JP2004526725A5 - - Google Patents

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Publication number
JP2004526725A5
JP2004526725A5 JP2002571445A JP2002571445A JP2004526725A5 JP 2004526725 A5 JP2004526725 A5 JP 2004526725A5 JP 2002571445 A JP2002571445 A JP 2002571445A JP 2002571445 A JP2002571445 A JP 2002571445A JP 2004526725 A5 JP2004526725 A5 JP 2004526725A5
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JP
Japan
Prior art keywords
optionally substituted
represented
alkyl
methyl
structural formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002571445A
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English (en)
Japanese (ja)
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JP2004526725A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2002/007718 external-priority patent/WO2002072528A1/en
Publication of JP2004526725A publication Critical patent/JP2004526725A/ja
Publication of JP2004526725A5 publication Critical patent/JP2004526725A5/ja
Pending legal-status Critical Current

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JP2002571445A 2001-03-14 2002-03-12 フッ化トリエンおよびrxrモジュレータとしてのその使用 Pending JP2004526725A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27580801P 2001-03-14 2001-03-14
PCT/US2002/007718 WO2002072528A1 (en) 2001-03-14 2002-03-12 Fluorinated trienes and their use as rxr modulators

Publications (2)

Publication Number Publication Date
JP2004526725A JP2004526725A (ja) 2004-09-02
JP2004526725A5 true JP2004526725A5 (https=) 2005-12-22

Family

ID=23053886

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002571445A Pending JP2004526725A (ja) 2001-03-14 2002-03-12 フッ化トリエンおよびrxrモジュレータとしてのその使用

Country Status (7)

Country Link
US (1) US20040248919A1 (https=)
EP (1) EP1368296A1 (https=)
JP (1) JP2004526725A (https=)
AU (1) AU2002255732B2 (https=)
CA (1) CA2438874A1 (https=)
MX (1) MXPA03008229A (https=)
WO (1) WO2002072528A1 (https=)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE158816T1 (de) 1990-11-26 1997-10-15 Genetics Inst Expression von pace in wirtszellen und verfahren zu dessen verwendung
MXPA04000613A (es) * 2001-07-20 2004-05-05 Ligand Pharm Inc DERIVADOS DE aCIDO PIRIDINILO Y PIRIMIDILTRIENOICO COMO MODULADORES DE RECEPTOR DE RETINOIDE X.
GB0308335D0 (en) 2003-04-10 2003-05-14 Novartis Ag Organic compounds
US6887896B1 (en) * 2003-10-29 2005-05-03 Allergan, Inc. 7-[(7-Alkoxy)-chrom-3-en-6-yl]-heptatrienoic acid and 7-[(3-alkoxy)-5,6-dihydronaphthalen-2-yl]-heptatrienoic acid derivatives having serum glucose reducing activity
CN1882327A (zh) 2003-11-19 2006-12-20 症变治疗公司 含磷的新的拟甲状腺素药
MX2007014502A (es) 2005-05-26 2008-02-07 Metabasis Therapeutics Inc Tiromimeticos para el tratamiento de enfermedades del higado graso.
WO2009035673A1 (en) 2007-09-12 2009-03-19 Trustees Of Columbia University In The City Of Newyork Compositions and methods for treating macular degeneration
JP6723752B2 (ja) * 2015-02-10 2020-07-15 公益財団法人相模中央化学研究所 二次電池用電解液
JP2020500199A (ja) 2016-11-21 2020-01-09 バイキング・セラピューティクス・インコーポレイテッド グリコーゲン蓄積症の治療方法
AU2018280118B2 (en) 2017-06-05 2021-07-15 Viking Therapeutics, Inc. Compositions for the treatment of fibrosis
ES3053674T3 (en) 2018-03-22 2026-01-23 Viking Therapeutics Inc Crystalline forms and methods of producing crystalline forms of a compound
WO2020117962A1 (en) 2018-12-05 2020-06-11 Viking Therapeutics, Inc. Compositions for the treatment of fibrosis and inflammation

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5071773A (en) * 1986-10-24 1991-12-10 The Salk Institute For Biological Studies Hormone receptor-related bioassays
US4981784A (en) * 1987-12-02 1991-01-01 The Salk Institute For Biological Studies Retinoic acid receptor method
US5977125A (en) * 1994-10-31 1999-11-02 Eisai Co., Ltd. Mono-or polyenic carboxylic acid derivatives
CA2204616C (en) * 1995-09-18 2002-12-17 Ranjan Mukherjee Ppar gamma antagonists for treating obesity
WO1997012853A1 (en) * 1995-10-06 1997-04-10 Ligand Pharmaceuticals Incorporated Dimer-selective rxr modulators and methods for their use
AU9556298A (en) * 1998-11-03 2000-05-22 Ligand Pharmaceuticals Incorporated Trienoic retinoid compounds as retinoic acid receptor antagonists
AU762492B2 (en) * 1999-03-08 2003-06-26 Basilea Pharmaceutica Ag Retinoid antagonists and use thereof
AU7586600A (en) * 1999-09-14 2001-04-17 Ligand Pharmaceuticals Incorporated Rxr modulators with improved pharmacologic profile
MXPA04000613A (es) * 2001-07-20 2004-05-05 Ligand Pharm Inc DERIVADOS DE aCIDO PIRIDINILO Y PIRIMIDILTRIENOICO COMO MODULADORES DE RECEPTOR DE RETINOIDE X.

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