JP2004536843A - ピオグリタゾンおよびビグアナイドを含むコア製剤 - Google Patents
ピオグリタゾンおよびビグアナイドを含むコア製剤 Download PDFInfo
- Publication number
- JP2004536843A JP2004536843A JP2003511802A JP2003511802A JP2004536843A JP 2004536843 A JP2004536843 A JP 2004536843A JP 2003511802 A JP2003511802 A JP 2003511802A JP 2003511802 A JP2003511802 A JP 2003511802A JP 2004536843 A JP2004536843 A JP 2004536843A
- Authority
- JP
- Japan
- Prior art keywords
- core
- glucopyranosyl
- metformin
- alpha
- drug
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/501—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Inorganic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/US2001/021615 WO2003005995A1 (fr) | 2001-07-10 | 2001-07-10 | Preparation de noyau comprenant un hydrochlorure de pioglitazone et un biguanide |
Publications (1)
Publication Number | Publication Date |
---|---|
JP2004536843A true JP2004536843A (ja) | 2004-12-09 |
Family
ID=21742689
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2003511802A Pending JP2004536843A (ja) | 2001-07-10 | 2001-07-10 | ピオグリタゾンおよびビグアナイドを含むコア製剤 |
Country Status (6)
Country | Link |
---|---|
EP (1) | EP1429747A4 (fr) |
JP (1) | JP2004536843A (fr) |
AU (1) | AU2001273289B2 (fr) |
CA (1) | CA2453775A1 (fr) |
MX (1) | MXPA04000180A (fr) |
WO (1) | WO2003005995A1 (fr) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1429732A4 (fr) * | 2001-07-10 | 2005-01-26 | Kos Life Sciences Inc | Formulation de noyau |
EP1552832A1 (fr) * | 2002-07-11 | 2005-07-13 | Takeda Pharmaceutical Company Limited | Procede de production d'une preparation recouverte |
EP1588708A4 (fr) | 2003-01-29 | 2006-03-01 | Takeda Pharmaceutical | Procede pour realiser une preparation enrobee |
GB0316940D0 (en) * | 2003-07-19 | 2003-08-27 | Ward Warren | Treatment of skin and other medical conditions |
CA2532344A1 (fr) | 2003-07-19 | 2005-02-17 | Warren Ward | Compositions comprenant des composants enrobes d'une couche permeable aux gaz mais impermeables aux liquides, leur utilisation pour le traitement d'affections de la peau et de la glande exocrine |
WO2005021542A2 (fr) * | 2003-08-28 | 2005-03-10 | Ranbaxy Laboratories Limited | Procede pour la preparation de pioglitazone |
US20060153889A1 (en) * | 2005-01-10 | 2006-07-13 | Friel Francis M | Discontinuous surface coating for particles |
MXPA05014092A (es) * | 2005-12-20 | 2007-06-20 | Leopoldo De Jesus Espinosa Abdala | Composiciones farmaceuticas que comprenden sustancias derivadas de la tiazolidinedionas combinadas con una biguanida para su uso en diabetes mellitus tipo 2. |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW438587B (en) * | 1995-06-20 | 2001-06-07 | Takeda Chemical Industries Ltd | A pharmaceutical composition for prophylaxis and treatment of diabetes |
US6416774B1 (en) * | 1996-05-09 | 2002-07-09 | The Trustees Of The University Of Pennsyvania | Hollow bone mineral-like calcium phosphate particles |
US6011049A (en) * | 1997-02-19 | 2000-01-04 | Warner-Lambert Company | Combinations for diabetes |
GB9715295D0 (en) * | 1997-07-18 | 1997-09-24 | Smithkline Beecham Plc | Novel method of treatment |
US6358531B1 (en) * | 1999-02-01 | 2002-03-19 | The Curators Of The University Of Missouri | Method for preparing porous shells or gels from glass particles |
US6451342B2 (en) * | 2000-05-01 | 2002-09-17 | Aeropharm Technology Incorporated | Core formulation comprised of troglitazone and a biguanide |
US6780432B1 (en) * | 2000-05-01 | 2004-08-24 | Aeropharm Technology, Inc. | Core formulation |
EP1429732A4 (fr) * | 2001-07-10 | 2005-01-26 | Kos Life Sciences Inc | Formulation de noyau |
-
2001
- 2001-07-10 MX MXPA04000180A patent/MXPA04000180A/es unknown
- 2001-07-10 JP JP2003511802A patent/JP2004536843A/ja active Pending
- 2001-07-10 CA CA002453775A patent/CA2453775A1/fr not_active Abandoned
- 2001-07-10 WO PCT/US2001/021615 patent/WO2003005995A1/fr not_active Application Discontinuation
- 2001-07-10 AU AU2001273289A patent/AU2001273289B2/en not_active Ceased
- 2001-07-10 EP EP01952548A patent/EP1429747A4/fr not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
MXPA04000180A (es) | 2004-11-22 |
EP1429747A1 (fr) | 2004-06-23 |
CA2453775A1 (fr) | 2003-01-23 |
AU2001273289B2 (en) | 2004-10-07 |
WO2003005995A1 (fr) | 2003-01-23 |
EP1429747A4 (fr) | 2005-01-05 |
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