JP2004517943A5 - - Google Patents

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Publication number
JP2004517943A5
JP2004517943A5 JP2002561044A JP2002561044A JP2004517943A5 JP 2004517943 A5 JP2004517943 A5 JP 2004517943A5 JP 2002561044 A JP2002561044 A JP 2002561044A JP 2002561044 A JP2002561044 A JP 2002561044A JP 2004517943 A5 JP2004517943 A5 JP 2004517943A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2002561044A
Other versions
JP2004517943A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2002/000831 external-priority patent/WO2002060895A1/en
Publication of JP2004517943A publication Critical patent/JP2004517943A/ja
Publication of JP2004517943A5 publication Critical patent/JP2004517943A5/ja
Withdrawn legal-status Critical Current

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JP2002561044A 2001-01-31 2002-01-26 ジアゾシン誘導体およびトリプターゼインヒビターとしてのその使用 Withdrawn JP2004517943A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01102098 2001-01-31
PCT/EP2002/000831 WO2002060895A1 (en) 2001-01-31 2002-01-26 Diazocine derivatives and their use as tryptase inhibitors

Publications (2)

Publication Number Publication Date
JP2004517943A JP2004517943A (ja) 2004-06-17
JP2004517943A5 true JP2004517943A5 (ja) 2005-12-22

Family

ID=8176347

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002561044A Withdrawn JP2004517943A (ja) 2001-01-31 2002-01-26 ジアゾシン誘導体およびトリプターゼインヒビターとしてのその使用

Country Status (12)

Country Link
US (1) US6924305B2 (ja)
EP (1) EP1358182B1 (ja)
JP (1) JP2004517943A (ja)
AT (1) ATE273302T1 (ja)
AU (1) AU2002238522B8 (ja)
CA (1) CA2438594A1 (ja)
DE (1) DE60200935T2 (ja)
DK (1) DK1358182T3 (ja)
ES (1) ES2225758T3 (ja)
PT (1) PT1358182E (ja)
SI (1) SI1358182T1 (ja)
WO (1) WO2002060895A1 (ja)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002102771A1 (en) 2001-06-19 2002-12-27 Altana Pharma Ag Tryptase inhibitors
WO2006044133A1 (en) * 2004-09-24 2006-04-27 Axys Pharmaceuticals, Inc. Active ketone inhibitors of tryptase

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995032945A1 (en) 1994-06-01 1995-12-07 Arris Pharmaceutical Corporation Compositions and methods for treating mast-cell mediated conditions
WO1996009297A1 (en) * 1994-09-23 1996-03-28 Arris Pharmaceutical Corporation Compositions and methods for treating mast-cell inflammatory condition
HUP0003267A3 (en) * 1996-07-30 2002-02-28 Arris Pharmaceutical Corp San Heteroaryl derivatives, pharmaceutical compositions containing them and process for producing them
AU8997498A (en) 1997-09-05 1999-03-29 Yoshitomi Pharmaceutical Industries, Ltd. Tryptase inhibitor
EP1030844A1 (en) 1997-11-10 2000-08-30 Array Biopharma Inc. Compounds which inhibit tryptase activity
US6221914B1 (en) 1997-11-10 2001-04-24 Array Biopharma Inc. Sulfonamide bridging compounds that inhibit tryptase activity
ATE282607T1 (de) 1998-02-06 2004-12-15 Max Planck Gesellschaft Tryptase-inhibitoren
JP2002502845A (ja) 1998-02-06 2002-01-29 マックス−プランク−ゲゼルシャフト・ツア・フェルデルング・デア・ヴィッセンシャフテン・エー・ファオ トリプターゼ阻害物質
WO2000014097A2 (de) 1998-09-04 2000-03-16 Byk Gulden Lomberg Chemische Fabrik Gmbh Neue pyranosen
DE19937721A1 (de) 1999-08-10 2001-02-15 Max Planck Gesellschaft Neue Diketopiperazine
SI1208089T1 (en) 1999-08-10 2005-04-30 Altana Pharma Ag Diazocin-dione derivatives and their use as tryptase inhibitors
WO2001019809A1 (en) 1999-09-14 2001-03-22 Byk Gulden Lomberg Chemische Fabrik Gmbh Tryptase inhibitors
CA2392121A1 (en) 1999-12-20 2001-06-28 Byk Gulden Lomberg Chemische Fabrik Gmbh Tryptase inhibitors
CA2392127A1 (en) 1999-12-20 2001-06-28 Byk Gulden Lomberg Chemische Fabrik Gmbh Tryptase inhibitors

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