IT8048062A0 - Derivati di acidi mercaptoacildii dropirazol carbossilici dotati di attivita' ipotensiva e procedimento per la loro preparazione - Google Patents

Derivati di acidi mercaptoacildii dropirazol carbossilici dotati di attivita' ipotensiva e procedimento per la loro preparazione

Info

Publication number
IT8048062A0
IT8048062A0 IT8048062A IT4806280A IT8048062A0 IT 8048062 A0 IT8048062 A0 IT 8048062A0 IT 8048062 A IT8048062 A IT 8048062A IT 4806280 A IT4806280 A IT 4806280A IT 8048062 A0 IT8048062 A0 IT 8048062A0
Authority
IT
Italy
Prior art keywords
mercaptoacildii
dropyrazol
derivatives
procedure
preparation
Prior art date
Application number
IT8048062A
Other languages
English (en)
Other versions
IT1127384B (it
Inventor
George Charles Rovnyak
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of IT8048062A0 publication Critical patent/IT8048062A0/it
Application granted granted Critical
Publication of IT1127384B publication Critical patent/IT1127384B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IT48062/80A 1979-03-08 1980-03-03 Derivati di acidi mercaptoacildii dropirazol carbossilici dotati di attivita' ipotensiva e procedimento per la loro preparazione IT1127384B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/018,548 US4211786A (en) 1979-03-08 1979-03-08 Mercaptoacyldihydropyrazole carboxylic acid derivatives

Publications (2)

Publication Number Publication Date
IT8048062A0 true IT8048062A0 (it) 1980-03-03
IT1127384B IT1127384B (it) 1986-05-21

Family

ID=21788501

Family Applications (1)

Application Number Title Priority Date Filing Date
IT48062/80A IT1127384B (it) 1979-03-08 1980-03-03 Derivati di acidi mercaptoacildii dropirazol carbossilici dotati di attivita' ipotensiva e procedimento per la loro preparazione

Country Status (16)

Country Link
US (1) US4211786A (it)
JP (1) JPS55122766A (it)
AU (1) AU534582B2 (it)
BE (1) BE882133A (it)
CA (1) CA1137497A (it)
CH (1) CH645630A5 (it)
DE (1) DE3008904A1 (it)
DK (1) DK99980A (it)
FR (1) FR2450820A1 (it)
GB (1) GB2048850B (it)
IE (1) IE49541B1 (it)
IT (1) IT1127384B (it)
LU (1) LU82223A1 (it)
NL (1) NL8001349A (it)
SE (1) SE450382B (it)
ZA (1) ZA801016B (it)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA794723B (en) * 1978-09-11 1980-08-27 Univ Miami Anti-hypertensive agents
US4288368A (en) * 1979-07-30 1981-09-08 E. R. Squibb & Sons, Inc. Dithioacylproline derivatives
US4331806A (en) * 1979-07-30 1982-05-25 E. R. Squibb & Sons, Inc. Dithioacyldihydropyrazole carboxylic acid derivatives
CA1156236A (en) * 1979-10-25 1983-11-01 George C. Rovnyak Mercaptoacyldihydropyrazole carboxylic acid derivatives
US4254267A (en) * 1979-10-25 1981-03-03 E. R. Squibb & Sons, Inc. Mercaptoacyldihydropyrazole carboxylic acid derivatives
US4266065A (en) * 1980-04-14 1981-05-05 E. R. Squibb & Sons, Inc. Mercaptoacyldihydropyrazole carboxylic acid derivatives
US4692458A (en) * 1980-03-05 1987-09-08 University Of Miami Anti-hypertensive agents
US4312990A (en) * 1980-09-11 1982-01-26 E. R. Squibb & Sons, Inc. 1-Mercaptoacyl-3-[(aminosulfonyl) phenyl]-4,5-dihydro-1H-pyrazole-5-carboxylic acid
US4371526A (en) * 1981-08-21 1983-02-01 E. R. Squibb & Sons, Inc. Phosphinylalkanoyl substituted 4,5-dihydropyrazole-5-carboxylic acid derivatives and hypotensive method and composition
JPS58133376U (ja) * 1982-03-05 1983-09-08 吉原 靖人 バツテイング練習用バツト
US4470973A (en) * 1982-07-19 1984-09-11 E. R. Squibb & Sons, Inc. Substituted peptide compounds
US4621092A (en) * 1982-07-22 1986-11-04 E. R. Squibb & Sons, Inc. Substituted proline compounds, composition and method of use
US4742067A (en) * 1982-07-22 1988-05-03 E. R. Squibb & Sons, Inc. Acylalkylaminocarbonyl substituted amino and imino acid compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4105776A (en) * 1976-06-21 1978-08-08 E. R. Squibb & Sons, Inc. Proline derivatives and related compounds
US4046889A (en) * 1976-02-13 1977-09-06 E. R. Squibb & Sons, Inc. Azetidine-2-carboxylic acid derivatives
US4053651A (en) * 1976-05-10 1977-10-11 E. R. Squibb & Sons, Inc. Compounds and method for alleviating angiotensin related hypertension
ZA777062B (en) * 1976-12-03 1979-02-28 Squibb & Sons Inc Derivatives of thiazolidinecarboxylic acids and related acids
US4129566A (en) * 1978-02-15 1978-12-12 E. R. Squibb & Sons, Inc. Derivatives of dehydrocyclicimino acids

Also Published As

Publication number Publication date
SE450382B (sv) 1987-06-22
SE8001818L (sv) 1980-09-09
FR2450820A1 (fr) 1980-10-03
IE49541B1 (en) 1985-10-30
JPH0141628B2 (it) 1989-09-06
CH645630A5 (de) 1984-10-15
FR2450820B1 (it) 1983-04-22
AU534582B2 (en) 1984-02-09
JPS55122766A (en) 1980-09-20
IT1127384B (it) 1986-05-21
US4211786A (en) 1980-07-08
GB2048850A (en) 1980-12-17
LU82223A1 (de) 1980-09-24
CA1137497A (en) 1982-12-14
BE882133A (fr) 1980-09-08
DK99980A (da) 1980-09-09
GB2048850B (en) 1983-04-27
DE3008904A1 (de) 1980-09-18
NL8001349A (nl) 1980-09-10
AU5582280A (en) 1980-09-11
ZA801016B (en) 1981-02-25
IE800449L (en) 1980-09-08

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Effective date: 19930315