JP2002523450A - ニトロソ化およびニトロシル化されたホスホジエステラーゼ阻害剤、組成物および使用方法 - Google Patents
ニトロソ化およびニトロシル化されたホスホジエステラーゼ阻害剤、組成物および使用方法Info
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- JP2002523450A JP2002523450A JP2000567194A JP2000567194A JP2002523450A JP 2002523450 A JP2002523450 A JP 2002523450A JP 2000567194 A JP2000567194 A JP 2000567194A JP 2000567194 A JP2000567194 A JP 2000567194A JP 2002523450 A JP2002523450 A JP 2002523450A
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- Pending
Links
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/145,142 US5958926A (en) | 1996-11-01 | 1998-09-01 | Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses |
| US09/145,142 | 1998-09-01 | ||
| PCT/US1999/020024 WO2000012076A1 (en) | 1998-09-01 | 1999-09-01 | Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2002523450A true JP2002523450A (ja) | 2002-07-30 |
| JP2002523450A5 JP2002523450A5 (enExample) | 2006-10-19 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000567194A Pending JP2002523450A (ja) | 1998-09-01 | 1999-09-01 | ニトロソ化およびニトロシル化されたホスホジエステラーゼ阻害剤、組成物および使用方法 |
Country Status (6)
| Country | Link |
|---|---|
| US (11) | US5958926A (enExample) |
| EP (1) | EP1109543A4 (enExample) |
| JP (1) | JP2002523450A (enExample) |
| AU (1) | AU773269B2 (enExample) |
| CA (1) | CA2339189A1 (enExample) |
| WO (1) | WO2000012076A1 (enExample) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2013518851A (ja) * | 2010-02-05 | 2013-05-23 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング | ｓＧＣ刺激剤又はｓＧＣ活性化剤単独及びＰＤＥ５阻害剤と組合せた嚢胞性線維症処置 |
| JP2020520945A (ja) * | 2017-05-22 | 2020-07-16 | トパドゥール ファーマ アーゲー | 新規二重作用モード可溶性グアニル酸シクラーゼ活性化因子およびホスホジエステラーゼ阻害剤ならびにその使用 |
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| US6476037B1 (en) * | 2000-03-23 | 2002-11-05 | The Regents Of The University Of California | L-arginine and phosphodiesterase (PDE) inhibitor synergism |
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Cited By (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013518851A (ja) * | 2010-02-05 | 2013-05-23 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング | ｓＧＣ刺激剤又はｓＧＣ活性化剤単独及びＰＤＥ５阻害剤と組合せた嚢胞性線維症処置 |
| JP2016155857A (ja) * | 2010-02-05 | 2016-09-01 | アドヴェリオ・ファーマ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング | 嚢胞性線維症処置用のｓＧＣ刺激剤又はｓＧＣ活性化剤単独及びＰＤＥ５阻害剤との組み合わせ物 |
| JP2020520945A (ja) * | 2017-05-22 | 2020-07-16 | トパドゥール ファーマ アーゲー | 新規二重作用モード可溶性グアニル酸シクラーゼ活性化因子およびホスホジエステラーゼ阻害剤ならびにその使用 |
| JP7182568B2 (ja) | 2017-05-22 | 2022-12-02 | トパドゥール ファーマ アーゲー | 新規二重作用モード可溶性グアニル酸シクラーゼ活性化因子およびホスホジエステラーゼ阻害剤ならびにその使用 |
| US11905293B2 (en) | 2017-05-22 | 2024-02-20 | Topadur Pharma Ag | Dual mode of action soluble guanylate cyclase activators and phosphodiesterase inhibitors and uses thereof |
Also Published As
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|---|---|
| AU6133499A (en) | 2000-03-21 |
| US6197778B1 (en) | 2001-03-06 |
| US5958926A (en) | 1999-09-28 |
| WO2000012076A1 (en) | 2000-03-09 |
| US6211179B1 (en) | 2001-04-03 |
| US6197782B1 (en) | 2001-03-06 |
| US6316457B1 (en) | 2001-11-13 |
| US6221881B1 (en) | 2001-04-24 |
| US6232321B1 (en) | 2001-05-15 |
| CA2339189A1 (en) | 2000-03-09 |
| AU773269B2 (en) | 2004-05-20 |
| US6172068B1 (en) | 2001-01-09 |
| US6133272A (en) | 2000-10-17 |
| EP1109543A1 (en) | 2001-06-27 |
| WO2000012076A9 (en) | 2000-08-17 |
| US6177428B1 (en) | 2001-01-23 |
| US6172060B1 (en) | 2001-01-09 |
| EP1109543A4 (en) | 2006-03-08 |
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