JP2003501109A - μＯ−コノペプチドおよび局所麻酔剤としてのその使用 - Google Patents
μＯ−コノペプチドおよび局所麻酔剤としてのその使用Info
- Publication number
- JP2003501109A JP2003501109A JP2001502865A JP2001502865A JP2003501109A JP 2003501109 A JP2003501109 A JP 2003501109A JP 2001502865 A JP2001502865 A JP 2001502865A JP 2001502865 A JP2001502865 A JP 2001502865A JP 2003501109 A JP2003501109 A JP 2003501109A
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- Prior art keywords
- xaa
- tyr
- cys
- lys
- ile
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/43504—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from invertebrates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
- A61P23/02—Local anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Anesthesiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Zoology (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Tropical Medicine & Parasitology (AREA)
- Toxicology (AREA)
- Engineering & Computer Science (AREA)
- Gastroenterology & Hepatology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US13850799P | 1999-06-10 | 1999-06-10 | |
| US60/138,507 | 1999-06-10 | ||
| PCT/US2000/015779 WO2000076532A1 (en) | 1999-06-10 | 2000-06-09 | νO-CONOPEPTIDES AND THEIR USE AS LOCAL ANESTHETICS |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2003501109A true JP2003501109A (ja) | 2003-01-14 |
| JP2003501109A5 JP2003501109A5 (enExample) | 2007-07-05 |
Family
ID=22482336
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001502865A Pending JP2003501109A (ja) | 1999-06-10 | 2000-06-09 | μＯ−コノペプチドおよび局所麻酔剤としてのその使用 |
Country Status (5)
| Country | Link |
|---|---|
| EP (1) | EP1185286A4 (enExample) |
| JP (1) | JP2003501109A (enExample) |
| AU (1) | AU5474200A (enExample) |
| CA (1) | CA2376357A1 (enExample) |
| WO (1) | WO2000076532A1 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2740401A (en) | 1999-12-30 | 2001-07-16 | Cognetix, Inc. | O-superfamily conotoxin peptides |
| GB0011202D0 (en) * | 2000-05-09 | 2000-06-28 | Kci Licensing Inc | Abdominal wound dressing |
| WO2002007756A1 (en) * | 2000-07-20 | 2002-01-31 | Cognetix, Inc. | MuO-CONOPEPTIDES AND THEIR USE AS LOCAL ANESTHETICS |
| JP2004537253A (ja) * | 2000-07-21 | 2004-12-16 | ユニバーシティ・オブ・ユタ・リサーチ・ファウンデーション | ミュー−コノペプチド |
| DK2051991T3 (da) * | 2006-08-17 | 2012-01-30 | Eribis Pharmaceuticals Ab | Cardiobeskyttende forbindelser |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH11503909A (ja) * | 1995-04-17 | 1999-04-06 | ユニバーシティ・オブ・ユタ・リサーチ・ファウンデーション | コノトキシンペプチド |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5719264A (en) * | 1994-10-07 | 1998-02-17 | Univ. Of Utah Research Foundation | Conotoxin peptides |
| FR2785613B1 (fr) * | 1998-11-10 | 2001-01-05 | Commissariat Energie Atomique | Conotoxine isolee a partir du venin de conus ermineus, ses analogues et ses applications |
-
2000
- 2000-06-09 AU AU54742/00A patent/AU5474200A/en not_active Abandoned
- 2000-06-09 EP EP00939692A patent/EP1185286A4/en not_active Withdrawn
- 2000-06-09 CA CA002376357A patent/CA2376357A1/en not_active Abandoned
- 2000-06-09 JP JP2001502865A patent/JP2003501109A/ja active Pending
- 2000-06-09 WO PCT/US2000/015779 patent/WO2000076532A1/en not_active Ceased
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH11503909A (ja) * | 1995-04-17 | 1999-04-06 | ユニバーシティ・オブ・ユタ・リサーチ・ファウンデーション | コノトキシンペプチド |
Non-Patent Citations (3)
| Title |
|---|
| JPN6010012355, 生体の科学 （１９９８） ｖｏｌ．４９， ｎｏ．５， ｐ．４３３−４３６ * |
| JPN6010012358, Ｔｏｘｉｃｏｌ． Ｌｅｔｔ． （１９９８） ｖｏｌ．１００−１０１， ｐ．２４７−２５４ * |
| JPN6010012362, Ｊ． Ｂｉｏｌ． Ｃｈｅｍ． （１９９５） ｖｏｌ．２７０， ｎｏ．２８， ｐ．１６７９６−１６８０２ * |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2000076532A1 (en) | 2000-12-21 |
| AU5474200A (en) | 2001-01-02 |
| EP1185286A1 (en) | 2002-03-13 |
| EP1185286A4 (en) | 2004-09-08 |
| CA2376357A1 (en) | 2000-12-21 |
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