JP2003523995A - フェニルヘテロアルキルアミン誘導体の新規なる使用 - Google Patents

フェニルヘテロアルキルアミン誘導体の新規なる使用

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Publication number
JP2003523995A
JP2003523995A JP2001561730A JP2001561730A JP2003523995A JP 2003523995 A JP2003523995 A JP 2003523995A JP 2001561730 A JP2001561730 A JP 2001561730A JP 2001561730 A JP2001561730 A JP 2001561730A JP 2003523995 A JP2003523995 A JP 2003523995A
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JP
Japan
Prior art keywords
formula
compound
alkyl
pharmaceutically acceptable
alkoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2001561730A
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English (en)
Japanese (ja)
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JP2003523995A5 (enExample
Inventor
デイビッド・チェシャー
スティーブン・コノリー
デイビッド・コックス
イアン・ミリチップ
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AstraZeneca AB
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AstraZeneca AB
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Publication of JP2003523995A publication Critical patent/JP2003523995A/ja
Publication of JP2003523995A5 publication Critical patent/JP2003523995A5/ja
Withdrawn legal-status Critical Current

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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
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    • C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C323/31—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
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    • C07C323/24—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/29—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
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  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Epidemiology (AREA)
  • Neurosurgery (AREA)
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  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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  • Hospice & Palliative Care (AREA)
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  • Anesthesiology (AREA)
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JP2001561730A 2000-02-23 2001-02-20 フェニルヘテロアルキルアミン誘導体の新規なる使用 Withdrawn JP2003523995A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0004151.7A GB0004151D0 (en) 2000-02-23 2000-02-23 Novel use
GB0004151.7 2000-02-23
PCT/SE2001/000371 WO2001062721A1 (en) 2000-02-23 2001-02-20 Novel use of phenylheteroalkylamine derivatives

Publications (2)

Publication Number Publication Date
JP2003523995A true JP2003523995A (ja) 2003-08-12
JP2003523995A5 JP2003523995A5 (enExample) 2008-04-03

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JP2001561730A Withdrawn JP2003523995A (ja) 2000-02-23 2001-02-20 フェニルヘテロアルキルアミン誘導体の新規なる使用

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US (1) US6953797B2 (enExample)
EP (1) EP1263718B1 (enExample)
JP (1) JP2003523995A (enExample)
KR (1) KR100721087B1 (enExample)
CN (1) CN1210270C (enExample)
AT (1) ATE265428T1 (enExample)
AU (1) AU780781B2 (enExample)
BR (1) BR0108539A (enExample)
CA (1) CA2396960A1 (enExample)
CO (1) CO5660084A1 (enExample)
DE (1) DE60103035T2 (enExample)
GB (1) GB0004151D0 (enExample)
IL (1) IL150640A0 (enExample)
MX (1) MXPA02008204A (enExample)
NO (1) NO20024013L (enExample)
WO (1) WO2001062721A1 (enExample)
ZA (1) ZA200205801B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0004152D0 (en) 2000-02-23 2000-04-12 Astrazeneca Uk Ltd Novel compounds
AR035700A1 (es) * 2001-05-08 2004-06-23 Astrazeneca Ab Derivados de arilheteroalquilamina, composicion farmaceutica, usos de estos derivados para la fabricacion de medicamentos, metodos de tratamiento, y proceso para la preparacion de estos derivados
WO2002100848A1 (en) * 2001-06-12 2002-12-19 Sk Corporation Novel phenylalkyl diamine and amide analogs
SE0102640D0 (sv) 2001-07-31 2001-07-31 Astrazeneca Ab Novel compounds
SE0203304D0 (sv) * 2002-11-07 2002-11-07 Astrazeneca Ab Novel Coumpounds

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US6953797B2 (en) 2005-10-11
CA2396960A1 (en) 2001-08-30
DE60103035T2 (de) 2005-03-24
NO20024013D0 (no) 2002-08-22
ATE265428T1 (de) 2004-05-15
EP1263718A1 (en) 2002-12-11
BR0108539A (pt) 2002-10-22
GB0004151D0 (en) 2000-04-12
KR20020091096A (ko) 2002-12-05
KR100721087B1 (ko) 2007-05-23
NO20024013L (no) 2002-09-06
CN1404468A (zh) 2003-03-19
MXPA02008204A (es) 2002-11-29
ZA200205801B (en) 2003-10-20
AU780781B2 (en) 2005-04-14
WO2001062721A1 (en) 2001-08-30
EP1263718B1 (en) 2004-04-28
US20030073685A1 (en) 2003-04-17
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CN1210270C (zh) 2005-07-13

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