IN2015DN01197A - - Google Patents
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- Publication number
- IN2015DN01197A IN2015DN01197A IN1197DEN2015A IN2015DN01197A IN 2015DN01197 A IN2015DN01197 A IN 2015DN01197A IN 1197DEN2015 A IN1197DEN2015 A IN 1197DEN2015A IN 2015DN01197 A IN2015DN01197 A IN 2015DN01197A
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- IN
- India
- Prior art keywords
- compounds
- cse
- lyase
- benefit
- conditions
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 3
- 102000004317 Lyases Human genes 0.000 abstract 1
- 108090000856 Lyases Proteins 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 230000005764 inhibitory process Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/18—Sulfonamides
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- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid
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- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4196—1,2,4-Triazoles
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- A61K31/445—Non condensed piperidines, e.g. piperocaine
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- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D249/04—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
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- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
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- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4245—Oxadiazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/04—Systems containing only non-condensed rings with a four-membered ring
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Dermatology (AREA)
- Pulmonology (AREA)
- Physical Education & Sports Medicine (AREA)
- Diabetes (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Immunology (AREA)
- Emergency Medicine (AREA)
- Hematology (AREA)
- Toxicology (AREA)
- Urology & Nephrology (AREA)
- Obesity (AREA)
- Endocrinology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261675753P | 2012-07-25 | 2012-07-25 | |
PCT/US2013/051744 WO2014018569A1 (fr) | 2012-07-25 | 2013-07-23 | Inhibiteurs de la cystathionine-y-gamma-lyase (cse) |
Publications (1)
Publication Number | Publication Date |
---|---|
IN2015DN01197A true IN2015DN01197A (fr) | 2015-06-26 |
Family
ID=49997790
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IN1197DEN2015 IN2015DN01197A (fr) | 2012-07-25 | 2015-02-13 |
Country Status (13)
Country | Link |
---|---|
US (2) | US9771339B2 (fr) |
EP (1) | EP2877458A4 (fr) |
JP (2) | JP6407864B2 (fr) |
KR (1) | KR20150041634A (fr) |
CN (2) | CN109748881A (fr) |
AR (1) | AR091858A1 (fr) |
AU (2) | AU2013293089A1 (fr) |
CA (1) | CA2879986C (fr) |
HK (1) | HK1210615A1 (fr) |
IN (1) | IN2015DN01197A (fr) |
RU (1) | RU2640418C2 (fr) |
TW (1) | TWI606040B (fr) |
WO (1) | WO2014018569A1 (fr) |
Families Citing this family (23)
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CA2856520C (fr) | 2011-11-23 | 2021-04-06 | Therapeuticsmd, Inc. | Preparations et therapies de substitution pour hormonotherapie naturelle combinee |
US9301920B2 (en) | 2012-06-18 | 2016-04-05 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
US10806740B2 (en) | 2012-06-18 | 2020-10-20 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
US10806697B2 (en) | 2012-12-21 | 2020-10-20 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US20150196640A1 (en) | 2012-06-18 | 2015-07-16 | Therapeuticsmd, Inc. | Progesterone formulations having a desirable pk profile |
US20130338122A1 (en) | 2012-06-18 | 2013-12-19 | Therapeuticsmd, Inc. | Transdermal hormone replacement therapies |
AR091858A1 (es) | 2012-07-25 | 2015-03-04 | Sova Pharmaceuticals Inc | INHIBIDORES DE CISTATIONIN-g-LIASA (CSE) |
US11246875B2 (en) | 2012-12-21 | 2022-02-15 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US10568891B2 (en) | 2012-12-21 | 2020-02-25 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US11266661B2 (en) | 2012-12-21 | 2022-03-08 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US10471072B2 (en) | 2012-12-21 | 2019-11-12 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US9180091B2 (en) | 2012-12-21 | 2015-11-10 | Therapeuticsmd, Inc. | Soluble estradiol capsule for vaginal insertion |
US10537581B2 (en) | 2012-12-21 | 2020-01-21 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
EP3096755A4 (fr) * | 2014-01-23 | 2017-12-27 | Sova Pharmaceuticals, Inc. | Inhibiteurs de cystathionine- (gamma)-lyase (cse) pour le traitement de la douleur |
AU2015264003A1 (en) | 2014-05-22 | 2016-11-17 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
CA2975682A1 (fr) | 2015-02-13 | 2016-08-18 | Oxford Drug Design Limited | Derives de n-acyl-arylsulfonamide comme inhibiteurs d'aminoacyl-arnt synthetase |
US10328087B2 (en) | 2015-07-23 | 2019-06-25 | Therapeuticsmd, Inc. | Formulations for solubilizing hormones |
US20180313801A1 (en) * | 2015-10-21 | 2018-11-01 | Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College | Method for diagnosing rheumatoid arthritis |
WO2017173044A1 (fr) | 2016-04-01 | 2017-10-05 | Therapeuticsmd Inc. | Compositions d'hormones stéroïdes dans des huiles à chaîne moyenne |
CA3020153A1 (fr) | 2016-04-01 | 2017-10-05 | Therapeuticsmd, Inc. | Composition pharmaceutique d'hormone steroide |
GB201617064D0 (en) | 2016-10-07 | 2016-11-23 | Inhibox Limited And Latvian Institute Of Organic Synthesis The | Compounds and their therapeutic use |
CA3107412A1 (fr) * | 2018-11-30 | 2020-06-04 | Amerilab Technologies, Inc. | Comprimes effervescents comprenant un liant de sucre cristallin et leurs procedes de fabrication |
CN111233704B (zh) * | 2020-03-16 | 2023-01-06 | 湖北三宁碳磷基新材料产业技术研究院有限公司 | 一种制备6-氨基己腈产品的方法 |
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US4229447A (en) | 1979-06-04 | 1980-10-21 | American Home Products Corporation | Intraoral methods of using benzodiazepines |
US4476116A (en) | 1982-12-10 | 1984-10-09 | Syntex (U.S.A.) Inc. | Polypeptides/chelating agent nasal compositions having enhanced peptide absorption |
US5116817A (en) | 1982-12-10 | 1992-05-26 | Syntex (U.S.A.) Inc. | LHRH preparations for intranasal administration |
US4596795A (en) | 1984-04-25 | 1986-06-24 | The United States Of America As Represented By The Secretary, Dept. Of Health & Human Services | Administration of sex hormones in the form of hydrophilic cyclodextrin derivatives |
DE3684446D1 (de) | 1985-12-28 | 1992-04-23 | Sumitomo Pharma | Arzneimittel mit verzoegerter stossweiser freisetzung. |
US4755386A (en) | 1986-01-22 | 1988-07-05 | Schering Corporation | Buccal formulation |
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US5739136A (en) | 1989-10-17 | 1998-04-14 | Ellinwood, Jr.; Everett H. | Intraoral dosing method of administering medicaments |
US5017381A (en) | 1990-05-02 | 1991-05-21 | Alza Corporation | Multi-unit pulsatile delivery system |
US5229135A (en) | 1991-11-22 | 1993-07-20 | Prographarm Laboratories | Sustained release diltiazem formulation |
DE4211536A1 (de) | 1992-04-06 | 1993-10-07 | Hoechst Ag | Verfahren zur Herstellung von Derivaten der Bis(aminomethyl)phosphinsäure |
US5837284A (en) | 1995-12-04 | 1998-11-17 | Mehta; Atul M. | Delivery of multiple doses of medications |
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US6391452B1 (en) | 1997-07-18 | 2002-05-21 | Bayer Corporation | Compositions for nasal drug delivery, methods of making same, and methods of removing residual solvent from pharmaceutical preparations |
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CN100580087C (zh) * | 2003-10-10 | 2010-01-13 | 诺和诺德医疗保健公司 | 肽的缀合 |
WO2005049602A1 (fr) | 2003-11-18 | 2005-06-02 | Warner-Lambert Company Llc | Agents antibacteriens a la quinolone |
DE102005022977A1 (de) | 2005-05-19 | 2006-12-07 | Merck Patent Gmbh | Phenylchinazolinderivate |
WO2007005737A2 (fr) * | 2005-07-01 | 2007-01-11 | Case Western Reserve University | Inhibiteurs d'amine oxydase |
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ATE524454T1 (de) * | 2006-11-01 | 2011-09-15 | Chroma Therapeutics Ltd | Inhibitoren von ikk-beta serinthreoninproteinkinase |
TW200906818A (en) | 2007-07-31 | 2009-02-16 | Astrazeneca Ab | Chemical compounds |
EP2296659B1 (fr) | 2008-06-05 | 2016-12-21 | Janssen Pharmaceutica, N.V. | Combinaisons de médicaments comprenant un inhibiteur de DGAT et un agoniste de PPAR |
CN102227425A (zh) * | 2008-09-26 | 2011-10-26 | 贝林格尔·英格海姆国际有限公司 | 作为ccr1受体拮抗剂的氮杂吲唑化合物 |
US8633322B2 (en) | 2009-10-29 | 2014-01-21 | Janssen Pharmaceutica Nv | Alkynyl derivatives useful as DPP-1 inhibitors |
US8481547B2 (en) | 2009-12-18 | 2013-07-09 | Janssen Pharmaceutica Nv | Substituted benzothiazole and benzoxazole derivatives useful as inhibitors of DPP-1 |
AR091858A1 (es) | 2012-07-25 | 2015-03-04 | Sova Pharmaceuticals Inc | INHIBIDORES DE CISTATIONIN-g-LIASA (CSE) |
WO2014018571A2 (fr) * | 2012-07-25 | 2014-01-30 | Sova Pharmaceuticals, Inc. | Utilisation d'inhibiteurs de cse pour le traitement de lésions ou d'affections cutanées et de troubles respiratoires du sommeil |
EP3096755A4 (fr) * | 2014-01-23 | 2017-12-27 | Sova Pharmaceuticals, Inc. | Inhibiteurs de cystathionine- (gamma)-lyase (cse) pour le traitement de la douleur |
-
2013
- 2013-07-22 AR ARP130102599A patent/AR091858A1/es unknown
- 2013-07-23 RU RU2015105893A patent/RU2640418C2/ru active
- 2013-07-23 CN CN201811165284.4A patent/CN109748881A/zh active Pending
- 2013-07-23 CN CN201380049533.2A patent/CN104684901A/zh active Pending
- 2013-07-23 US US14/416,574 patent/US9771339B2/en not_active Expired - Fee Related
- 2013-07-23 AU AU2013293089A patent/AU2013293089A1/en not_active Abandoned
- 2013-07-23 EP EP13823562.7A patent/EP2877458A4/fr not_active Withdrawn
- 2013-07-23 KR KR1020157004421A patent/KR20150041634A/ko not_active Application Discontinuation
- 2013-07-23 CA CA2879986A patent/CA2879986C/fr not_active Expired - Fee Related
- 2013-07-23 WO PCT/US2013/051744 patent/WO2014018569A1/fr active Application Filing
- 2013-07-23 JP JP2015524401A patent/JP6407864B2/ja not_active Expired - Fee Related
- 2013-07-24 TW TW102126482A patent/TWI606040B/zh not_active IP Right Cessation
-
2015
- 2015-02-13 IN IN1197DEN2015 patent/IN2015DN01197A/en unknown
- 2015-11-18 HK HK15111387.1A patent/HK1210615A1/xx unknown
-
2017
- 2017-08-09 US US15/672,511 patent/US10227314B2/en not_active Expired - Fee Related
-
2018
- 2018-01-25 AU AU2018200635A patent/AU2018200635B2/en not_active Ceased
- 2018-06-07 JP JP2018109810A patent/JP2018172397A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
TWI606040B (zh) | 2017-11-21 |
US20170334866A1 (en) | 2017-11-23 |
EP2877458A1 (fr) | 2015-06-03 |
JP6407864B2 (ja) | 2018-10-17 |
HK1210615A1 (en) | 2016-04-29 |
TW201406732A (zh) | 2014-02-16 |
KR20150041634A (ko) | 2015-04-16 |
WO2014018569A1 (fr) | 2014-01-30 |
CA2879986C (fr) | 2020-09-29 |
US20150175561A1 (en) | 2015-06-25 |
EP2877458A4 (fr) | 2016-08-10 |
AU2013293089A1 (en) | 2015-02-19 |
CN109748881A (zh) | 2019-05-14 |
CA2879986A1 (fr) | 2014-01-30 |
CN104684901A (zh) | 2015-06-03 |
AU2018200635B2 (en) | 2019-07-04 |
AR091858A1 (es) | 2015-03-04 |
RU2015105893A (ru) | 2016-09-10 |
JP2015530368A (ja) | 2015-10-15 |
US10227314B2 (en) | 2019-03-12 |
RU2640418C2 (ru) | 2018-01-09 |
US9771339B2 (en) | 2017-09-26 |
AU2018200635A1 (en) | 2018-02-15 |
JP2018172397A (ja) | 2018-11-08 |
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