IT1171557B - Composizione farmaceutica a base di un sale di 1-(2,3,4-trimetossibenzil)-piperazina in particolare ad azione anti-ischemica - Google Patents

Composizione farmaceutica a base di un sale di 1-(2,3,4-trimetossibenzil)-piperazina in particolare ad azione anti-ischemica

Info

Publication number
IT1171557B
IT1171557B IT49377/81A IT4937781A IT1171557B IT 1171557 B IT1171557 B IT 1171557B IT 49377/81 A IT49377/81 A IT 49377/81A IT 4937781 A IT4937781 A IT 4937781A IT 1171557 B IT1171557 B IT 1171557B
Authority
IT
Italy
Prior art keywords
trimetossibenzil
piperazine
salt
pharmaceutical composition
composition based
Prior art date
Application number
IT49377/81A
Other languages
English (en)
Italian (it)
Other versions
IT8149377A0 (it
Inventor
Jean Claude Arnaud
Michelle Devissaguet
Original Assignee
Science Union & Cie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9246419&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IT1171557(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Science Union & Cie filed Critical Science Union & Cie
Publication of IT8149377A0 publication Critical patent/IT8149377A0/it
Application granted granted Critical
Publication of IT1171557B publication Critical patent/IT1171557B/it

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
IT49377/81A 1980-09-30 1981-09-28 Composizione farmaceutica a base di un sale di 1-(2,3,4-trimetossibenzil)-piperazina in particolare ad azione anti-ischemica IT1171557B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8020919A FR2490963B1 (fr) 1980-09-30 1980-09-30 Nouvelle composition therapeutique a action anti-ischemique contenant de la trimethoxy 2, 3, 4-benzyl 1-piperazine

Publications (2)

Publication Number Publication Date
IT8149377A0 IT8149377A0 (it) 1981-09-28
IT1171557B true IT1171557B (it) 1987-06-10

Family

ID=9246419

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49377/81A IT1171557B (it) 1980-09-30 1981-09-28 Composizione farmaceutica a base di un sale di 1-(2,3,4-trimetossibenzil)-piperazina in particolare ad azione anti-ischemica

Country Status (14)

Country Link
US (1) US4407801A (en, 2012)
AU (1) AU550761B2 (en, 2012)
BE (1) BE890568A (en, 2012)
CA (1) CA1169775A (en, 2012)
CH (1) CH650675A5 (en, 2012)
DE (1) DE3139005A1 (en, 2012)
FR (1) FR2490963B1 (en, 2012)
GB (1) GB2084019B (en, 2012)
GR (1) GR75803B (en, 2012)
IE (1) IE51764B1 (en, 2012)
IT (1) IT1171557B (en, 2012)
LU (1) LU83654A1 (en, 2012)
NZ (1) NZ198435A (en, 2012)
ZA (1) ZA816766B (en, 2012)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4448776A (en) * 1981-02-12 1984-05-15 Karl Bucher Method of using certain substituted aliphatic secondary amines or their salts for easing breathing
SE8403912D0 (sv) * 1984-07-30 1984-07-30 Pharmacia Ab Lekemedelssats eller -komposition
FR2717687B1 (fr) * 1994-03-24 1996-06-14 Adir Compositions pharmaceutiques permettant la libération prolongée de trimétazidine après administration par voie orale.
EP1104673A1 (en) * 1999-11-30 2001-06-06 Bayer Classics A hydrogen carbonate-containing, desintegrating agent-free pharmaceutical composition
FR2802424B1 (fr) * 1999-12-17 2002-02-15 Adir Comprime matriciel permettant la liberation prolongee de trimetazidine apres administration par voie orale
FR2805463B1 (fr) * 2000-02-25 2003-01-24 Adir UTILISATION DE LA TRIMETAZIDINE POUR L'OBTENTION DE COMPOSITIONS PHARMACEUTIQUES DESTINEES A INHIBER L'ACYL-CoA ACETYLTRANSFERASE
FR2818549B1 (fr) * 2000-12-26 2003-02-07 Servier Lab Composition pharmaceutique solide thermoformable pour la liberation controlee de trimetazidine
WO2007116243A2 (en) * 2006-04-10 2007-10-18 Mintails Limited Method for treating fibromyalgia and related conditions
EA009776B1 (ru) * 2006-07-18 2008-04-28 Мераб Ревазович Кокеладзе Способ изготовления таблетированной лекарственной формы триметазидина дигидрохлорида и ее состав
FR2986431B1 (fr) * 2012-02-03 2017-03-17 Servier Lab Composition pharmaceutique a liberation prolongee de trimetazidine, son procede de fabrication et son utilisation dans des traitements therapeutiques
US8920855B1 (en) 2012-10-30 2014-12-30 Setem Hemth, Inc Methods of topically treating tinnitus and related disorders
CN105055352A (zh) * 2015-08-11 2015-11-18 瑞阳制药有限公司 盐酸曲美他嗪片及其制备方法
EP3525771A4 (en) * 2016-11-21 2020-05-27 Saghmos Therapeutics, Inc. PREVENTION AND / OR TREATMENT OF ACUTE RENAL FAILURE INDUCED BY CONTRAST AGENTS
CN107982231B (zh) * 2018-01-03 2021-05-07 江苏吴中医药集团有限公司 一种盐酸曲美他嗪片及其制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3262852A (en) * 1966-07-26 Vasodilator and anti-anginose com- pounds containing methoxy benzyl piperazines and method of using the same
FR805M (en, 2012) * 1960-06-30 1961-09-01

Also Published As

Publication number Publication date
GB2084019B (en) 1984-09-12
US4407801A (en) 1983-10-04
ZA816766B (en) 1982-09-29
AU550761B2 (en) 1986-04-10
GR75803B (en, 2012) 1984-08-02
IE812256L (en) 1982-03-30
IT8149377A0 (it) 1981-09-28
FR2490963A1 (fr) 1982-04-02
DE3139005A1 (de) 1982-05-06
LU83654A1 (fr) 1982-04-14
AU7574481A (en) 1982-04-08
CA1169775A (fr) 1984-06-26
CH650675A5 (fr) 1985-08-15
NZ198435A (en) 1984-02-03
GB2084019A (en) 1982-04-07
FR2490963B1 (fr) 1986-04-18
BE890568A (fr) 1982-03-30
IE51764B1 (en) 1987-03-18

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Effective date: 19960926