ITMI920940A0 - Benzossazinoni e benzotiazinoni ad attivita' cardiovascolare - Google Patents

Benzossazinoni e benzotiazinoni ad attivita' cardiovascolare

Info

Publication number
ITMI920940A0
ITMI920940A0 IT92MI940A ITMI920940A ITMI920940A0 IT MI920940 A0 ITMI920940 A0 IT MI920940A0 IT 92MI940 A IT92MI940 A IT 92MI940A IT MI920940 A ITMI920940 A IT MI920940A IT MI920940 A0 ITMI920940 A0 IT MI920940A0
Authority
IT
Italy
Prior art keywords
benzothiazinones
benzoxazinones
cardiovascular activity
cardiovascular
activity
Prior art date
Application number
IT92MI940A
Other languages
English (en)
Inventor
Alberto Sala
Roberto Barani
Francesca Benedini
Giorgio Bertolini
Gianni Gromo
Silvio Levi
Original Assignee
Italfarmaco Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Italfarmaco Spa filed Critical Italfarmaco Spa
Publication of ITMI920940A0 publication Critical patent/ITMI920940A0/it
Priority to ITMI920940A priority Critical patent/IT1254884B/it
Priority to ZA932030A priority patent/ZA932030B/xx
Priority to CA002092342A priority patent/CA2092342A1/en
Priority to IL10515893A priority patent/IL105158A/en
Priority to NZ247249A priority patent/NZ247249A/xx
Priority to AU35617/93A priority patent/AU655540B2/en
Priority to NO93931225A priority patent/NO931225L/no
Priority to DE69320087T priority patent/DE69320087T2/de
Priority to AT93105752T priority patent/ATE169293T1/de
Priority to EP93105752A priority patent/EP0566018B1/en
Priority to MX9302165A priority patent/MX9302165A/es
Priority to FI931688A priority patent/FI931688A/fi
Priority to TW082102853A priority patent/TW288013B/zh
Priority to HU9301106A priority patent/HUT68605A/hu
Priority to JP11214993A priority patent/JP3257716B2/ja
Priority to CN 93104624 priority patent/CN1078466A/zh
Publication of ITMI920940A1 publication Critical patent/ITMI920940A1/it
Priority to US08/347,217 priority patent/US5480882A/en
Application granted granted Critical
Publication of IT1254884B publication Critical patent/IT1254884B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/041,3-Oxazines; Hydrogenated 1,3-oxazines
    • C07D265/121,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
    • C07D265/141,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D265/201,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 4
    • C07D265/22Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/041,3-Thiazines; Hydrogenated 1,3-thiazines
    • C07D279/081,3-Thiazines; Hydrogenated 1,3-thiazines condensed with carbocyclic rings or ring systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Control Of Transmission Device (AREA)
  • Optical Filters (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
ITMI920940A 1992-04-16 1992-04-16 Benzossazinoni e benzotiazinoni ad attivita' cardiovascolare IT1254884B (it)

Priority Applications (17)

Application Number Priority Date Filing Date Title
ITMI920940A IT1254884B (it) 1992-04-16 1992-04-16 Benzossazinoni e benzotiazinoni ad attivita' cardiovascolare
ZA932030A ZA932030B (en) 1992-04-16 1993-03-22 Benzoxazinone and benzothiazinone derivatives endowed with cardiovascular activity
CA002092342A CA2092342A1 (en) 1992-04-16 1993-03-24 Benzoxazinone and benzothiazinone derivatives endowed with cardiovascular activity
IL10515893A IL105158A (en) 1992-04-16 1993-03-24 Benzoxazinone and benzothiazinone derivatives having cardiovascular activity
NZ247249A NZ247249A (en) 1992-04-16 1993-03-25 Benzoxazinone and benzothiazinone derivatives; medicaments and use
AU35617/93A AU655540B2 (en) 1992-04-16 1993-03-30 Benzoxazinone and benzothiazinone derivatives endowed with cardiovascular activity
NO93931225A NO931225L (no) 1992-04-16 1993-03-31 Benzoksazinon- og benzotiazinon-derivater med kardiovaskulaer akrivitet
AT93105752T ATE169293T1 (de) 1992-04-16 1993-04-07 Benzoxazinon- und benzothiazinonderivate mit kardiovasculärer wirkung
DE69320087T DE69320087T2 (de) 1992-04-16 1993-04-07 Benzoxazinon- und Benzothiazinonderivate mit kardiovasculärer Wirkung
EP93105752A EP0566018B1 (en) 1992-04-16 1993-04-07 Benzoxazinone and benzothiazinone derivatives endowed with cardiovascular activity
MX9302165A MX9302165A (es) 1992-04-16 1993-04-14 Derivados de benzoxazinona y benzothiazinona y composiciones farmaceuticas que los comprende
FI931688A FI931688A (fi) 1992-04-16 1993-04-14 Benzoxazinon- och benzotiazinonderivat med effekt pao hjaertblodkaerlen
TW082102853A TW288013B (it) 1992-04-16 1993-04-14
HU9301106A HUT68605A (en) 1992-04-16 1993-04-15 Benzoxazinone and benzothiazinone derivatives of cardiovascular activity, process for preparing them and pharmaceutical preparations containing them
JP11214993A JP3257716B2 (ja) 1992-04-16 1993-04-15 心臓血管活性を有するベンゾオキサジノン及びベンゾチアジノン誘導体
CN 93104624 CN1078466A (zh) 1992-04-16 1993-04-16 具有心血管作用的苯并嗪酮和苯并噻嗪酮
US08/347,217 US5480882A (en) 1992-04-16 1994-11-23 Benzoxazinone and benzothiazinone derivatives having cardiovascular activity

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITMI920940A IT1254884B (it) 1992-04-16 1992-04-16 Benzossazinoni e benzotiazinoni ad attivita' cardiovascolare

Publications (3)

Publication Number Publication Date
ITMI920940A0 true ITMI920940A0 (it) 1992-04-16
ITMI920940A1 ITMI920940A1 (it) 1993-10-16
IT1254884B IT1254884B (it) 1995-10-11

Family

ID=11362985

Family Applications (1)

Application Number Title Priority Date Filing Date
ITMI920940A IT1254884B (it) 1992-04-16 1992-04-16 Benzossazinoni e benzotiazinoni ad attivita' cardiovascolare

Country Status (17)

Country Link
US (1) US5480882A (it)
EP (1) EP0566018B1 (it)
JP (1) JP3257716B2 (it)
CN (1) CN1078466A (it)
AT (1) ATE169293T1 (it)
AU (1) AU655540B2 (it)
CA (1) CA2092342A1 (it)
DE (1) DE69320087T2 (it)
FI (1) FI931688A (it)
HU (1) HUT68605A (it)
IL (1) IL105158A (it)
IT (1) IT1254884B (it)
MX (1) MX9302165A (it)
NO (1) NO931225L (it)
NZ (1) NZ247249A (it)
TW (1) TW288013B (it)
ZA (1) ZA932030B (it)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1264812B1 (it) * 1993-07-28 1996-10-10 Italfarmaco Spa Derivati benzossazinonici e benzotiazinonici terapeuticamente attivi
AU5826100A (en) * 1999-07-13 2001-01-30 F. Hoffmann-La Roche Ag Benzazepinones and quinazolines
AU2001282551A1 (en) 2000-08-31 2002-03-13 Takeda Chemical Industries Ltd. Heart muscular cell apoptosis inhibitors and remedies/preventives for heart diseases
JP5700547B2 (ja) 2011-05-30 2015-04-15 国立大学法人京都大学 バイオチップ形成用感光性樹脂組成物、及びバイオチップ
CN102367239B (zh) * 2011-07-20 2015-10-28 沈阳药科大学 2-芳基-2,3-二氢-4h-1,3-苯并噻嗪-4-酮衍生物及其用途
CN103012188A (zh) * 2011-09-20 2013-04-03 北京京卫信康医药科技发展有限公司 一种龙胆酸乙醇胺的制备方法
CN102631108A (zh) * 2012-04-25 2012-08-15 张家港市立达金属制品有限公司 帽子展示架
ITMI20122221A1 (it) * 2012-12-21 2014-06-22 C4T S C A R L Nuovi composti del 2,3-diidro-4h-1,3-benzossazin-4-one, metodo per prepararli e forma farmaceutica che li comprende

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3539563A (en) * 1965-09-27 1970-11-10 Istituto Chemioterapico Tetracycline: 6-amino-4-oxo-2-(beta-chloroethyl) - 2,3 - dihydrobenzene - 1,3-oxazine double salt dihydrate
US3459748A (en) * 1967-04-28 1969-08-05 Squibb & Sons Inc Hydroxyalkylene-substituted benzoxazines and benzothiazines
FR2636065B1 (fr) * 1988-09-08 1993-05-07 Fabre Sa Pierre Nouveaux derives de dihydro-2,3 arylacoylaminoalcoyl-3 4h-benzoxazine-1,3 ones-4, leur preparation et leur application en tant que medicaments utiles en therapeutique
IT1244472B (it) * 1990-12-14 1994-07-15 Italfarmaco Spa Benzossazinoni e benzotiazinoni ad attivita' cardiovascolare

Also Published As

Publication number Publication date
AU3561793A (en) 1993-10-21
IT1254884B (it) 1995-10-11
EP0566018A3 (en) 1994-06-01
MX9302165A (es) 1993-10-01
IL105158A (en) 1996-10-31
ZA932030B (en) 1993-10-19
EP0566018A2 (en) 1993-10-20
FI931688A0 (fi) 1993-04-14
ATE169293T1 (de) 1998-08-15
HUT68605A (en) 1995-06-28
CA2092342A1 (en) 1993-10-17
DE69320087D1 (de) 1998-09-10
NO931225D0 (no) 1993-03-31
NZ247249A (en) 1995-01-27
NO931225L (no) 1993-10-18
FI931688A (fi) 1993-10-17
TW288013B (it) 1996-10-11
JPH0625194A (ja) 1994-02-01
DE69320087T2 (de) 1998-12-10
US5480882A (en) 1996-01-02
EP0566018B1 (en) 1998-08-05
HU9301106D0 (en) 1993-07-28
AU655540B2 (en) 1994-12-22
JP3257716B2 (ja) 2002-02-18
CN1078466A (zh) 1993-11-17
ITMI920940A1 (it) 1993-10-16

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19970428