BE882133A - Derives d'acides 1-omega-mercaptoacyl)-4,5-dihydropyrazole-5-carboxyliques et leur procede de preparation - Google Patents

Derives d'acides 1-omega-mercaptoacyl)-4,5-dihydropyrazole-5-carboxyliques et leur procede de preparation

Info

Publication number
BE882133A
BE882133A BE0/199718A BE199718A BE882133A BE 882133 A BE882133 A BE 882133A BE 0/199718 A BE0/199718 A BE 0/199718A BE 199718 A BE199718 A BE 199718A BE 882133 A BE882133 A BE 882133A
Authority
BE
Belgium
Prior art keywords
mercaptoacyl
dihydropyrazole
omega
carboxylic acid
preparation process
Prior art date
Application number
BE0/199718A
Other languages
English (en)
Inventor
G Rovnyak
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of BE882133A publication Critical patent/BE882133A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BE0/199718A 1979-03-08 1980-03-07 Derives d'acides 1-omega-mercaptoacyl)-4,5-dihydropyrazole-5-carboxyliques et leur procede de preparation BE882133A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/018,548 US4211786A (en) 1979-03-08 1979-03-08 Mercaptoacyldihydropyrazole carboxylic acid derivatives

Publications (1)

Publication Number Publication Date
BE882133A true BE882133A (fr) 1980-09-08

Family

ID=21788501

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/199718A BE882133A (fr) 1979-03-08 1980-03-07 Derives d'acides 1-omega-mercaptoacyl)-4,5-dihydropyrazole-5-carboxyliques et leur procede de preparation

Country Status (16)

Country Link
US (1) US4211786A (fr)
JP (1) JPS55122766A (fr)
AU (1) AU534582B2 (fr)
BE (1) BE882133A (fr)
CA (1) CA1137497A (fr)
CH (1) CH645630A5 (fr)
DE (1) DE3008904A1 (fr)
DK (1) DK99980A (fr)
FR (1) FR2450820A1 (fr)
GB (1) GB2048850B (fr)
IE (1) IE49541B1 (fr)
IT (1) IT1127384B (fr)
LU (1) LU82223A1 (fr)
NL (1) NL8001349A (fr)
SE (1) SE450382B (fr)
ZA (1) ZA801016B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA794723B (en) * 1978-09-11 1980-08-27 Univ Miami Anti-hypertensive agents
US4331806A (en) * 1979-07-30 1982-05-25 E. R. Squibb & Sons, Inc. Dithioacyldihydropyrazole carboxylic acid derivatives
US4288368A (en) * 1979-07-30 1981-09-08 E. R. Squibb & Sons, Inc. Dithioacylproline derivatives
US4266065A (en) * 1980-04-14 1981-05-05 E. R. Squibb & Sons, Inc. Mercaptoacyldihydropyrazole carboxylic acid derivatives
CA1156236A (fr) * 1979-10-25 1983-11-01 George C. Rovnyak Derives de l'acide mercaptoacyldihydropyrazole carboxylique
US4254267A (en) * 1979-10-25 1981-03-03 E. R. Squibb & Sons, Inc. Mercaptoacyldihydropyrazole carboxylic acid derivatives
US4692458A (en) * 1980-03-05 1987-09-08 University Of Miami Anti-hypertensive agents
US4312990A (en) * 1980-09-11 1982-01-26 E. R. Squibb & Sons, Inc. 1-Mercaptoacyl-3-[(aminosulfonyl) phenyl]-4,5-dihydro-1H-pyrazole-5-carboxylic acid
US4371526A (en) * 1981-08-21 1983-02-01 E. R. Squibb & Sons, Inc. Phosphinylalkanoyl substituted 4,5-dihydropyrazole-5-carboxylic acid derivatives and hypotensive method and composition
JPS58133376U (ja) * 1982-03-05 1983-09-08 吉原 靖人 バツテイング練習用バツト
US4470973A (en) * 1982-07-19 1984-09-11 E. R. Squibb & Sons, Inc. Substituted peptide compounds
US4742067A (en) * 1982-07-22 1988-05-03 E. R. Squibb & Sons, Inc. Acylalkylaminocarbonyl substituted amino and imino acid compounds
US4621092A (en) * 1982-07-22 1986-11-04 E. R. Squibb & Sons, Inc. Substituted proline compounds, composition and method of use

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4105776A (en) * 1976-06-21 1978-08-08 E. R. Squibb & Sons, Inc. Proline derivatives and related compounds
US4046889A (en) * 1976-02-13 1977-09-06 E. R. Squibb & Sons, Inc. Azetidine-2-carboxylic acid derivatives
US4053651A (en) * 1976-05-10 1977-10-11 E. R. Squibb & Sons, Inc. Compounds and method for alleviating angiotensin related hypertension
ZA777062B (en) * 1976-12-03 1979-02-28 Squibb & Sons Inc Derivatives of thiazolidinecarboxylic acids and related acids
US4129566A (en) * 1978-02-15 1978-12-12 E. R. Squibb & Sons, Inc. Derivatives of dehydrocyclicimino acids

Also Published As

Publication number Publication date
ZA801016B (en) 1981-02-25
CH645630A5 (de) 1984-10-15
CA1137497A (fr) 1982-12-14
DE3008904A1 (de) 1980-09-18
FR2450820A1 (fr) 1980-10-03
NL8001349A (nl) 1980-09-10
JPS55122766A (en) 1980-09-20
AU534582B2 (en) 1984-02-09
LU82223A1 (de) 1980-09-24
DK99980A (da) 1980-09-09
SE450382B (sv) 1987-06-22
IE49541B1 (en) 1985-10-30
IT8048062A0 (it) 1980-03-03
US4211786A (en) 1980-07-08
FR2450820B1 (fr) 1983-04-22
AU5582280A (en) 1980-09-11
GB2048850A (en) 1980-12-17
IT1127384B (it) 1986-05-21
IE800449L (en) 1980-09-08
JPH0141628B2 (fr) 1989-09-06
GB2048850B (en) 1983-04-27
SE8001818L (sv) 1980-09-09

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: E.R. SQUIBB & SONS INC.

Effective date: 19940331