JP2004526675A5 - - Google Patents

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Publication number
JP2004526675A5
JP2004526675A5 JP2002546541A JP2002546541A JP2004526675A5 JP 2004526675 A5 JP2004526675 A5 JP 2004526675A5 JP 2002546541 A JP2002546541 A JP 2002546541A JP 2002546541 A JP2002546541 A JP 2002546541A JP 2004526675 A5 JP2004526675 A5 JP 2004526675A5
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JP
Japan
Prior art keywords
methyl
furan
phenylamino
acetic acid
chloro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2002546541A
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English (en)
Japanese (ja)
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JP2004526675A (ja
JP4340063B2 (ja
Filing date
Publication date
Priority claimed from DE10059864A external-priority patent/DE10059864A1/de
Application filed filed Critical
Publication of JP2004526675A publication Critical patent/JP2004526675A/ja
Publication of JP2004526675A5 publication Critical patent/JP2004526675A5/ja
Application granted granted Critical
Publication of JP4340063B2 publication Critical patent/JP4340063B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2002546541A 2000-11-30 2001-11-28 置換されたアミノ−フラン−2−イル−酢酸−及び置換されたアミノ−チエン−2−イル−酢酸−誘導体及びこれを偏頭痛又は苦痛の治療に使用する方法 Expired - Fee Related JP4340063B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10059864A DE10059864A1 (de) 2000-11-30 2000-11-30 Substituierte Amino-furan-2-yl-essigsäure- und Amino-thien-2-yl-essigsäure-Derivate
PCT/EP2001/013910 WO2002044171A1 (de) 2000-11-30 2001-11-28 Substituierte amino-furan-2-yl-essigsaure- und amino-thien-2-yl-essigsaure-derivate und ihre verwendung zur behandlung von migraine bzw. schmerz

Publications (3)

Publication Number Publication Date
JP2004526675A JP2004526675A (ja) 2004-09-02
JP2004526675A5 true JP2004526675A5 (https=) 2009-02-12
JP4340063B2 JP4340063B2 (ja) 2009-10-07

Family

ID=7665508

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002546541A Expired - Fee Related JP4340063B2 (ja) 2000-11-30 2001-11-28 置換されたアミノ−フラン−2−イル−酢酸−及び置換されたアミノ−チエン−2−イル−酢酸−誘導体及びこれを偏頭痛又は苦痛の治療に使用する方法

Country Status (29)

Country Link
US (1) US6797712B2 (https=)
EP (1) EP1341786B9 (https=)
JP (1) JP4340063B2 (https=)
KR (1) KR20030055334A (https=)
CN (1) CN1326854C (https=)
AR (1) AR035658A1 (https=)
AT (1) ATE418552T1 (https=)
AU (2) AU2073502A (https=)
BR (1) BR0115883A (https=)
CA (1) CA2430280A1 (https=)
CY (1) CY1108871T1 (https=)
CZ (1) CZ20031509A3 (https=)
DE (2) DE10059864A1 (https=)
DK (1) DK1341786T3 (https=)
EC (1) ECSDI034631S (https=)
ES (1) ES2320198T3 (https=)
HU (1) HUP0303041A3 (https=)
IL (2) IL156139A0 (https=)
MX (1) MXPA03004303A (https=)
NO (1) NO20032340L (https=)
NZ (1) NZ526554A (https=)
PE (1) PE20020599A1 (https=)
PL (1) PL362978A1 (https=)
PT (1) PT1341786E (https=)
RU (1) RU2003117703A (https=)
SI (1) SI1341786T1 (https=)
SK (1) SK5942003A3 (https=)
WO (1) WO2002044171A1 (https=)
ZA (1) ZA200305009B (https=)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6794506B2 (en) * 2000-07-21 2004-09-21 Elan Pharmaceuticals, Inc. 3-(heteroaryl) alanine derivatives-inhibitors of leukocyte adhesion mediated by VLA-4
DE10125145A1 (de) 2001-05-22 2002-11-28 Gruenenthal Gmbh Substituierte C-Furan-2-yl-methylamin- und C-Thiophen-2-yl-methylamin-Derivate
GB0302094D0 (en) 2003-01-29 2003-02-26 Pharmagene Lab Ltd EP4 receptor antagonists
DE10306203A1 (de) 2003-02-13 2004-08-26 Grünenthal GmbH Arzneimittel enthaltend substituierte 2-Heteroaryl-Aminoessigsäure-Verbindungen
DE10306202A1 (de) * 2003-02-13 2004-08-26 Grünenthal GmbH Arzneimittel enthaltend substituierte 2-Aryl-Aminoessigsäure-Verbindungen und/oder substituierte 2-Heteroaryl-Aminoessigsäure-Verbindungen
GB0324269D0 (en) * 2003-10-16 2003-11-19 Pharmagene Lab Ltd EP4 receptor antagonists
WO2008009079A2 (en) * 2006-07-20 2008-01-24 Gilead Sciences, Inc. Substituted pteridines useful for the treatment and prevention of viral infections
US9259426B2 (en) 2006-07-20 2016-02-16 Gilead Sciences, Inc. 4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for treating viral infections
WO2016141092A1 (en) 2015-03-04 2016-09-09 Gilead Sciences, Inc. Toll-like receptor modulating 4,6-diamino-pyrido[3,2-d]pyrimidine compounds
EP3507288B1 (en) 2016-09-02 2020-08-26 Gilead Sciences, Inc. 4,6-diamino-pyrido[3,2-d]pyrimidine derivaties as toll like receptor modulators
CN109923106B (zh) 2016-09-02 2022-09-13 吉利德科学公司 toll样受体调节剂化合物
TW202212339A (zh) 2019-04-17 2022-04-01 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TW202210480A (zh) 2019-04-17 2022-03-16 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TWI879779B (zh) 2019-06-28 2025-04-11 美商基利科學股份有限公司 類鐸受體調節劑化合物的製備方法
CN115382297B (zh) * 2022-04-12 2023-10-31 江阴市华思诚无纺布有限公司 熔体直纺双组分pet纺粘液体过滤材料及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU3718397A (en) * 1996-06-28 1998-01-21 University Of Southern California Method for the synthesis of amines and amino acids with organoboron derivatives
US6441237B1 (en) 1999-02-20 2002-08-27 Boehringer Ingelheim Pharma Kg Substituted 3-phenoxy- and 3-phenylalkyloxy-2-phenyl-propylamines
DE19907385A1 (de) * 1999-02-20 2000-08-24 Boehringer Ingelheim Pharma Neue substituierte 3-Phenoxy- und 3-Phenylalkyloxy-2-phenyl-propylamine
GB0030304D0 (en) * 2000-12-13 2001-01-24 Lilly Co Eli Compounds

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