IT8167533A0 - Composto della categoria delle benzossazepine utilizzabile come farmaco attivo sul sistema nervoso centrale - Google Patents
Composto della categoria delle benzossazepine utilizzabile come farmaco attivo sul sistema nervoso centraleInfo
- Publication number
- IT8167533A0 IT8167533A0 IT8167533A IT6753381A IT8167533A0 IT 8167533 A0 IT8167533 A0 IT 8167533A0 IT 8167533 A IT8167533 A IT 8167533A IT 6753381 A IT6753381 A IT 6753381A IT 8167533 A0 IT8167533 A0 IT 8167533A0
- Authority
- IT
- Italy
- Prior art keywords
- benzoxazepine
- compound
- nervous system
- central nervous
- active drug
- Prior art date
Links
- ZCXLTWVZYXBHJS-UHFFFAOYSA-N 1,2-benzoxazepine Chemical compound O1N=CC=CC2=CC=CC=C12 ZCXLTWVZYXBHJS-UHFFFAOYSA-N 0.000 title 1
- 210000003169 central nervous system Anatomy 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D267/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D267/02—Seven-membered rings
- C07D267/08—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D267/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D267/14—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP5218580A JPS56147778A (en) | 1980-04-18 | 1980-04-18 | 4,1-benzoxazepines |
JP55136646A JPS5759893A (en) | 1980-09-29 | 1980-09-29 | 4,1-benzoxazepin derivative |
Publications (2)
Publication Number | Publication Date |
---|---|
IT8167533A0 true IT8167533A0 (it) | 1981-04-17 |
IT1146746B IT1146746B (it) | 1986-11-19 |
Family
ID=26392810
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT67533/81A IT1146746B (it) | 1980-04-18 | 1981-04-17 | Composto della categoria delle benzossazepine utilizzabilecome farmaco attivo sul sistema nervoso centrale |
Country Status (7)
Country | Link |
---|---|
US (2) | US4374842A (it) |
AU (1) | AU544637B2 (it) |
CH (1) | CH645637A5 (it) |
DE (1) | DE3115552A1 (it) |
FR (1) | FR2480751A1 (it) |
GB (1) | GB2075012B (it) |
IT (1) | IT1146746B (it) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4590187A (en) * | 1983-11-17 | 1986-05-20 | The Upjohn Company | Phospholipase A2 inhibition using 4,1-benzoxazepine-2-(3H)-ones |
US4960767A (en) * | 1988-08-01 | 1990-10-02 | Hoechst-Roussel Pharmaceuticals Inc. | Isoxazolobenzoxazepines |
US4873234A (en) * | 1988-08-01 | 1989-10-10 | Hoechst-Roussel Pharmaceuticals Inc. | Isoxazolobenzoxazepines |
GB8823475D0 (en) * | 1988-10-06 | 1988-11-16 | Merck Sharp & Dohme | Chemical compounds |
US5726306A (en) * | 1992-04-20 | 1998-03-10 | Takeda Chemical Industries, Ltd. | 4,1-benzoxazepin derivatives and their use |
DE69332792T2 (de) * | 1992-04-20 | 2004-01-15 | Takeda Chemical Industries Ltd | 4,1-Benzoxazepinderivate als Squalen-Synthetase Inhibitoren und ihre Verwendung zur Behandlung von Hypercholesterämie und als Fungizide |
AU678503B2 (en) * | 1993-09-24 | 1997-05-29 | Takeda Chemical Industries Ltd. | Condensed heterocyclic compounds and their use as squalene synthetase inhibitors |
WO1999011635A1 (en) * | 1997-09-02 | 1999-03-11 | Du Pont Pharmaceuticals Company | 5,5-disubstituted-1,5-dihydro-4,1-benzoxazepin-2(3h)-ones useful as hiv reverse transcriptase inhibitors |
DE102004001871A1 (de) * | 2004-01-14 | 2005-09-01 | Bayer Healthcare Ag | Tricyclische Benzazepin-Derivate und ihre Verwendung |
US7323455B2 (en) * | 2004-03-24 | 2008-01-29 | Wyeth | 7-aryl 1,5-dihydro-4,1-benzoxazepin-2(3H)-one derivatives and their use as progesterone receptor modulators |
KR20140082765A (ko) * | 2011-10-05 | 2014-07-02 | 에프. 호프만-라 로슈 아게 | V1a 길항제로서의 사이클로헥실-4H,6H-5-옥사-2,3,10b-트라이아자-벤조[e]아줄렌 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3681343A (en) * | 1971-05-11 | 1972-08-01 | Upjohn Co | 6-phenyl-s-triazolo{8 4,3-a{9 {8 1,4{9 {0 benzodiazepines |
JPS5572177A (en) | 1978-11-27 | 1980-05-30 | Shionogi & Co Ltd | 4,1-benzoxazepine or 4,1-benzothiazepine |
-
1981
- 1981-04-02 US US06/250,299 patent/US4374842A/en not_active Expired - Fee Related
- 1981-04-15 CH CH253081A patent/CH645637A5/de not_active IP Right Cessation
- 1981-04-16 FR FR8107700A patent/FR2480751A1/fr active Granted
- 1981-04-16 AU AU69623/81A patent/AU544637B2/en not_active Ceased
- 1981-04-16 DE DE19813115552 patent/DE3115552A1/de not_active Withdrawn
- 1981-04-17 IT IT67533/81A patent/IT1146746B/it active
- 1981-04-21 GB GB8112387A patent/GB2075012B/en not_active Expired
-
1982
- 1982-07-13 US US06/397,855 patent/US4476133A/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
GB2075012B (en) | 1984-02-15 |
CH645637A5 (de) | 1984-10-15 |
AU544637B2 (en) | 1985-06-06 |
AU6962381A (en) | 1981-10-22 |
US4476133A (en) | 1984-10-09 |
FR2480751B1 (it) | 1983-03-25 |
IT1146746B (it) | 1986-11-19 |
DE3115552A1 (de) | 1982-02-18 |
FR2480751A1 (fr) | 1981-10-23 |
GB2075012A (en) | 1981-11-11 |
US4374842A (en) | 1983-02-22 |
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