DK251386A - 11-BETA-SUBSTITUTED STEROIDS, PROCEDURES FOR PREPARING IT, AND PHARMACEUTICAL AND VETERINARY PREPARATIONS CONTAINING THESE COMPOUNDS - Google Patents

11-BETA-SUBSTITUTED STEROIDS, PROCEDURES FOR PREPARING IT, AND PHARMACEUTICAL AND VETERINARY PREPARATIONS CONTAINING THESE COMPOUNDS Download PDF

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Publication number
DK251386A
DK251386A DK251386A DK251386A DK251386A DK 251386 A DK251386 A DK 251386A DK 251386 A DK251386 A DK 251386A DK 251386 A DK251386 A DK 251386A DK 251386 A DK251386 A DK 251386A
Authority
DK
Denmark
Prior art keywords
beta
pharmaceutical
procedures
preparing
compounds
Prior art date
Application number
DK251386A
Other languages
Danish (da)
Other versions
DK251386D0 (en
Inventor
Franco Faustini
Alessio Roberto D
Vittoria Villa
Enrico Di Salle
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of DK251386D0 publication Critical patent/DK251386D0/en
Publication of DK251386A publication Critical patent/DK251386A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0077Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0066Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
    • C07J1/007Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C07J1/0074Esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051Estrane derivatives
    • C07J1/0081Substituted in position 17 alfa and 17 beta
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J21/00Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005Ketals
    • C07J21/006Ketals at position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0077Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
    • C07J41/0083Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring
    • C07J71/001Oxiranes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK251386A 1985-05-31 1986-05-29 11-BETA-SUBSTITUTED STEROIDS, PROCEDURES FOR PREPARING IT, AND PHARMACEUTICAL AND VETERINARY PREPARATIONS CONTAINING THESE COMPOUNDS DK251386A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858513723A GB8513723D0 (en) 1985-05-31 1985-05-31 11-beta substituted steroids

Publications (2)

Publication Number Publication Date
DK251386D0 DK251386D0 (en) 1986-05-29
DK251386A true DK251386A (en) 1986-12-01

Family

ID=10579949

Family Applications (1)

Application Number Title Priority Date Filing Date
DK251386A DK251386A (en) 1985-05-31 1986-05-29 11-BETA-SUBSTITUTED STEROIDS, PROCEDURES FOR PREPARING IT, AND PHARMACEUTICAL AND VETERINARY PREPARATIONS CONTAINING THESE COMPOUNDS

Country Status (21)

Country Link
JP (1) JPS6212796A (en)
KR (1) KR860009035A (en)
AU (1) AU587031B2 (en)
BE (1) BE904846A (en)
CH (1) CH669385A5 (en)
DE (1) DE3617883A1 (en)
DK (1) DK251386A (en)
ES (1) ES8707972A1 (en)
FI (1) FI862278A (en)
FR (1) FR2582654B1 (en)
GB (2) GB8513723D0 (en)
GR (1) GR861405B (en)
HU (1) HU197925B (en)
IL (1) IL78957A (en)
IT (1) IT1190014B (en)
NL (1) NL8601387A (en)
NZ (1) NZ216325A (en)
PT (1) PT82665B (en)
SE (1) SE8602449L (en)
SU (1) SU1508963A3 (en)
ZA (1) ZA864065B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3866410D1 (en) * 1987-04-24 1992-01-09 Akzo Nv 11-ARYLESTRANDERIVATIVES AND 11-ARYLPREGNANDERIVATIVES.
ES2053714T3 (en) * 1987-12-12 1994-08-01 Akzo Nv PROCESS FOR THE PREPARATION OF 11-ARILESTEROIDES.
FR2665901B2 (en) * 1989-02-24 1994-07-29 Roussel Uclaf NEW 19-NOR STEROUIDES HAVING IN THE 11BETA POSITION A CARBON CHAIN COMPRISING AN AMIDE FUNCTION, THEIR PREPARATION, THEIR APPLICATION AS MEDICAMENTS.
FR2643638B1 (en) * 1989-02-24 1991-06-14 Roussel Uclaf NOVEL 19-NOR STEROIDS HAVING IN THE 11BETA POSITION A CARBON CHAIN COMPRISING AN AMIDE OR CARBAMATE FUNCTION, THEIR PREPARATION METHOD AND INTERMEDIATES THEREOF, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
TWI265167B (en) * 1999-11-29 2006-11-01 Akzo Nobel Nv 3-methylene steroid derivatives
DE19961219A1 (en) * 1999-12-15 2001-07-19 Jenapharm Gmbh 11beta-phenyltratriene derivatives with fluoroalkyl groups in the aromatic side chain, their preparation and pharmaceutical compositions containing these compounds
TW200531977A (en) 2004-03-25 2005-10-01 Akzo Nobel Nv Progesterone receptor modulators

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH488682A (en) * 1965-07-30 1970-04-15 Ciba Geigy Process for the preparation of 4,9,11-trienes of the 19-nor-androstane series
FR190F (en) * 1965-10-22
FR5913M (en) * 1965-12-02 1968-04-01
NL128375C (en) * 1966-02-18
FR2054525B1 (en) * 1969-07-28 1973-01-12 Roussel Uclaf
FR2054527B1 (en) * 1969-07-28 1973-06-08 Roussel Uclaf
FR2377418A1 (en) * 1977-01-13 1978-08-11 Roussel Uclaf NEW 4,9-DIENIC 11B-SUBSTITUTE STEROID DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS
ZA8231B (en) * 1981-01-09 1982-11-24 Roussel Uclaf New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained
FR2522328B1 (en) * 1982-03-01 1986-02-14 Roussel Uclaf NEW PRODUCTS DERIVED FROM THE STRUCTURE 3-CETO 4,9 19-NOR STEROIDS, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS
AU580843B2 (en) * 1985-02-07 1989-02-02 Schering Aktiengesellschaft 11``-phenyl-gonanes, their manufacture and pharmaceutical preparations containing them

Also Published As

Publication number Publication date
ES555298A0 (en) 1987-09-01
BE904846A (en) 1986-12-01
DK251386D0 (en) 1986-05-29
AU587031B2 (en) 1989-08-03
PT82665B (en) 1988-08-17
IT8620598A1 (en) 1987-11-28
ES8707972A1 (en) 1987-09-01
FI862278A0 (en) 1986-05-29
SU1508963A3 (en) 1989-09-15
SE8602449L (en) 1986-12-01
HU197925B (en) 1989-06-28
JPS6212796A (en) 1987-01-21
CH669385A5 (en) 1989-03-15
GB8513723D0 (en) 1985-07-03
ZA864065B (en) 1987-01-28
HUT44575A (en) 1988-03-28
GB8612866D0 (en) 1986-07-02
SE8602449D0 (en) 1986-05-29
FR2582654A1 (en) 1986-12-05
IL78957A0 (en) 1986-09-30
FR2582654B1 (en) 1988-06-03
KR860009035A (en) 1986-12-19
GB2175905B (en) 1989-01-18
DE3617883A1 (en) 1986-12-04
IT1190014B (en) 1988-02-10
IT8620598A0 (en) 1986-05-28
AU5806286A (en) 1986-12-04
FI862278A (en) 1986-12-01
PT82665A (en) 1986-06-01
NL8601387A (en) 1986-12-16
GB2175905A (en) 1986-12-10
IL78957A (en) 1990-11-29
GR861405B (en) 1986-09-26
NZ216325A (en) 1989-01-27

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