JP2001524931A5 - - Google Patents
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- Publication number
- JP2001524931A5 JP2001524931A5 JP1998508118A JP50811898A JP2001524931A5 JP 2001524931 A5 JP2001524931 A5 JP 2001524931A5 JP 1998508118 A JP1998508118 A JP 1998508118A JP 50811898 A JP50811898 A JP 50811898A JP 2001524931 A5 JP2001524931 A5 JP 2001524931A5
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US69242096A | 1996-08-05 | 1996-08-05 | |
| US08/692,420 | 1996-08-05 | ||
| US72507396A | 1996-10-02 | 1996-10-02 | |
| US08/725,073 | 1996-10-02 | ||
| US79791597A | 1997-02-10 | 1997-02-10 | |
| US08/797,915 | 1997-02-10 | ||
| US4706797P | 1997-05-19 | 1997-05-19 | |
| US60/047,067 | 1997-05-19 | ||
| PCT/US1997/013622 WO1998005333A1 (en) | 1996-08-05 | 1997-08-05 | Use of beta-sheet mimetics as protease and kinase inhibitors and as inhibitors of transcription factors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2001524931A JP2001524931A (ja) | 2001-12-04 |
| JP2001524931A5 true JP2001524931A5 (enExample) | 2005-04-07 |
Family
ID=27489127
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP50811898A Pending JP2001524931A (ja) | 1996-08-05 | 1997-08-05 | プロテアーゼおよびキナーゼのインヒビターとしてならびに転写因子のインヒビターとしてのβシート模倣物の使用 |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP0915700B1 (enExample) |
| JP (1) | JP2001524931A (enExample) |
| KR (1) | KR20000029838A (enExample) |
| AT (1) | ATE320811T1 (enExample) |
| AU (1) | AU732174B2 (enExample) |
| CA (1) | CA2262900A1 (enExample) |
| DE (1) | DE69735545T2 (enExample) |
| ES (1) | ES2262184T3 (enExample) |
| NO (1) | NO990522L (enExample) |
| NZ (1) | NZ334227A (enExample) |
| WO (1) | WO1998005333A1 (enExample) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6184223B1 (en) * | 1995-10-27 | 2001-02-06 | Molecumetics Ltd. | Reverse-turn mimetics and methods relating thereto |
| EP1053246B1 (en) * | 1998-02-12 | 2003-01-02 | Molecumetics, Ltd. | Beta-sheet mimetics and methods relating to the use thereof |
| US6323219B1 (en) | 1998-04-02 | 2001-11-27 | Ortho-Mcneil Pharmaceutical, Inc. | Methods for treating immunomediated inflammatory disorders |
| US8106094B2 (en) | 1998-07-06 | 2012-01-31 | Johnson & Johnson Consumer Companies, Inc. | Compositions and methods for treating skin conditions |
| US8093293B2 (en) | 1998-07-06 | 2012-01-10 | Johnson & Johnson Consumer Companies, Inc. | Methods for treating skin conditions |
| EP1058549A4 (en) | 1998-12-23 | 2003-11-12 | Bristol Myers Squibb Pharma Co | FACTOR Xa OR THROMBIN INHIBITORS |
| CA2361479A1 (en) | 1999-01-27 | 2000-08-03 | Ortho-Mcneil Pharmaceutical, Inc. | Peptidyl heterocyclic ketones useful as tryptase inhibitors |
| US7309688B2 (en) | 2000-10-27 | 2007-12-18 | Johnson & Johnson Consumer Companies | Topical anti-cancer compositions and methods of use thereof |
| US6417189B1 (en) * | 1999-11-12 | 2002-07-09 | Gpi Nil Holdings, Inc. | AZA compounds, pharmaceutical compositions and methods of use |
| US7253169B2 (en) | 1999-11-12 | 2007-08-07 | Gliamed, Inc. | Aza compounds, pharmaceutical compositions and methods of use |
| AU2001245356A1 (en) * | 2000-02-29 | 2001-09-12 | Bristol-Myers Squibb Pharma Company | Inhibitors of hepatitis c virus ns3 protease |
| US8431550B2 (en) | 2000-10-27 | 2013-04-30 | Johnson & Johnson Consumer Companies, Inc. | Topical anti-cancer compositions and methods of use thereof |
| DE10100053A1 (de) * | 2001-01-02 | 2002-08-22 | Keyneurotek Ag I G | Verwendung von Enzyminhibitoren der Dipeptidylpeptidase IV sowie der Aminopeptidase N und pharmazeutischen Zubereitungen daraus zur Prävention und/oder Therapie Ischämie-bedingter akuter und chronischer neurodegenerativer Prozesse und Erkrankungen |
| US7192615B2 (en) | 2001-02-28 | 2007-03-20 | J&J Consumer Companies, Inc. | Compositions containing legume products |
| US8080657B2 (en) | 2001-10-12 | 2011-12-20 | Choongwae Pharma Corporation | Compounds of reverse turn mimetics and the use thereof |
| US7232822B2 (en) | 2001-10-12 | 2007-06-19 | Choongwae Pharma Corporation | Reverse-turn mimetics and method relating thereto |
| US7566711B2 (en) | 2001-10-12 | 2009-07-28 | Choongwae Pharma Corporation | Reverse-turn mimetics and method relating thereto |
| US7576084B2 (en) | 2001-10-12 | 2009-08-18 | Choongwae Pharma Corporation | Reverse-turn mimetics and method relating thereto |
| US7671054B1 (en) | 2001-10-12 | 2010-03-02 | Choongwae Pharma Corporation | Reverse-turn mimetics and method relating thereto |
| WO2003055856A2 (en) | 2001-10-17 | 2003-07-10 | Bristol-Myers Squibb Company | BICYCLIC LACTAM DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-α CONVERTING ENZYME (TACE) |
| TWI286476B (en) * | 2001-12-12 | 2007-09-11 | Tibotec Pharm Ltd | Combination of cytochrome P450 dependent protease inhibitors |
| WO2004035587A1 (en) | 2002-10-17 | 2004-04-29 | Myriad Genetics, Inc. | Reverse-turn mimetics and composition and methods relating thereto |
| JPWO2011096440A1 (ja) * | 2010-02-03 | 2013-06-10 | 株式会社 ＰＲＩＳＭ ＢｉｏＬａｂ | 天然変性タンパク質に結合する化合物およびそのスクリーニング方法 |
| CA2963305A1 (en) | 2014-10-06 | 2016-04-14 | Cortexyme, Inc. | Inhibitors of lysine gingipain |
| CA3004095A1 (en) | 2015-11-09 | 2017-05-18 | Cortexyme, Inc. | Inhibitors of arginine gingipain |
| CA3036862A1 (en) | 2016-09-16 | 2018-03-22 | Cortexyme, Inc. | Ketone inhibitors of lysine gingipain |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1600880A (en) * | 1978-05-23 | 1981-10-21 | Lilly Industries Ltd | Pharmaceutical compositions comprising hydantoin derivatives |
| IL60617A0 (en) * | 1979-07-23 | 1980-09-16 | Sparamedica Ag | Triazolopyridazine derivative,their preparation and pharmaceutical compositions containing them |
| US4594431A (en) * | 1983-08-01 | 1986-06-10 | Eli Lilly Company | Octahydroindolizinepropanoic acids and related compounds as enzyme inhibitors |
| JPH0676373B2 (ja) * | 1985-12-27 | 1994-09-28 | エーザイ株式会社 | グアニジノ安息香酸エステル誘導体 |
| AU653024B2 (en) * | 1991-05-30 | 1994-09-15 | Novartis Ag | Substituted diaminophthalimides and analogues |
| US5463063A (en) * | 1993-07-02 | 1995-10-31 | Celgene Corporation | Ring closure of N-phthaloylglutamines |
| US5716929A (en) * | 1994-06-17 | 1998-02-10 | Vertex Pharmaceuticals, Inc. | Inhibitors of interleukin-1β converting enzyme |
| AU4250596A (en) * | 1994-12-22 | 1996-07-10 | Biochem Pharma Inc. | Low molecular weight bicyclic thrombin inhibitors |
| EP0797437B1 (en) * | 1994-12-30 | 2001-04-18 | Celgene Corporation | IMMUNOTHERAPEUTIC IMIDES/AMIDES AND THEIR USE FOR REDUCING LEVELS OF TNFalpha |
| WO1996030396A1 (en) * | 1995-03-24 | 1996-10-03 | Molecumetics Ltd. | β-SHEET MIMETICS AND USE THEREOF AS PROTEASE INHIBITORS |
| CA2215695C (en) * | 1995-03-24 | 2003-09-16 | Molecumetics, Ltd | .beta.-sheet mimetics and use thereof as protease inhibitors |
| IT1277405B1 (it) * | 1995-08-01 | 1997-11-10 | Menarini Farma Ind | Derivati di lattami biciclici come inibitori della trombina |
-
1997
- 1997-08-05 AT AT97936371T patent/ATE320811T1/de not_active IP Right Cessation
- 1997-08-05 DE DE69735545T patent/DE69735545T2/de not_active Expired - Lifetime
- 1997-08-05 AU AU39058/97A patent/AU732174B2/en not_active Ceased
- 1997-08-05 CA CA002262900A patent/CA2262900A1/en not_active Abandoned
- 1997-08-05 JP JP50811898A patent/JP2001524931A/ja active Pending
- 1997-08-05 ES ES97936371T patent/ES2262184T3/es not_active Expired - Lifetime
- 1997-08-05 EP EP97936371A patent/EP0915700B1/en not_active Expired - Lifetime
- 1997-08-05 NZ NZ334227A patent/NZ334227A/xx not_active IP Right Cessation
- 1997-08-05 WO PCT/US1997/013622 patent/WO1998005333A1/en not_active Ceased
- 1997-08-05 KR KR1019997000994A patent/KR20000029838A/ko not_active Ceased
-
1999
- 1999-02-04 NO NO990522A patent/NO990522L/no unknown