JP2003533469A - 口腔及び経肺投与用ミセル薬学的組成物 - Google Patents
口腔及び経肺投与用ミセル薬学的組成物Info
- Publication number
- JP2003533469A JP2003533469A JP2001583737A JP2001583737A JP2003533469A JP 2003533469 A JP2003533469 A JP 2003533469A JP 2001583737 A JP2001583737 A JP 2001583737A JP 2001583737 A JP2001583737 A JP 2001583737A JP 2003533469 A JP2003533469 A JP 2003533469A
- Authority
- JP
- Japan
- Prior art keywords
- composition
- micelle
- alkali metal
- acid
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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- NOOLISFMXDJSKH-UTLUCORTSA-N (+)-Neomenthol Chemical compound CC(C)[C@@H]1CC[C@@H](C)C[C@@H]1O NOOLISFMXDJSKH-UTLUCORTSA-N 0.000 claims description 10
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Classifications
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/008—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy comprising drug dissolved or suspended in liquid propellant for inhalation via a pressurized metered dose inhaler [MDI]
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Organic Chemistry (AREA)
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- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
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- Otolaryngology (AREA)
- Emergency Medicine (AREA)
- Tropical Medicine & Parasitology (AREA)
- Endocrinology (AREA)
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- Obesity (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/574,504 | 2000-05-19 | ||
| US09/574,504 US6451286B1 (en) | 1998-12-21 | 2000-05-19 | Pharmaceutical compositions for buccal and pulmonary administration comprising an alkali metal alkyl sulfate and at least three micelle-forming compounds |
| PCT/CA2001/000661 WO2001087268A1 (en) | 2000-05-19 | 2001-05-07 | Micellar pharmaceutical compositions for buccal and pulmonary application |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| JP2011157744A Division JP2012006934A (ja) | 2000-05-19 | 2011-07-19 | 口腔及び経肺投与用ミセル薬学的組成物 |
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| JP2003533469A true JP2003533469A (ja) | 2003-11-11 |
| JP2003533469A5 JP2003533469A5 (https=) | 2008-07-03 |
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| JP2001583737A Pending JP2003533469A (ja) | 2000-05-19 | 2001-05-07 | 口腔及び経肺投与用ミセル薬学的組成物 |
| JP2011157744A Withdrawn JP2012006934A (ja) | 2000-05-19 | 2011-07-19 | 口腔及び経肺投与用ミセル薬学的組成物 |
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| JP2011157744A Withdrawn JP2012006934A (ja) | 2000-05-19 | 2011-07-19 | 口腔及び経肺投与用ミセル薬学的組成物 |
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| Country | Link |
|---|---|
| US (1) | US6451286B1 (https=) |
| EP (1) | EP1296648A1 (https=) |
| JP (2) | JP2003533469A (https=) |
| AU (1) | AU2001258112A1 (https=) |
| CA (1) | CA2410065C (https=) |
| MX (1) | MXPA02011436A (https=) |
| NZ (1) | NZ522524A (https=) |
| WO (1) | WO2001087268A1 (https=) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013527189A (ja) * | 2010-05-28 | 2013-06-27 | ノヴォ ノルディスク アー／エス | 抗体及び防腐剤を含む安定した多用量組成物 |
| US9795674B2 (en) | 2010-02-26 | 2017-10-24 | Novo Nordisk A/S | Stable antibody containing compositions |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7087215B2 (en) * | 1998-12-21 | 2006-08-08 | Generex Pharmaceuticals Incorporated | Methods of administering and enhancing absorption of pharmaceutical agents |
| US6849263B2 (en) * | 1998-12-21 | 2005-02-01 | Generex Pharmaceutical Incorporated | Pharmaceutical compositions for buccal delivery of pain relief medications |
| DE10007771A1 (de) * | 2000-02-14 | 2001-08-23 | Kleine & Steube Entoxin Gmbh | Immunmodulatorisch wirksame Zusammensetzungen, Verfahren zu ihrer Herstellung und ihre Verwendung |
| WO2003097094A1 (en) * | 2002-05-21 | 2003-11-27 | Anadis Ltd | Method of prophylaxis of infection |
| EP1369113B1 (en) * | 2002-06-06 | 2006-11-22 | CHIESI FARMACEUTICI S.p.A. | Solubilisation of drugs in HFA propellant by means of emulsions |
| US20050238632A1 (en) * | 2004-04-23 | 2005-10-27 | Alburty David S | Propellant formulations |
| ES2660172T3 (es) * | 2004-05-19 | 2018-03-21 | Los Angeles Biomedical Research Institute At Harbor-Ucla Medical Center | Composición inyectable que comprende desoxicolato de sodio |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9795674B2 (en) | 2010-02-26 | 2017-10-24 | Novo Nordisk A/S | Stable antibody containing compositions |
| US10709782B2 (en) | 2010-02-26 | 2020-07-14 | Novo Nordisk A/S | Stable antibody containing compositions |
| JP2013527189A (ja) * | 2010-05-28 | 2013-06-27 | ノヴォ ノルディスク アー／エス | 抗体及び防腐剤を含む安定した多用量組成物 |
| JP2018030879A (ja) * | 2010-05-28 | 2018-03-01 | ノヴォ ノルディスク アー／エス | 抗体及び防腐剤を含む安定した多用量組成物 |
| US10835602B2 (en) | 2010-05-28 | 2020-11-17 | Novo Nordisk A/S | Stable multi-dose compositions comprising an antibody and a preservative |
Also Published As
| Publication number | Publication date |
|---|---|
| CA2410065A1 (en) | 2001-11-22 |
| CA2410065C (en) | 2009-04-07 |
| WO2001087268A1 (en) | 2001-11-22 |
| AU2001258112A1 (en) | 2001-11-26 |
| JP2012006934A (ja) | 2012-01-12 |
| MXPA02011436A (es) | 2003-06-06 |
| US6451286B1 (en) | 2002-09-17 |
| EP1296648A1 (en) | 2003-04-02 |
| NZ522524A (en) | 2003-07-25 |
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