JP2004514002A - 新規ポリエステル、その製法および前記ポリエステルから製造されるデポー剤 - Google Patents

新規ポリエステル、その製法および前記ポリエステルから製造されるデポー剤 Download PDF

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Publication number
JP2004514002A
JP2004514002A JP2002541975A JP2002541975A JP2004514002A JP 2004514002 A JP2004514002 A JP 2004514002A JP 2002541975 A JP2002541975 A JP 2002541975A JP 2002541975 A JP2002541975 A JP 2002541975A JP 2004514002 A JP2004514002 A JP 2004514002A
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JP
Japan
Prior art keywords
polyester
extruder
electrolyte
hydroxycarboxylic acid
resorbable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002541975A
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English (en)
Japanese (ja)
Other versions
JP2004514002A5 (https=
Inventor
ユクシン　リ
デトレフ　モア
ティム　ザイフェルト
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
UCB Pharma GmbH
Original Assignee
Schwarz Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schwarz Pharma AG filed Critical Schwarz Pharma AG
Publication of JP2004514002A publication Critical patent/JP2004514002A/ja
Publication of JP2004514002A5 publication Critical patent/JP2004514002A5/ja
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08G—MACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
    • C08G63/00—Macromolecular compounds obtained by reactions forming a carboxylic ester link in the main chain of the macromolecule
    • C08G63/02—Polyesters derived from hydroxycarboxylic acids or from polycarboxylic acids and polyhydroxy compounds
    • C08G63/06—Polyesters derived from hydroxycarboxylic acids or from polycarboxylic acids and polyhydroxy compounds derived from hydroxycarboxylic acids
    • C08G63/08—Lactones or lactides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08G—MACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
    • C08G63/00—Macromolecular compounds obtained by reactions forming a carboxylic ester link in the main chain of the macromolecule
    • C08G63/78—Preparation processes
    • C08G63/82—Preparation processes characterised by the catalyst used
    • C08G63/823—Preparation processes characterised by the catalyst used for the preparation of polylactones or polylactides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Polymers & Plastics (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Polyesters Or Polycarbonates (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
JP2002541975A 2000-11-10 2001-11-08 新規ポリエステル、その製法および前記ポリエステルから製造されるデポー剤 Pending JP2004514002A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10055742A DE10055742B4 (de) 2000-11-10 2000-11-10 Neue Polyester, Verfahren zu ihrer Herstellung und aus den Polyestern hergestellte Depot-Arzneiformen
PCT/EP2001/012888 WO2002038646A2 (de) 2000-11-10 2001-11-08 Neue polyester, verfahren zu ihrer herstellung und aus den polyestern hergestellte depot-arzneiformen

Publications (2)

Publication Number Publication Date
JP2004514002A true JP2004514002A (ja) 2004-05-13
JP2004514002A5 JP2004514002A5 (https=) 2005-05-26

Family

ID=7662818

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002541975A Pending JP2004514002A (ja) 2000-11-10 2001-11-08 新規ポリエステル、その製法および前記ポリエステルから製造されるデポー剤

Country Status (8)

Country Link
US (1) US7087247B2 (https=)
EP (1) EP1345979B1 (https=)
JP (1) JP2004514002A (https=)
AT (1) ATE271083T1 (https=)
AU (1) AU2002229539A1 (https=)
DE (2) DE10055742B4 (https=)
ES (1) ES2225636T3 (https=)
WO (1) WO2002038646A2 (https=)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008513524A (ja) * 2004-09-21 2008-05-01 山▲東緑▼叶制▲薬▼有限公司 ドーパミン受容体アゴニストを含む長時間作用する持続放出製剤、及びそれらの製造方法
WO2024166833A1 (ja) * 2023-02-08 2024-08-15 Ｓｐｉｂｅｒ株式会社 ブロック共重合体もしくはこれを含有する水分散液、接着剤、塗液、コーティング剤、又は成形体の製造方法

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1074923C (zh) 1993-11-19 2001-11-21 詹森药业有限公司 微囊密封的3-哌啶基取代的1,2-苯并异唑类和1,2-苯并异噻唑类
CN100443546C (zh) * 2000-04-12 2008-12-17 三光化学工业株式会社 抗静电组合物
DE10041478A1 (de) 2000-08-24 2002-03-14 Sanol Arznei Schwarz Gmbh Neue pharmazeutische Zusammensetzung
DE10041479A1 (de) * 2000-08-24 2002-03-14 Sanol Arznei Schwarz Gmbh Neue pharmazeutische Zusammensetzung zur Verabreichung von N-0923
DE10055857A1 (de) * 2000-11-10 2002-08-22 Creative Peptides Sweden Ab Dj Neue pharmazeutische Depotformulierung
DE10334188B4 (de) 2003-07-26 2007-07-05 Schwarz Pharma Ag Verwendung von Rotigotin zur Behandlung von Depressionen
DE10361258A1 (de) 2003-12-24 2005-07-28 Schwarz Pharma Ag Verwendung von substituierten 2-Aminotetralinen zur vorbeugenden Behandlung von Morbus Parkinson
DE102004014841B4 (de) 2004-03-24 2006-07-06 Schwarz Pharma Ag Verwendung von Rotigotin zur Behandlung und Prävention des Parkinson-Plus-Syndroms
KR101297937B1 (ko) 2006-07-14 2013-08-19 킴벌리-클라크 월드와이드, 인크. 부직 웹에 사용하기 위한 생분해성 지방족 폴리에스테르
MX2009000527A (es) 2006-07-14 2009-01-27 Kimberly Clark Co Acido polilactico biodegradable para su uso en telas no tejidas.
DE602006018078D1 (de) 2006-07-14 2010-12-16 Kimberly Clark Co Biologisch abbaubarer aliphatisch-aromatischer copolyester zur verwendung in vliesstoffen
CA2659012A1 (en) * 2006-07-26 2008-01-31 Diamedica Inc. Methods of diagnosis and treatment for metabolic disorders
KR101422317B1 (ko) 2007-08-22 2014-07-30 킴벌리-클라크 월드와이드, 인크. 다성분 생분해성 필라멘트 및 그로부터 형성되는 부직 웹
MX2010013139A (es) 2008-05-30 2011-03-04 Kimberly Clark Worldwide Incorporated Fibras de acido polilactico.
CA2798518A1 (en) 2010-05-17 2011-11-24 Cebix, Inc. Pegylated c-peptide
US8461262B2 (en) 2010-12-07 2013-06-11 Kimberly-Clark Worldwide, Inc. Polylactic acid fibers
EP2559435A1 (en) 2011-08-19 2013-02-20 UCB Pharma GmbH Rotigotine in the treatment of hemispatial neglect, stroke and deficits following stroke
US20130315891A1 (en) 2012-05-25 2013-11-28 Matthew Charles Formulations of human tissue kallikrein-1 for parenteral delivery and related methods
EP2854841B1 (en) 2012-06-04 2017-02-22 Diamedica Inc. Human tissue kallikrein 1 glycosylation isoforms
DE102014005782A1 (de) * 2014-04-23 2015-10-29 Martin-Luther-Universität Halle-Wittenberg lnjizierbare und implantierbare Trägersysteme auf Basis von modifizierten Poly(dikarbonsäure-multiol estern) zur kontrollierten Wirkstofffreisetzung
CN110446501A (zh) 2017-03-09 2019-11-12 代阿麦迪卡股份有限公司 组织激肽释放酶1的剂型

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US3773919A (en) 1969-10-23 1973-11-20 Du Pont Polylactide-drug mixtures
IE52535B1 (en) 1981-02-16 1987-12-09 Ici Plc Continuous release pharmaceutical compositions
ATE37983T1 (de) 1982-04-22 1988-11-15 Ici Plc Mittel mit verzoegerter freigabe.
CH656884A5 (de) 1983-08-26 1986-07-31 Sandoz Ag Polyolester, deren herstellung und verwendung.
US4726076A (en) 1985-06-26 1988-02-23 Francoise Douez Childs garment
JPH0613602B2 (ja) 1987-07-14 1994-02-23 三井東圧化学株式会社 ｄ▲ｌ▼−乳酸−グリコール酸共重合物の製造方法
EP0372221B1 (de) 1988-11-01 2000-01-19 Boehringer Ingelheim Pharma KG Kontinuierliches Verfahren zur Herstellung von resorbierbaren Polyestern und deren Verwendung
CA2025893A1 (en) 1989-01-27 1990-07-28 Hosei Shinoda Biocompatible polyester and production thereof
DE4406172C2 (de) * 1994-02-25 2003-10-02 Sanol Arznei Schwarz Gmbh Polyester
JP3307777B2 (ja) * 1994-07-07 2002-07-24 栄修 永田 ハンダ付け方法および装置
US6046882A (en) * 1996-07-11 2000-04-04 International Business Machines Corporation Solder balltape and method for making electrical connection between a head transducer and an electrical lead
US6595408B1 (en) * 1998-10-07 2003-07-22 Micron Technology, Inc. Method of attaching solder balls to BGA package utilizing a tool to pick and dip the solder ball in flux prior to placement
US6336581B1 (en) * 2000-06-19 2002-01-08 International Business Machines Corporation Solder ball connection device and capillary tube thereof
JP2002025025A (ja) * 2000-06-23 2002-01-25 Internatl Business Mach Corp <Ibm> はんだボール接合装置及びはんだボール接合方法
US6589594B1 (en) * 2000-08-31 2003-07-08 Micron Technology, Inc. Method for filling a wafer through-via with a conductive material
JP2002251705A (ja) * 2001-02-16 2002-09-06 Internatl Business Mach Corp <Ibm> はんだボール配設装置、はんだボールリフロー装置、及びはんだボール接合装置。
DE10132567B4 (de) * 2001-07-10 2005-03-31 Pac Tech - Packaging Technologies Gmbh Verfahren und Vorrichtung zum Aufbringen eines Lötmittels auf ein Substrat
JP3753968B2 (ja) * 2001-10-11 2006-03-08 ヒタチグローバルストレージテクノロジーズネザーランドビーブイ 配線一体型サスペンション及びその製造方法
JP4212992B2 (ja) * 2003-09-03 2009-01-21 Ｔｄｋ株式会社 半田ボールの供給方法および供給装置

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008513524A (ja) * 2004-09-21 2008-05-01 山▲東緑▼叶制▲薬▼有限公司 ドーパミン受容体アゴニストを含む長時間作用する持続放出製剤、及びそれらの製造方法
WO2024166833A1 (ja) * 2023-02-08 2024-08-15 Ｓｐｉｂｅｒ株式会社 ブロック共重合体もしくはこれを含有する水分散液、接着剤、塗液、コーティング剤、又は成形体の製造方法

Also Published As

Publication number Publication date
ES2225636T3 (es) 2005-03-16
EP1345979A2 (de) 2003-09-24
WO2002038646A2 (de) 2002-05-16
DE50102886D1 (de) 2004-08-19
EP1345979B1 (de) 2004-07-14
US20040072986A1 (en) 2004-04-15
DE10055742A1 (de) 2002-05-29
WO2002038646A3 (de) 2002-08-01
US7087247B2 (en) 2006-08-08
AU2002229539A1 (en) 2002-05-21
ATE271083T1 (de) 2004-07-15
DE10055742B4 (de) 2006-05-11

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