JP2004525140A - ガンの治療方法及び該治療方法に使用する組成物 - Google Patents
ガンの治療方法及び該治療方法に使用する組成物 Download PDFInfo
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/44—Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
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| US27843501P | 2001-03-26 | 2001-03-26 | |
| CA 2342472 CA2342472A1 (en) | 2001-03-30 | 2001-03-30 | Ram having dynamically switchable addressing modes |
| PCT/AU2002/000339 WO2002076454A1 (en) | 2001-03-26 | 2002-03-20 | Method for treatment of cancer and compositions for use therein |
Publications (2)
| Publication Number | Publication Date |
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| JP2004525140A true JP2004525140A (ja) | 2004-08-19 |
| JP2004525140A5 JP2004525140A5 (enExample) | 2006-01-05 |
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| JP2002574969A Pending JP2004525140A (ja) | 2001-03-26 | 2002-03-20 | ガンの治療方法及び該治療方法に使用する組成物 |
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| Country | Link |
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| US (1) | US20050038022A1 (enExample) |
| EP (1) | EP1379242B1 (enExample) |
| JP (1) | JP2004525140A (enExample) |
| WO (1) | WO2002076454A1 (enExample) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2008511549A (ja) * | 2004-08-31 | 2008-04-17 | ニューサウス・イノベイションズ・プロプライエタリー・リミテッド | Ｖｅｇｆ阻害剤 |
| JP2009510033A (ja) * | 2005-09-27 | 2009-03-12 | アバンテイス・フアルマ・エス・アー | 新規ベンゾイミダゾール及びベンゾチアゾール誘導体、その調製方法、薬物としてのその使用、薬剤組成物、並びに特にｃ−ｍｅｔ阻害剤としての新規使用 |
| WO2018003829A1 (ja) * | 2016-06-29 | 2018-01-04 | 国立大学法人東京大学 | オートファジー阻害剤 |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20020164715A1 (en) | 2000-07-10 | 2002-11-07 | Lin Ji | Chromosome 3p21.3 genes are tumor suppressors |
| WO2002067932A1 (en) | 2001-01-11 | 2002-09-06 | Board Of Regents, The University Of Texas System | Antihelminthic drugs as a treatment for hyperproliferative diseases |
| WO2004041277A1 (en) | 2002-11-01 | 2004-05-21 | Merck & Co., Inc. | Carbonylamino-benzimidazole derivatives as androgen receptor modulators |
| BRPI0413234A (pt) * | 2003-08-01 | 2006-10-03 | Genelabs Tech Inc | derivados de imidazola bicìclica contra flaviviridae |
| EP1723138B1 (en) * | 2004-02-11 | 2010-07-14 | Basilea Pharmaceutica AG | Substituted benzimidazoles and their use for inducing apoptosis |
| FR2868421B1 (fr) | 2004-04-01 | 2008-08-01 | Aventis Pharma Sa | Nouveaux benzothiazoles et leur utilisation comme medicaments |
| ES2528363T3 (es) | 2004-12-06 | 2015-02-09 | Pitney Pharmaceuticals Pty Limited | Tratamiento para el cáncer |
| CN101103026A (zh) * | 2005-01-14 | 2008-01-09 | 健亚生物科技公司 | 用于治疗病毒感染的吲哚衍生物 |
| TW200720255A (en) * | 2005-07-13 | 2007-06-01 | Taiho Pharmaceutical Co Ltd | Benzoimidazole compound capable of inhibiting prostaglandin d synthetase |
| PE20070335A1 (es) * | 2005-08-30 | 2007-04-21 | Novartis Ag | Benzimidazoles sustituidos y metodos para su preparacion |
| WO2009043093A1 (en) * | 2007-10-04 | 2009-04-09 | Newsouth Innovations Pty Limited | Hif inhibition |
| WO2009148623A2 (en) | 2008-06-05 | 2009-12-10 | Stc.Unm | Methods and related compositions for the treatment of cancer |
| WO2010135534A2 (en) * | 2009-05-20 | 2010-11-25 | Children's Medical Center Corporation | Compositions for the treatment of metastatic cancer and methods of use thereof |
| JP2013520502A (ja) | 2010-02-25 | 2013-06-06 | メルク・シャープ・エンド・ドーム・コーポレイション | 有用な抗糖尿病薬である新規な環状ベンズイミダゾール誘導体 |
| EP3383852A4 (en) * | 2015-11-30 | 2019-08-28 | Children's Medical Center Corporation | COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISEASES |
| GB2559162A (en) * | 2017-01-27 | 2018-08-01 | Univ Bradford | Compound for use in medicine |
| TW202214245A (zh) * | 2020-08-10 | 2022-04-16 | 國立彰化師範大學 | 雙非癌藥物用於製備治療癌症之醫藥組合物的用途 |
| CN113648308A (zh) * | 2021-09-14 | 2021-11-16 | 东莞市人民医院 | 奥芬达唑作为抗卵巢癌药物的应用 |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1998056387A1 (en) * | 1997-06-10 | 1998-12-17 | Unisearch Limited | Method of treatment of liver tumours and pharmaceutical compositions for use therein |
| WO1999056697A2 (en) * | 1998-05-04 | 1999-11-11 | Unisearch Limited | Pharmaceutical composition |
| WO2000041669A2 (en) * | 1999-01-15 | 2000-07-20 | Angiogene Pharmaceuticals Ltd. | Benzimidazole vascular damaging agents |
| WO2001012169A2 (en) * | 1999-08-13 | 2001-02-22 | The Procter & Gamble Company | Method of cancer treatment |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA962879B (en) * | 1995-04-12 | 1997-03-17 | Procter & Gamble | A pharmaceutical composition for inhibiting the growth of viruses and cancers |
| CA2344316A1 (en) * | 1998-09-16 | 2000-03-23 | Saira Sayed Singh | Treatment of oncologic tumors with an injectable formulation of a golgi apparatus disturbing agent |
| MXPA02002360A (es) * | 1999-09-03 | 2002-07-30 | Janssen Pharmaceutica Nv | Formulacion veterinaria para administracion de un farmaco insoluble en agua a un animal objetivo mediante un sistema de distribucion de agua. |
| US6693125B2 (en) * | 2001-01-24 | 2004-02-17 | Combinatorx Incorporated | Combinations of drugs (e.g., a benzimidazole and pentamidine) for the treatment of neoplastic disorders |
-
2002
- 2002-03-20 EP EP02713920A patent/EP1379242B1/en not_active Expired - Lifetime
- 2002-03-20 WO PCT/AU2002/000339 patent/WO2002076454A1/en not_active Ceased
- 2002-03-20 US US10/472,888 patent/US20050038022A1/en not_active Abandoned
- 2002-03-20 JP JP2002574969A patent/JP2004525140A/ja active Pending
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1998056387A1 (en) * | 1997-06-10 | 1998-12-17 | Unisearch Limited | Method of treatment of liver tumours and pharmaceutical compositions for use therein |
| WO1999056697A2 (en) * | 1998-05-04 | 1999-11-11 | Unisearch Limited | Pharmaceutical composition |
| WO2000041669A2 (en) * | 1999-01-15 | 2000-07-20 | Angiogene Pharmaceuticals Ltd. | Benzimidazole vascular damaging agents |
| WO2001012169A2 (en) * | 1999-08-13 | 2001-02-22 | The Procter & Gamble Company | Method of cancer treatment |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2008511549A (ja) * | 2004-08-31 | 2008-04-17 | ニューサウス・イノベイションズ・プロプライエタリー・リミテッド | Ｖｅｇｆ阻害剤 |
| JP2009510033A (ja) * | 2005-09-27 | 2009-03-12 | アバンテイス・フアルマ・エス・アー | 新規ベンゾイミダゾール及びベンゾチアゾール誘導体、その調製方法、薬物としてのその使用、薬剤組成物、並びに特にｃ−ｍｅｔ阻害剤としての新規使用 |
| WO2018003829A1 (ja) * | 2016-06-29 | 2018-01-04 | 国立大学法人東京大学 | オートファジー阻害剤 |
Also Published As
| Publication number | Publication date |
|---|---|
| US20050038022A1 (en) | 2005-02-17 |
| EP1379242B1 (en) | 2012-08-15 |
| EP1379242A1 (en) | 2004-01-14 |
| EP1379242A4 (en) | 2007-10-03 |
| WO2002076454A1 (en) | 2002-10-03 |
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