JP2001510173A - カルボニル化合物の触媒フッ素化 - Google Patents

カルボニル化合物の触媒フッ素化

Info

Publication number
JP2001510173A
JP2001510173A JP2000503036A JP2000503036A JP2001510173A JP 2001510173 A JP2001510173 A JP 2001510173A JP 2000503036 A JP2000503036 A JP 2000503036A JP 2000503036 A JP2000503036 A JP 2000503036A JP 2001510173 A JP2001510173 A JP 2001510173A
Authority
JP
Japan
Prior art keywords
compound
cycloalkyl
group
alkyl
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2000503036A
Other languages
English (en)
Japanese (ja)
Other versions
JP2001510173A5 (enExample
Inventor
チェンバーズ，リチャード・ディッキンソン
ハッチンソン，ジョン
モイリエット，ジョン・スチュワート
Original Assignee
エフ２・ケミカルズ・リミテッド
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB9715140A external-priority patent/GB9715140D0/en
Priority claimed from GB9715139A external-priority patent/GB9715139D0/en
Priority claimed from GBGB9808777.8A external-priority patent/GB9808777D0/en
Application filed by エフ２・ケミカルズ・リミテッド filed Critical エフ２・ケミカルズ・リミテッド
Publication of JP2001510173A publication Critical patent/JP2001510173A/ja
Publication of JP2001510173A5 publication Critical patent/JP2001510173A5/ja
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C315/00—Preparation of sulfones; Preparation of sulfoxides
    • C07C315/04—Preparation of sulfones; Preparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B39/00—Halogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C201/00—Preparation of esters of nitric or nitrous acid or of compounds containing nitro or nitroso groups bound to a carbon skeleton
    • C07C201/06—Preparation of nitro compounds
    • C07C201/12—Preparation of nitro compounds by reactions not involving the formation of nitro groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/307—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
JP2000503036A 1997-07-18 1998-07-16 カルボニル化合物の触媒フッ素化 Withdrawn JP2001510173A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
GB9715140.1 1997-07-18
GB9715140A GB9715140D0 (en) 1997-07-18 1997-07-18 Fluorination of organic compounds
GB9715139A GB9715139D0 (en) 1997-07-18 1997-07-18 Fluorination of organic compounds
GB9715139.3 1997-07-18
GBGB9808777.8A GB9808777D0 (en) 1998-04-25 1998-04-25 Fluorination of organic compounds
GB9808777.8 1998-04-25
PCT/GB1998/001905 WO1999003802A1 (en) 1997-07-18 1998-07-16 Catalysed fluorination of carbonyl compounds

Publications (2)

Publication Number Publication Date
JP2001510173A true JP2001510173A (ja) 2001-07-31
JP2001510173A5 JP2001510173A5 (enExample) 2006-01-05

Family

ID=27268933

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000503036A Withdrawn JP2001510173A (ja) 1997-07-18 1998-07-16 カルボニル化合物の触媒フッ素化

Country Status (7)

Country Link
US (1) US6300511B1 (enExample)
EP (1) EP0996606B1 (enExample)
JP (1) JP2001510173A (enExample)
AT (1) ATE212008T1 (enExample)
AU (1) AU8346698A (enExample)
DE (1) DE69803186T2 (enExample)
WO (1) WO1999003802A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2006519815A (ja) * 2003-03-07 2006-08-31 サノフィ−アベンティス ピリジニル及びピリミジニルモノフッ素化βケトエステルの製造方法

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013028639A1 (en) * 2011-08-19 2013-02-28 The Trustees Of Princeton University C-halogen bond formation
CN104418739A (zh) * 2013-08-19 2015-03-18 上海元符医药科技有限公司 一种2-氟丙二酸二甲酯(i)的合成方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4929317A (en) 1986-12-01 1990-05-29 Tokuyama Soda Kabushiki Kaisha Process for preparation of perfluoro organic compounds
DE3827436A1 (de) * 1988-08-12 1990-02-15 Bayer Ag Verfahren zum einfuehren von fluoratomen an aromatische kerne durch nucleophilen austausch
EP0781752B1 (en) 1992-10-30 2001-02-21 Daikin Industries, Limited Process for preparing fluorine-containing dicarbonyl compound
WO1995014646A1 (en) * 1993-11-20 1995-06-01 Bnfl Fluorochemicals Ltd The preparation of dicarbonyls

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2006519815A (ja) * 2003-03-07 2006-08-31 サノフィ−アベンティス ピリジニル及びピリミジニルモノフッ素化βケトエステルの製造方法

Also Published As

Publication number Publication date
AU8346698A (en) 1999-02-10
US6300511B1 (en) 2001-10-09
EP0996606A1 (en) 2000-05-03
EP0996606B1 (en) 2002-01-16
ATE212008T1 (de) 2002-02-15
DE69803186D1 (de) 2002-02-21
DE69803186T2 (de) 2002-07-18
WO1999003802A1 (en) 1999-01-28

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