用
US7259266B2 (en) * 2003-03-31 2007-08-21 Pharmacia Corporation Benzopyran compounds useful for treating inflammatory conditions
US20050009733A1 (en) * 2003-04-22 2005-01-13 Pharmacia Corporation Compositions of a cyclooxygenase-2 selective inhibitor and a potassium ion channel modulator for the treatment of central nervous system damage
US20040229803A1 (en) * 2003-04-22 2004-11-18 Pharmacia Corporation Compositions of a cyclooxygenase-2 selective inhibitor and a potassium ion channel modulator for the treatment of pain, inflammation or inflammation mediated disorders
EA200601648A1 (ru) * 2004-04-07 2007-04-27 Зе Юниверсити Оф Джорджия Рисерч Фаундейшн, Инк. Глюкозамин и общие пролекарства глюкозамин/противовоспалительный агент, композиции и способы
US8034796B2 (en) * 2004-04-07 2011-10-11 The University Of Georgia Research Foundation, Inc. Glucosamine and glucosamine/anti-inflammatory mutual prodrugs, compositions, and methods
CA2551613A1 (en) * 2004-05-21 2005-12-01 Tottori University A composition comprising n-acetyl-d-glucosamine for treatment of wound
JP5031567B2 (ja) * 2004-09-09 2012-09-19 ハワード・フローレイ・インスティテュート・オブ・イクスペリメンタル・フィジオロジー・アンド・メディスン 酵素阻害剤およびその使用
US7335384B2 (en) 2006-03-17 2008-02-26 4K Nutripharma International Nutrient compositions for the treatment and prevention of inflammation and disorders associated therewith
KR20080025900A (ko) * 2006-09-19 2008-03-24 (주) 서울바이오메드 글루코사민 또는 글루코사민 유도체를 포함하는 알레르기성결막염 치료용 조성물 및 이를 사용하여 알레르기성결막염을 치료하는 방법
US20100105634A1 (en) * 2007-03-07 2010-04-29 Cargill, Incorporated Use of glucosamine as a mental and physical stress recovery enhancer and a performance enhancer
NZ585338A (en) 2007-11-19 2012-08-31 Howard Florey Inst Insulin-regulated aminopeptidase (irap) inhibitors and uses thereof
FR2958157B1 (fr) * 2010-04-02 2012-06-29 Libragen Composition cosmetique et pharmaceutique comprenant du n-acetyl-glucosamine-6-phosphate

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IT1044707B (it) * 1968-10-26 1980-04-21 Rotta Research Lab Procedimento per la preparazione di sali di glucosanina e preparati farmaceutici comprendenti detti sali di glucosamina come agenti attivi
RO118291B1 (ro) * 1993-11-30 2003-04-30 Searle & Co Derivati de pirazol 1,3,4,5 - tetrasubstituiti si compozitie farmaceutica care ii contine
US6034256A (en) * 1997-04-21 2000-03-07 G.D. Searle & Co. Substituted benzopyran derivatives for the treatment of inflammation
SE9703693D0 (sv) * 1997-10-10 1997-10-10 Astra Pharma Prod Novel combination
US6706267B1 (en) * 1999-09-14 2004-03-16 Arkion Life Sciences Llc Glucosamine and egg for reducing inflammation
AU1953701A (en) * 1999-12-09 2001-06-18 Bruce Levin Methods and compositions for treatment of inflammatory disease
US20020086070A1 (en) * 2000-03-11 2002-07-04 Kuhrts Eric Hauser Anti-inflammatory and connective tissue repair formulations

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BR0211936A (pt) 2004-10-26
WO2003015797A1 (en) 2003-02-27
US20030114418A1 (en) 2003-06-19
CA2457453A1 (en) 2003-02-27
MXPA04001398A (es) 2004-05-27
PL368271A1 (en) 2005-03-21
WO2003015797A8 (en) 2004-12-29
AU2002331076A2 (en) 2003-03-03
EP1416940A1 (en) 2004-05-12

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