IT1107454B - Derivati alfa-alogenometilici di amminoacidi e relativo procedimento di produzione - Google Patents

Derivati alfa-alogenometilici di amminoacidi e relativo procedimento di produzione

Info

Publication number
IT1107454B
IT1107454B IT50463/78A IT5046378A IT1107454B IT 1107454 B IT1107454 B IT 1107454B IT 50463/78 A IT50463/78 A IT 50463/78A IT 5046378 A IT5046378 A IT 5046378A IT 1107454 B IT1107454 B IT 1107454B
Authority
IT
Italy
Prior art keywords
halogenometyl
alpha
derivatives
amino acids
production process
Prior art date
Application number
IT50463/78A
Other languages
English (en)
Italian (it)
Other versions
IT7850463A0 (it
Original Assignee
Merrell Toraude & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Toraude & Co filed Critical Merrell Toraude & Co
Publication of IT7850463A0 publication Critical patent/IT7850463A0/it
Application granted granted Critical
Publication of IT1107454B publication Critical patent/IT1107454B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IT50463/78A 1977-07-28 1978-07-25 Derivati alfa-alogenometilici di amminoacidi e relativo procedimento di produzione IT1107454B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/819,975 US4315095A (en) 1977-07-28 1977-07-28 α-Halomethyl derivatives of amino acids

Publications (2)

Publication Number Publication Date
IT7850463A0 IT7850463A0 (it) 1978-07-25
IT1107454B true IT1107454B (it) 1985-11-25

Family

ID=25229573

Family Applications (1)

Application Number Title Priority Date Filing Date
IT50463/78A IT1107454B (it) 1977-07-28 1978-07-25 Derivati alfa-alogenometilici di amminoacidi e relativo procedimento di produzione

Country Status (16)

Country Link
US (1) US4315095A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JPS5436262A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU521354B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BE (1) BE869322A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA1120041A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CH (1) CH638790A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE2832309A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES471594A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2398736A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB2001626B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IE (1) IE46928B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL54914A0 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IT (1) IT1107454B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NL (1) NL7807871A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NZ (1) NZ187537A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ZA (1) ZA783350B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4413141A (en) * 1977-07-11 1983-11-01 Merrell Toraude Et Compagnie 2-(Difluoromethyl)-2,5-diaminopentanoic acid
US4347374A (en) 1980-07-21 1982-08-31 Merck & Co., Inc. Acid addition salts of N-trityl-α-fluoromethylhistidine enantiomer derivatives
JPS591490A (ja) * 1982-06-29 1984-01-06 Dai Ichi Seiyaku Co Ltd 3−セフェム−4−カルボン酸誘導体
CA1302919C (en) * 1985-07-03 1992-06-09 Robert T. Buckler Histamine derivatives, immunogen conjugates and antibodies raised thereto
US5030645A (en) * 1990-10-15 1991-07-09 Merck & Co., Inc. Method of treating asthma using (S)-α-fluoromethyl-histidine and esters thereof
US6001926A (en) * 1997-10-02 1999-12-14 The United States Of America As Represented By The Secretary Of The Navy Fiber-reinforced phthalonitrile composite cured with low-reactivity aromatic amine curing agent
EP1321169A1 (en) * 2001-12-18 2003-06-25 Biofrontera Pharmaceuticals AG Combination of a serotonin receptor antagonist with a histidine decarboxylase inhibitor as a medicament

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3169971A (en) * 1965-02-16 A-alkyl histidines
GB715182A (en) * 1951-09-19 1954-09-08 Roche Products Ltd A novel imidazole derivative and process for the manufacture thereof
FR1493402A (fr) * 1962-01-22 1967-09-01 Merck & Co Inc Hydrazino-acides
US3387031A (en) * 1961-06-08 1968-06-04 Union Carbide Corp Synthesis of alpha-amino acid amide hydrohalides
FR1457259A (fr) * 1961-08-18 1966-01-24 Merck & Co Inc Production d'amino-acides du type alpha-alkyl-histidine
FR2392958A1 (fr) * 1977-06-01 1978-12-29 Merck & Co Inc Nouveaux amino-acides fluores utiles comme medicament

Also Published As

Publication number Publication date
AU3731778A (en) 1980-01-03
FR2398736B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1980-09-19
AU521354B2 (en) 1982-04-01
BE869322A (fr) 1978-11-16
CH638790A5 (de) 1983-10-14
ES471594A1 (es) 1979-10-01
DE2832309A1 (de) 1979-02-08
IT7850463A0 (it) 1978-07-25
US4315095A (en) 1982-02-09
IL54914A0 (en) 1978-08-31
NL7807871A (nl) 1979-01-30
FR2398736A1 (fr) 1979-02-23
DE2832309C2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1989-07-06
CA1120041A (en) 1982-03-16
JPS5436262A (en) 1979-03-16
GB2001626A (en) 1979-02-07
JPS6123792B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1986-06-07
ZA783350B (en) 1979-06-27
IE781149L (en) 1979-01-28
GB2001626B (en) 1982-04-07
NZ187537A (en) 1980-08-26
IE46928B1 (en) 1983-11-02

Similar Documents

Publication Publication Date Title
IT1112112B (it) Derivati acilici sostituiti di amminoacidi e relativo procedimento di produzione
IT7852280A0 (it) Procedimento per la produzione di derivati ammidici in particolare acilanilidi sostituite e prodotto ottenuto
IT1132392B (it) Derivati di acidi chinolincarbossilici e relativo procedimento di preparazione
IT1078981B (it) Derivati di acidi fenossi-fenossipropionici
IT7851499A0 (it) Procedimento per la produzione di derivati della xantina e prodotto relativo
IT1105176B (it) Derivati della morfina e relativo procedimento di produzione
IT1058013B (it) Derivati della salicilanilde e relativo procedimento di produzione
IT1092179B (it) Derivati di acidi tiazolidincarbossilici e elativo procedimento di produzione
BR7605959A (pt) Processo de preparacao de novos derivados de amidoxima e suas aplicacoes
IT1107454B (it) Derivati alfa-alogenometilici di amminoacidi e relativo procedimento di produzione
IT1105079B (it) Derivati alfa-acetilenici e vinilici di amminoacidi e relativo procedimento di produzione
IT1040613B (it) Derivati di 2 ammino 1 3 tiazina e procedimento per la loro produzione
IT1105172B (it) Derivati della morfina e relativo procedimento di produzione
IT1134448B (it) Derivati esterei di acidi ciclopropancarbossilici
IT1106121B (it) Derivati 25-alchilcolesterolici e relativo procedimento di produzione
IT1140954B (it) Amminpacil derivati di acidi mercaptoacil amminici
IT1113140B (it) Derivati di amminoalcoli
IT7821862A0 (it) Derivati di acidi ossi-alcanoici.
IT7850128A0 (it) Derivati di amminoacidi alfa-vinili ci utili in particolare come composti farmaceutici e relativo procedimento di produzione
IT7848192A0 (it) Procedimento per la produzione di derivati di 9-2-idrossietossimetilguanina e prodotto ottenuto
IT7850147A0 (it) Derivati di 4-omoisotwistano e relativo procedimento di produzione
IT1164693B (it) Derivati della idantoina e relativo procedimento di produzione
IT7850102A0 (it) Procedimento per la produzione di derivati di amminoacidi alfa-aceti lenici e prodotto ottenuto
IT1105099B (it) Derivati alfa-alogenometilici di alfa-amminoacidi e relativo procedimento di produzione
IT1105506B (it) Composizione farmaceutica comprendente prostaciclina o suoi derivati e relativo procedimento di produzione