JP2002356471A5 - - Google Patents

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Publication number
JP2002356471A5
JP2002356471A5 JP2001309558A JP2001309558A JP2002356471A5 JP 2002356471 A5 JP2002356471 A5 JP 2002356471A5 JP 2001309558 A JP2001309558 A JP 2001309558A JP 2001309558 A JP2001309558 A JP 2001309558A JP 2002356471 A5 JP2002356471 A5 JP 2002356471A5
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JP
Japan
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group
substituted
lower alkyl
cyano
trans
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JP2001309558A
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Japanese (ja)
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JP2002356471A (ja
JP4329290B2 (ja
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Publication of JP2002356471A5 publication Critical patent/JP2002356471A5/ja
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JP2001309558A 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物 Expired - Fee Related JP4329290B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2001309558A JP4329290B2 (ja) 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
JP2000308528 2000-10-06
JP2000-308528 2000-10-06
JP2000-312562 2000-10-12
JP2000312562 2000-10-12
JP2001-99251 2001-03-30
JP2001099251 2001-03-30
JP2001309558A JP4329290B2 (ja) 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物

Related Child Applications (1)

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JP2003368572A Division JP2004035574A (ja) 2000-10-06 2003-10-29 脂肪族含窒素五員環化合物

Publications (3)

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JP2002356471A JP2002356471A (ja) 2002-12-13
JP2002356471A5 true JP2002356471A5 (US07816364-20101019-C00135.png) 2004-10-28
JP4329290B2 JP4329290B2 (ja) 2009-09-09

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JP2001309558A Expired - Fee Related JP4329290B2 (ja) 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物

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JP (1) JP4329290B2 (US07816364-20101019-C00135.png)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7816364B2 (en) 2006-04-11 2010-10-19 Arena Pharmaceuticals, Inc. GRP119 receptor agonists in methods of increasing bone mass and of treating osteoporosis and other conditions characterized by low bone mass, and combination therapy relating thereto
US7833730B2 (en) 2006-04-11 2010-11-16 Arena Pharmaceuticals, Inc. Methods of using GPR119 to identify compounds useful for increasing bone mass in an individual
US8003597B2 (en) 2005-01-10 2011-08-23 Arena Pharmaceuticals, Inc. Combination therapy for the treatment of diabetes and conditions related thereto and for the treatment of conditions ameliorated by increasing a blood GLP-1 level
US8486646B2 (en) 2008-04-07 2013-07-16 Arena Pharmaceuticals, Inc. Methods of using a G protein-coupled receptor to identify peptide YY (PYY) secretagogues

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10213051B4 (de) * 2002-03-23 2013-03-07 Grünenthal GmbH Substituierte 4-Aminocyclohexanole
US20050197350A1 (en) * 2003-03-31 2005-09-08 Taisho Pharmaceutical Co., Ltd. Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof
SI1712547T1 (sl) 2004-02-05 2012-04-30 Kyorin Seiyaku Kk Bicikloestrski derivat
DE102004023632A1 (de) * 2004-05-10 2005-12-08 Grünenthal GmbH Substituierte Cyclohexylcarbonsäure-Derivate
NZ554515A (en) * 2004-10-12 2009-12-24 Glenmark Pharmaceuticals Sa Novel dipeptidyl peptidase IV inhibitors, pharmaceutical compositions containing them, and process for their preparation
CA2645154C (en) 2006-03-08 2011-11-29 Kyorin Pharmaceutical Co., Ltd. Method for producing aminoacetylpyrrolidinecarbonitrile derivative and production intermediate thereof
WO2008066083A1 (fr) * 2006-11-29 2008-06-05 Mitsubishi Tanabe Pharma Corporation Procédé de production d'un dérivé de n-(n'-glycyle substitué)-2-cyanopyrrolidine
ATE550319T1 (de) 2007-03-22 2012-04-15 Kyorin Seiyaku Kk Verfahren zur herstellung eines aminoacetylpyrrolidincarbonitrilderivats
EP2231687A4 (en) * 2008-01-10 2012-11-14 Sun Pharma Advanced Res Co Ltd NEW DERIVATIVES OF ACYL-CYANPYRROLIDINES
EP2322499A4 (en) 2008-08-07 2011-12-21 Kyorin Seiyaku Kk PROCESS FOR PRODUCING A BICYCLOÝ2.2.2¨OCTYLAMINE DERIVATIVE
AR077642A1 (es) 2009-07-09 2011-09-14 Arena Pharm Inc Moduladores del metabolismo y el tratamiento de trastornos relacionados con el mismo
US20130023494A1 (en) 2010-04-06 2013-01-24 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
BR112013008100A2 (pt) 2010-09-22 2016-08-09 Arena Pharm Inc "moduladores do receptor de gpr19 e o tratamento de distúrbios relacionados a eles."
WO2012135570A1 (en) 2011-04-01 2012-10-04 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
US20140066369A1 (en) 2011-04-19 2014-03-06 Arena Pharmaceuticals, Inc. Modulators Of The GPR119 Receptor And The Treatment Of Disorders Related Thereto
WO2012145604A1 (en) 2011-04-22 2012-10-26 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
US20140038889A1 (en) 2011-04-22 2014-02-06 Arena Pharmaceuticals, Inc. Modulators Of The GPR119 Receptor And The Treatment Of Disorders Related Thereto
WO2012170702A1 (en) 2011-06-08 2012-12-13 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2013055910A1 (en) 2011-10-12 2013-04-18 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2014074668A1 (en) 2012-11-08 2014-05-15 Arena Pharmaceuticals, Inc. Modulators of gpr119 and the treatment of disorders related thereto
KR20180006881A (ko) 2015-03-09 2018-01-19 인테크린 테라퓨틱스, 아이엔씨. 비알코올성 지방간 질환 및/또는 지방이영양증의 치료 방법
AU2018249822A1 (en) 2017-04-03 2019-10-31 Coherus Biosciences Inc. PPArgamma agonist for treatment of progressive supranuclear palsy
KR102614814B1 (ko) * 2017-05-15 2023-12-20 카그니션 테라퓨틱스, 인코퍼레이티드 신경변성 질환 치료용 조성물

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8003597B2 (en) 2005-01-10 2011-08-23 Arena Pharmaceuticals, Inc. Combination therapy for the treatment of diabetes and conditions related thereto and for the treatment of conditions ameliorated by increasing a blood GLP-1 level
US8198232B2 (en) 2005-01-10 2012-06-12 Arena Pharmaceuticals, Inc. Combination therapy for the treatment of diabetes and conditions related thereto and for the treatment of conditions ameliorated by increasing a blood GLP-1 level
US7816364B2 (en) 2006-04-11 2010-10-19 Arena Pharmaceuticals, Inc. GRP119 receptor agonists in methods of increasing bone mass and of treating osteoporosis and other conditions characterized by low bone mass, and combination therapy relating thereto
US7833730B2 (en) 2006-04-11 2010-11-16 Arena Pharmaceuticals, Inc. Methods of using GPR119 to identify compounds useful for increasing bone mass in an individual
US8580526B2 (en) 2006-04-11 2013-11-12 Arena Pharmaceuticals, Inc. Methods of using GPR119 receptor to identify compounds which stimulate glucose-dependent insulinotropic peptide secretion
US8486646B2 (en) 2008-04-07 2013-07-16 Arena Pharmaceuticals, Inc. Methods of using a G protein-coupled receptor to identify peptide YY (PYY) secretagogues

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