IT9019133A0 - Acido 3-l-(5-tioxo-l-prolil)tiazolidin-4-carbossilico e derivati, loro preparazione e composizioni farmaceutiche che li contengono - Google Patents

Acido 3-l-(5-tioxo-l-prolil)tiazolidin-4-carbossilico e derivati, loro preparazione e composizioni farmaceutiche che li contengono

Info

Publication number
IT9019133A0
IT9019133A0 IT19133A IT1913390A IT9019133A0 IT 9019133 A0 IT9019133 A0 IT 9019133A0 IT 19133 A IT19133 A IT 19133A IT 1913390 A IT1913390 A IT 1913390A IT 9019133 A0 IT9019133 A0 IT 9019133A0
Authority
IT
Italy
Prior art keywords
thiazolidin
prolyl
thioxo
derivatives
contain
Prior art date
Application number
IT19133A
Other languages
English (en)
Other versions
IT9019133A1 (it
IT1237998B (it
Inventor
Stefano Poli
Corona Lucio Del
Germano Coppi
Original Assignee
Poli Ind Chimica Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Poli Ind Chimica Spa filed Critical Poli Ind Chimica Spa
Publication of IT9019133A0 publication Critical patent/IT9019133A0/it
Priority to IT01913390A priority Critical patent/IT1237998B/it
Priority to IL96814A priority patent/IL96814A0/xx
Priority to IE473590A priority patent/IE904735A1/en
Priority to ZA9198A priority patent/ZA9198B/xx
Priority to CA002033682A priority patent/CA2033682A1/en
Priority to EP91100394A priority patent/EP0439044A1/en
Priority to ES91100394T priority patent/ES2025026A4/es
Priority to DE199191100394T priority patent/DE439044T1/de
Priority to US07/652,792 priority patent/US5212160A/en
Priority to NZ236832A priority patent/NZ236832A/en
Priority to NO91910231A priority patent/NO910231L/no
Priority to KR1019910001010A priority patent/KR910014374A/ko
Priority to JP3005782A priority patent/JPH04210980A/ja
Priority to HU91229A priority patent/HU210248B/hu
Priority to FI910330A priority patent/FI910330A/fi
Priority to AU69912/91A priority patent/AU632896B2/en
Publication of IT9019133A1 publication Critical patent/IT9019133A1/it
Priority to GR91300116T priority patent/GR910300116T1/el
Application granted granted Critical
Publication of IT1237998B publication Critical patent/IT1237998B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06139Dipeptides with the first amino acid being heterocyclic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Plural Heterocyclic Compounds (AREA)
IT01913390A 1990-01-23 1990-01-23 Acido 3-l-(5-tioxo-l-prolil)tiazolidin-4-carbossilico e derivati, loro preparazione e composizioni farmaceutiche che li contengono IT1237998B (it)

Priority Applications (17)

Application Number Priority Date Filing Date Title
IT01913390A IT1237998B (it) 1990-01-23 1990-01-23 Acido 3-l-(5-tioxo-l-prolil)tiazolidin-4-carbossilico e derivati, loro preparazione e composizioni farmaceutiche che li contengono
IL96814A IL96814A0 (en) 1990-01-23 1990-12-27 3-l-(5-thioxo-l-prolyl)thiazolidine-4-carboxylic acid and derivatives therefrom,processes for the preparation thereof and pharmaceutical compositions containing them
IE473590A IE904735A1 (en) 1990-01-23 1990-12-31 3-l-(5-thioxo-l-prolyl)thiazolidine-4-carboxylic acid and¹derivatives therefrom, processes for the preparation thereof¹and pharmaceutical compositions containing them
ZA9198A ZA9198B (en) 1990-01-23 1991-01-04 3-l-(5-thioxo-l-prolyl)thiazolidine-4-carboxylic acid and derivatives therefrom,processes for the preparation thereof and pharmaceutical compositions containing them
CA002033682A CA2033682A1 (en) 1990-01-23 1991-01-07 3-l-(5-thioxo-l-propyl)thiazolidine-4-carboxylic acid and derivatives therefrom, processes for the preparation thereof and pharmaceutical compositions containing them
EP91100394A EP0439044A1 (en) 1990-01-23 1991-01-15 3-L-(5-thioxo-L-prolyl)thiazolidine-4-carboxylic acid and derivatives therefrom, processes for the preparation thereof and pharmaceutical compositions containing them
ES91100394T ES2025026A4 (es) 1990-01-23 1991-01-15 Acido 3-l-(5-tioxo-l-propil) tiazolidina-4-carboxilico y derivados del mismo, procedimiento para su preparacion y composiciones farmaceuticas que los contienen.
DE199191100394T DE439044T1 (de) 1990-01-23 1991-01-15 3-l-(5-thioxo-l-prolyl)thiazolidine-4-carbonsaeure und derivate davon, verfahren zu ihrer herstellung und diese verbindungen enthaltende pharmazeutische zusammensetzungen.
US07/652,792 US5212160A (en) 1990-01-23 1991-01-16 3-l-(5-thioxo-l-prolyl)thiazolidine-4-carboxylic acid and derivatives therefrom, processes for the preparation thereof and pharmaceutical compositions containing them
NZ236832A NZ236832A (en) 1990-01-23 1991-01-18 3-l-(5-thioxo-l-prolyl)thiazolidine-4-carboxylic acid derivatives, preparation and pharmaceutical compositions thereof
NO91910231A NO910231L (no) 1990-01-23 1991-01-21 3-l-(5-tiokso-l-prolyl)tiazolidin-4-karboksylsyre samt derivater derav.
KR1019910001010A KR910014374A (ko) 1990-01-23 1991-01-22 3-l-(5-티옥소-l-프롤릴)티아졸리딘-4- 카르복실산과 그 유도체, 이의 제법 및 이를 함유하는 약학적 조성물
JP3005782A JPH04210980A (ja) 1990-01-23 1991-01-22 3−l−(5−チオキソ−l−プロリル)チアゾリジン−4−カルボン酸およびその誘導体、その製造方法並びにそれを含む薬学的組成物
HU91229A HU210248B (en) 1990-01-23 1991-01-22 Process for preparing 3-l-(5-thioxo-l-prolyl)-thiazolidine-4-carboxylic acid, derivatives thereof and pharmaceutical compositions containing them
FI910330A FI910330A (fi) 1990-01-23 1991-01-22 3-l-(5-tioxo-l-prolyl) tiazolidin -4-karboxylsyra och dess derivat, processer foer deras framstaellning och farmaceutiska sammansaettningar, som innehaoller dem.
AU69912/91A AU632896B2 (en) 1990-01-23 1991-01-23 3-l-(5-thioxo-l-prolyl) thiazolidine-4-carboxylic acid and derivatives therefrom, processes for the preparation thereof and pharmaceutical compositions containing them
GR91300116T GR910300116T1 (en) 1990-01-23 1992-03-20 3-l-(5-thioxo-l-prolyl)thiazolidine-4-carboxylic acid and derivatives therefrom, processes for the preparation thereof and pharmaceutical compositions containing them

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT01913390A IT1237998B (it) 1990-01-23 1990-01-23 Acido 3-l-(5-tioxo-l-prolil)tiazolidin-4-carbossilico e derivati, loro preparazione e composizioni farmaceutiche che li contengono

Publications (3)

Publication Number Publication Date
IT9019133A0 true IT9019133A0 (it) 1990-01-23
IT9019133A1 IT9019133A1 (it) 1991-07-24
IT1237998B IT1237998B (it) 1993-06-21

Family

ID=11155105

Family Applications (1)

Application Number Title Priority Date Filing Date
IT01913390A IT1237998B (it) 1990-01-23 1990-01-23 Acido 3-l-(5-tioxo-l-prolil)tiazolidin-4-carbossilico e derivati, loro preparazione e composizioni farmaceutiche che li contengono

Country Status (17)

Country Link
US (1) US5212160A (it)
EP (1) EP0439044A1 (it)
JP (1) JPH04210980A (it)
KR (1) KR910014374A (it)
AU (1) AU632896B2 (it)
CA (1) CA2033682A1 (it)
DE (1) DE439044T1 (it)
ES (1) ES2025026A4 (it)
FI (1) FI910330A (it)
GR (1) GR910300116T1 (it)
HU (1) HU210248B (it)
IE (1) IE904735A1 (it)
IL (1) IL96814A0 (it)
IT (1) IT1237998B (it)
NO (1) NO910231L (it)
NZ (1) NZ236832A (it)
ZA (1) ZA9198B (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1230706B (it) * 1989-02-10 1991-10-29 Poli Ind Chimica Spa Derivati dell'acido 3 piroglutamoil tiazolidin 4 carbossilico e loro proprieta' farmacologiche.
CN111233854A (zh) * 2019-12-30 2020-06-05 常州寅盛药业有限公司 一种匹多莫德杂质的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1202426B (it) * 1987-01-26 1989-02-09 Poli Ind Chimica Spa Derivato di acido tiazolidin-4-carbossilico,sua preparazione e composizioni farmaceutiche che lo contengono
IT1230706B (it) * 1989-02-10 1991-10-29 Poli Ind Chimica Spa Derivati dell'acido 3 piroglutamoil tiazolidin 4 carbossilico e loro proprieta' farmacologiche.
IT1239029B (it) * 1989-10-12 1993-09-20 Poli Ind Chimica Spa Processo per la preparazione dell'acido 3-(l-piroglutamil)-l- tiazolidin-4-carbossilico e suoi derivati.

Also Published As

Publication number Publication date
KR910014374A (ko) 1991-08-31
HU210248B (en) 1995-03-28
FI910330A0 (fi) 1991-01-22
NZ236832A (en) 1993-05-26
US5212160A (en) 1993-05-18
ES2025026A4 (es) 1992-03-16
ZA9198B (en) 1991-10-30
GR910300116T1 (en) 1992-03-20
IL96814A0 (en) 1991-09-16
HU910229D0 (en) 1991-08-28
AU6991291A (en) 1991-07-25
JPH04210980A (ja) 1992-08-03
FI910330A (fi) 1991-07-24
IE904735A1 (en) 1991-07-31
NO910231D0 (no) 1991-01-21
NO910231L (no) 1991-07-24
IT9019133A1 (it) 1991-07-24
AU632896B2 (en) 1993-01-14
CA2033682A1 (en) 1991-07-24
EP0439044A1 (en) 1991-07-31
IT1237998B (it) 1993-06-21
DE439044T1 (de) 1992-03-19
HUT60736A (en) 1992-10-28

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Legal Events

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TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19940128