IT1265665B1 - Composizioni farmaceutiche comprendenti 8-cloro-3-(beta- dietilaminoetil)-4-metil-7-etossicarbonilmetossi cumarina base e - Google Patents

Composizioni farmaceutiche comprendenti 8-cloro-3-(beta- dietilaminoetil)-4-metil-7-etossicarbonilmetossi cumarina base e

Info

Publication number
IT1265665B1
IT1265665B1 IT93PD000141A ITPD930141A IT1265665B1 IT 1265665 B1 IT1265665 B1 IT 1265665B1 IT 93PD000141 A IT93PD000141 A IT 93PD000141A IT PD930141 A ITPD930141 A IT PD930141A IT 1265665 B1 IT1265665 B1 IT 1265665B1
Authority
IT
Italy
Prior art keywords
diethylaminoethyl
chloro
beta
methyl
pharmaceutical compositions
Prior art date
Application number
IT93PD000141A
Other languages
English (en)
Inventor
Rosa Massimo Di
Cirillo Rocco
Edward Joseph Hornby
Marco Prosdocimi
Original Assignee
Fidia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fidia Spa filed Critical Fidia Spa
Priority to IT93PD000141A priority Critical patent/IT1265665B1/it
Publication of ITPD930141A0 publication Critical patent/ITPD930141A0/it
Priority to PCT/EP1994/002008 priority patent/WO1995000142A1/en
Priority to AU71867/94A priority patent/AU7186794A/en
Publication of ITPD930141A1 publication Critical patent/ITPD930141A1/it
Application granted granted Critical
Publication of IT1265665B1 publication Critical patent/IT1265665B1/it

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • A61K31/366Lactones having six-membered rings, e.g. delta-lactones
    • A61K31/37Coumarins, e.g. psoralen

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invenzione si riferisce all'impiego del cloricromene (8-cloro-3-(Beta-dietilaminoetil)-4-metil-7-etossicarbonilmetossi cumarina) base e cloricromene cloridrato per la preparazione di composizioni farmaceutiche atte al trattamento di patologie caratterizzate da elevata produzione di ossido di azoto (NO) quali, in particolare, tutte quelle patologie in cui sia pregevole un'attività antiinfiammatoria e/o immunosoppressiva di suddetto farmaco, o più in generale in tutte quelle situazioni patologiche di vasodilatazione e/o danno tissutale conseguente ad iperproduzione di NO.
IT93PD000141A 1993-06-21 1993-06-21 Composizioni farmaceutiche comprendenti 8-cloro-3-(beta- dietilaminoetil)-4-metil-7-etossicarbonilmetossi cumarina base e IT1265665B1 (it)

Priority Applications (3)

Application Number Priority Date Filing Date Title
IT93PD000141A IT1265665B1 (it) 1993-06-21 1993-06-21 Composizioni farmaceutiche comprendenti 8-cloro-3-(beta- dietilaminoetil)-4-metil-7-etossicarbonilmetossi cumarina base e
PCT/EP1994/002008 WO1995000142A1 (en) 1993-06-21 1994-06-20 NEW PHARMACEUTICAL PREPARATIONS, CONTAINING 8-CHLORO-3(betaDIETHYLAMINOETHYL)-4-METHYL-7-ETHOXYCARBONYLMETHOXY COUMARIN AND THE SALTS THEREOF, IN THE TREATMENT OF PATHOLOGICAL CONDITIONS INVOLVING HIGH RELEASE OF NITRIC OXIDE
AU71867/94A AU7186794A (en) 1993-06-21 1994-06-20 New pharmaceutical preparations, containing 8-chloro-3(betadiethylaminoethyl)-4-methyl-7-ethoxycarbonylm ethoxy coumarin and the salts thereof, in the treatment of pathological conditions involving high release of nitric oxide

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT93PD000141A IT1265665B1 (it) 1993-06-21 1993-06-21 Composizioni farmaceutiche comprendenti 8-cloro-3-(beta- dietilaminoetil)-4-metil-7-etossicarbonilmetossi cumarina base e

Publications (3)

Publication Number Publication Date
ITPD930141A0 ITPD930141A0 (it) 1993-06-21
ITPD930141A1 ITPD930141A1 (it) 1994-12-21
IT1265665B1 true IT1265665B1 (it) 1996-11-22

Family

ID=11390384

Family Applications (1)

Application Number Title Priority Date Filing Date
IT93PD000141A IT1265665B1 (it) 1993-06-21 1993-06-21 Composizioni farmaceutiche comprendenti 8-cloro-3-(beta- dietilaminoetil)-4-metil-7-etossicarbonilmetossi cumarina base e

Country Status (3)

Country Link
AU (1) AU7186794A (it)
IT (1) IT1265665B1 (it)
WO (1) WO1995000142A1 (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1317356B1 (it) * 2000-07-31 2003-06-16 Fidia S P A Ora Fidia Farmaceu Derivati della cumarina e relativi sali, processo per la loropreparazione e loro impiego in campo farmaceutico.
WO2002024191A1 (fr) * 2000-09-20 2002-03-28 Yong Guang Pharmaceutical Co., Ltd. Medicament permettant de traiter et de prevenir la myopie

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1088554B (it) * 1977-11-17 1985-06-10 F I D I A Spa Procedimento sellettivo per la preparazione di derivati della 7-indrossi cumarina

Also Published As

Publication number Publication date
AU7186794A (en) 1995-01-17
ITPD930141A1 (it) 1994-12-21
WO1995000142A1 (en) 1995-01-05
ITPD930141A0 (it) 1993-06-21

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IT1265665B1 (it) Composizioni farmaceutiche comprendenti 8-cloro-3-(beta- dietilaminoetil)-4-metil-7-etossicarbonilmetossi cumarina base e

Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19980515