IT8620598A0 - SUBSTITUTED STEROIDS 11/B AND PROCEDURE FOR THEIR PREPARATION. - Google Patents

SUBSTITUTED STEROIDS 11/B AND PROCEDURE FOR THEIR PREPARATION.

Info

Publication number
IT8620598A0
IT8620598A0 IT8620598A IT2059886A IT8620598A0 IT 8620598 A0 IT8620598 A0 IT 8620598A0 IT 8620598 A IT8620598 A IT 8620598A IT 2059886 A IT2059886 A IT 2059886A IT 8620598 A0 IT8620598 A0 IT 8620598A0
Authority
IT
Italy
Prior art keywords
procedure
preparation
substituted steroids
steroids
substituted
Prior art date
Application number
IT8620598A
Other languages
Italian (it)
Other versions
IT8620598A1 (en
IT1190014B (en
Inventor
Franco Buzzetti
Natale Barbugian
Paolo Lombardi
Enrico Di Salle
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of IT8620598A0 publication Critical patent/IT8620598A0/en
Publication of IT8620598A1 publication Critical patent/IT8620598A1/en
Application granted granted Critical
Publication of IT1190014B publication Critical patent/IT1190014B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0077Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0066Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C07J1/0074Esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0081Substituted in position 17 alfa and 17 beta
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J21/00Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005Ketals
    • C07J21/006Ketals at position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0077Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
    • C07J41/0083Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring
    • C07J71/001Oxiranes
IT20598/86A 1985-05-31 1986-05-28 STEROIDS 11 / B / REPLACED AND PROCEDURE FOR THEIR PREPARATION IT1190014B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858513723A GB8513723D0 (en) 1985-05-31 1985-05-31 11-beta substituted steroids

Publications (3)

Publication Number Publication Date
IT8620598A0 true IT8620598A0 (en) 1986-05-28
IT8620598A1 IT8620598A1 (en) 1987-11-28
IT1190014B IT1190014B (en) 1988-02-10

Family

ID=10579949

Family Applications (1)

Application Number Title Priority Date Filing Date
IT20598/86A IT1190014B (en) 1985-05-31 1986-05-28 STEROIDS 11 / B / REPLACED AND PROCEDURE FOR THEIR PREPARATION

Country Status (21)

Country Link
JP (1) JPS6212796A (en)
KR (1) KR860009035A (en)
AU (1) AU587031B2 (en)
BE (1) BE904846A (en)
CH (1) CH669385A5 (en)
DE (1) DE3617883A1 (en)
DK (1) DK251386A (en)
ES (1) ES8707972A1 (en)
FI (1) FI862278A (en)
FR (1) FR2582654B1 (en)
GB (2) GB8513723D0 (en)
GR (1) GR861405B (en)
HU (1) HU197925B (en)
IL (1) IL78957A (en)
IT (1) IT1190014B (en)
NL (1) NL8601387A (en)
NZ (1) NZ216325A (en)
PT (1) PT82665B (en)
SE (1) SE8602449L (en)
SU (1) SU1508963A3 (en)
ZA (1) ZA864065B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE69820T1 (en) * 1987-04-24 1991-12-15 Akzo Nv 11-ARYLESTRAND DERIVATIVES AND 11-ARYLPREGNAN DERIVATIVES.
ATE85342T1 (en) * 1987-12-12 1993-02-15 Akzo Nv 11-ARYLSTEROID DERIVATIVES.
FR2643638B1 (en) * 1989-02-24 1991-06-14 Roussel Uclaf NOVEL 19-NOR STEROIDS HAVING IN THE 11BETA POSITION A CARBON CHAIN COMPRISING AN AMIDE OR CARBAMATE FUNCTION, THEIR PREPARATION METHOD AND INTERMEDIATES THEREOF, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
FR2665901B2 (en) * 1989-02-24 1994-07-29 Roussel Uclaf NEW 19-NOR STEROUIDES HAVING IN THE 11BETA POSITION A CARBON CHAIN COMPRISING AN AMIDE FUNCTION, THEIR PREPARATION, THEIR APPLICATION AS MEDICAMENTS.
TWI265167B (en) * 1999-11-29 2006-11-01 Akzo Nobel Nv 3-methylene steroid derivatives
DE19961219A1 (en) * 1999-12-15 2001-07-19 Jenapharm Gmbh 11beta-phenyltratriene derivatives with fluoroalkyl groups in the aromatic side chain, their preparation and pharmaceutical compositions containing these compounds
TW200531977A (en) 2004-03-25 2005-10-01 Akzo Nobel Nv Progesterone receptor modulators

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH488682A (en) * 1965-07-30 1970-04-15 Ciba Geigy Process for the preparation of 4,9,11-trienes of the 19-nor-androstane series
FR192F (en) * 1965-10-22
FR5913M (en) * 1965-12-02 1968-04-01
NL128375C (en) * 1966-02-18
FR2054525B1 (en) * 1969-07-28 1973-01-12 Roussel Uclaf
FR2054527B1 (en) * 1969-07-28 1973-06-08 Roussel Uclaf
FR2377418A1 (en) * 1977-01-13 1978-08-11 Roussel Uclaf NEW 4,9-DIENIC 11B-SUBSTITUTE STEROID DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS
ZA8231B (en) * 1981-01-09 1982-11-24 Roussel Uclaf New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained
FR2522328B1 (en) * 1982-03-01 1986-02-14 Roussel Uclaf NEW PRODUCTS DERIVED FROM THE STRUCTURE 3-CETO 4,9 19-NOR STEROIDS, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS
AU580843B2 (en) * 1985-02-07 1989-02-02 Schering Aktiengesellschaft 11``-phenyl-gonanes, their manufacture and pharmaceutical preparations containing them

Also Published As

Publication number Publication date
IT8620598A1 (en) 1987-11-28
FI862278A0 (en) 1986-05-29
BE904846A (en) 1986-12-01
ZA864065B (en) 1987-01-28
KR860009035A (en) 1986-12-19
GB8612866D0 (en) 1986-07-02
GB2175905A (en) 1986-12-10
JPS6212796A (en) 1987-01-21
ES8707972A1 (en) 1987-09-01
FR2582654A1 (en) 1986-12-05
SE8602449L (en) 1986-12-01
FR2582654B1 (en) 1988-06-03
NZ216325A (en) 1989-01-27
CH669385A5 (en) 1989-03-15
DK251386D0 (en) 1986-05-29
AU5806286A (en) 1986-12-04
SE8602449D0 (en) 1986-05-29
IL78957A0 (en) 1986-09-30
SU1508963A3 (en) 1989-09-15
ES555298A0 (en) 1987-09-01
IT1190014B (en) 1988-02-10
GB2175905B (en) 1989-01-18
NL8601387A (en) 1986-12-16
PT82665B (en) 1988-08-17
PT82665A (en) 1986-06-01
HU197925B (en) 1989-06-28
DE3617883A1 (en) 1986-12-04
DK251386A (en) 1986-12-01
FI862278A (en) 1986-12-01
GR861405B (en) 1986-09-26
AU587031B2 (en) 1989-08-03
GB8513723D0 (en) 1985-07-03
IL78957A (en) 1990-11-29
HUT44575A (en) 1988-03-28

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