IN2013MU01468A - - Google Patents

Info

Publication number
IN2013MU01468A
IN2013MU01468A IN1468MU2013A IN2013MU01468A IN 2013MU01468 A IN2013MU01468 A IN 2013MU01468A IN 1468MU2013 A IN1468MU2013 A IN 1468MU2013A IN 2013MU01468 A IN2013MU01468 A IN 2013MU01468A
Authority
IN
India
Prior art keywords
compound
formula
fatty liver
nonalcoholic
liver
Prior art date
Application number
Other languages
English (en)
Inventor
Pankaj Patel
Jani Rajendrakumar Hariprasad
Original Assignee
Cadila Healthcare Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to AU2013387996A priority Critical patent/AU2013387996B2/en
Priority to BR112015020600A priority patent/BR112015020600A2/pt
Priority to CN201380075905.9A priority patent/CN105377246B/zh
Priority to MA38385A priority patent/MA38385A1/fr
Priority to PCT/IN2013/000391 priority patent/WO2014174524A1/fr
Priority to US14/782,609 priority patent/US20160166539A1/en
Priority to IN1468MU2013 priority patent/IN2013MU01468A/en
Priority to EA201592020A priority patent/EA201592020A1/ru
Priority to JP2016505927A priority patent/JP6246895B2/ja
Priority to CA2900435A priority patent/CA2900435C/fr
Priority to SG11201506218UA priority patent/SG11201506218UA/en
Priority to GEAP201313941A priority patent/GEP201706663B/en
Application filed by Cadila Healthcare Ltd filed Critical Cadila Healthcare Ltd
Priority to UAA201509744A priority patent/UA114360C2/uk
Priority to KR1020157024370A priority patent/KR101617812B1/ko
Priority to AP2015008674A priority patent/AP2015008674A0/xx
Priority to MX2015010769A priority patent/MX346943B/es
Priority to EP13767126.9A priority patent/EP2988736A1/fr
Priority to MYPI2015002026A priority patent/MY180160A/en
Publication of IN2013MU01468A publication Critical patent/IN2013MU01468A/en
Priority to IL240183A priority patent/IL240183A/en
Priority to PH12015501795A priority patent/PH12015501795A1/en
Priority to HK16103017.5A priority patent/HK1214968A1/zh
Priority to IL247231A priority patent/IL247231A/en
Priority to US15/343,859 priority patent/US9814697B2/en
Priority to US15/801,738 priority patent/US20180185330A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
IN1468MU2013 2013-04-22 2013-06-25 IN2013MU01468A (fr)

Priority Applications (24)

Application Number Priority Date Filing Date Title
UAA201509744A UA114360C2 (uk) 2013-04-22 2013-06-25 Спосіб лікування та/або зменшення інтенсивності неалкогольної жирової хвороби печінки (нжхп)
BR112015020600A BR112015020600A2 (pt) 2013-04-22 2013-06-25 composição farmacêutica, método para o tratamento de e/ou melhorar doenças de gordura no fígado de origem não alcoólica e uso da composição
KR1020157024370A KR101617812B1 (ko) 2013-04-22 2013-06-25 비알콜성 지방간 질환을 위한 신규 조성물
PCT/IN2013/000391 WO2014174524A1 (fr) 2013-04-22 2013-06-25 Nouvelle composition pour la stéatose hépatique non alcoolique (nafld)
US14/782,609 US20160166539A1 (en) 2013-04-22 2013-06-25 A novel composition for nonalcoholic fatty liver disease (nafld)
IN1468MU2013 IN2013MU01468A (fr) 2013-04-22 2013-06-25
EA201592020A EA201592020A1 (ru) 2013-04-22 2013-06-25 Новая композиция для неалкогольной жировой болезни печени (нажбп)
JP2016505927A JP6246895B2 (ja) 2013-04-22 2013-06-25 非アルコール性脂肪性肝疾患(nafld)のための新規組成物
CA2900435A CA2900435C (fr) 2013-04-22 2013-06-25 Nouvelle composition pour la steatose hepatique non alcoolique (nafld)
SG11201506218UA SG11201506218UA (en) 2013-04-22 2013-06-25 A novel composition for nonalcoholic fatty liver disease (nafld)
GEAP201313941A GEP201706663B (en) 2013-04-22 2013-06-25 Novel composition for nonalcoholic fatty liver disease (nafld
AU2013387996A AU2013387996B2 (en) 2013-04-22 2013-06-25 A novel composition for nonalcoholic fatty liver disease (NAFLD)
CN201380075905.9A CN105377246B (zh) 2013-04-22 2013-06-25 针对非酒精性脂肪性肝病(nafld)的新组合物
MA38385A MA38385A1 (fr) 2013-04-22 2013-06-25 Nouvelle composition pour la stéatose hépatique non alcoolique (nafld)
AP2015008674A AP2015008674A0 (en) 2013-04-22 2013-06-25 A novel composition for nonalcoholic fatty liver disease (NAFLD)
MX2015010769A MX346943B (es) 2013-04-22 2013-06-25 Una nueva composición para esteatosis hepática no alcohólica (nafld).
EP13767126.9A EP2988736A1 (fr) 2013-04-22 2013-06-25 Nouvelle composition pour la stéatose hépatique non alcoolique (nafld)
MYPI2015002026A MY180160A (en) 2013-04-22 2013-06-25 A novel composition for nonalcoholic fatty liver disease (nafld)
IL240183A IL240183A (en) 2013-04-22 2015-07-28 Non-Alcoholic Obesity Preparation (nafld)
PH12015501795A PH12015501795A1 (en) 2013-04-22 2015-08-14 A novel composition for nonalcoholic fatty liver disease (nafld)
HK16103017.5A HK1214968A1 (zh) 2013-04-22 2016-03-15 用於非酒精性脂肪肝病 的新組合物
IL247231A IL247231A (en) 2013-04-22 2016-08-11 Preparation for the treatment of non-alcoholic obesity
US15/343,859 US9814697B2 (en) 2013-04-22 2016-11-04 Composition for nonalcoholic fatty liver disease (NAFLD)
US15/801,738 US20180185330A1 (en) 2013-04-22 2017-11-02 Novel composition for nonalcoholic fatty liver disease (nafld)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN1468MU2013 IN2013MU01468A (fr) 2013-04-22 2013-06-25

Publications (1)

Publication Number Publication Date
IN2013MU01468A true IN2013MU01468A (fr) 2015-04-17

Family

ID=49253372

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1468MU2013 IN2013MU01468A (fr) 2013-04-22 2013-06-25

Country Status (21)

Country Link
US (3) US20160166539A1 (fr)
EP (1) EP2988736A1 (fr)
JP (1) JP6246895B2 (fr)
KR (1) KR101617812B1 (fr)
CN (1) CN105377246B (fr)
AP (1) AP2015008674A0 (fr)
AU (1) AU2013387996B2 (fr)
BR (1) BR112015020600A2 (fr)
CA (1) CA2900435C (fr)
EA (1) EA201592020A1 (fr)
GE (1) GEP201706663B (fr)
HK (1) HK1214968A1 (fr)
IL (2) IL240183A (fr)
IN (1) IN2013MU01468A (fr)
MA (1) MA38385A1 (fr)
MX (1) MX346943B (fr)
MY (1) MY180160A (fr)
PH (1) PH12015501795A1 (fr)
SG (1) SG11201506218UA (fr)
UA (1) UA114360C2 (fr)
WO (1) WO2014174524A1 (fr)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3009136A1 (fr) 2011-01-31 2016-04-20 Cadila Healthcare Limited Traitement de la lipodystrophie
US20130158077A1 (en) 2011-12-19 2013-06-20 Ares Trading S.A. Pharmaceutical compositions
UA114360C2 (uk) 2013-04-22 2017-05-25 Каділа Хелткере Лімітед Спосіб лікування та/або зменшення інтенсивності неалкогольної жирової хвороби печінки (нжхп)
US20160107989A1 (en) 2013-05-30 2016-04-21 Cadila Healthcare Limited A process for preparation of pyrroles having hypolipidemic hypocholesteremic activities
TW201636015A (zh) 2013-07-05 2016-10-16 卡地拉保健有限公司 協同性組成物
IN2013MU02470A (fr) * 2013-07-25 2015-06-26 Cadila Healthcare Ltd
US10112898B2 (en) 2013-09-06 2018-10-30 Cadila Healthcare Limited Process for the preparation of saroglitazar pharmaceutical salts
WO2017064635A2 (fr) 2015-10-14 2017-04-20 Cadila Healthcare Limited Composé pyrrole, compositions et procédé de préparation associé
US20180243263A1 (en) * 2016-12-09 2018-08-30 Cadila Healthcare Ltd. Treatment for primary biliary cholangitis
PL3600309T3 (pl) 2017-03-28 2022-11-07 Gilead Sciences, Inc. Skojarzenia terapeutyczne do leczenia chorób wątroby
GB201710229D0 (en) * 2017-06-27 2017-08-09 Tdeltas Ltd Compounds for new use
TWI814744B (zh) * 2017-10-06 2023-09-11 美商基利科學股份有限公司 包含acc抑制劑之組合療法
CN109675016A (zh) * 2017-10-18 2019-04-26 上海贺普药业股份有限公司 非酒精性脂肪性肝病的治疗药物
CN110934866B (zh) * 2018-09-25 2023-12-01 深圳微芯生物科技股份有限公司 西格列羧及其相关化合物的应用
US20220071954A1 (en) * 2018-12-18 2022-03-10 Cadila Healthcare Limited Saroglitazar for the treatment of hepatocellular carcinoma
US20220175721A1 (en) * 2019-02-13 2022-06-09 Cadila Healthcare Limited Treatment for polycystic ovarian syndrome (pcos)
WO2022246243A1 (fr) * 2021-05-21 2022-11-24 HepQuant, LLC Procédés de définition d'un changement fonctionnel et de ralentissement de la progression dans une maladie hépatique chronique

Family Cites Families (42)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4231938A (en) 1979-06-15 1980-11-04 Merck & Co., Inc. Hypocholesteremic fermentation products and process of preparation
US4444784A (en) 1980-08-05 1984-04-24 Merck & Co., Inc. Antihypercholesterolemic compounds
MX7065E (es) 1980-06-06 1987-04-10 Sankyo Co Un procedimiento microbiologico para preparar derivados de ml-236b
US5354772A (en) 1982-11-22 1994-10-11 Sandoz Pharm. Corp. Indole analogs of mevalonolactone and derivatives thereof
FI94339C (fi) 1989-07-21 1995-08-25 Warner Lambert Co Menetelmä farmaseuttisesti käyttökelpoisen /R-(R*,R*)/-2-(4-fluorifenyyli)- , -dihydroksi-5-(1-metyylietyyli)-3-fenyyli-4-/(fenyyliamino)karbonyyli/-1H-pyrroli-1-heptaanihapon ja sen farmaseuttisesti hyväksyttävien suolojen valmistamiseksi
US5089514A (en) 1990-06-14 1992-02-18 Pfizer Inc. 3-coxazolyl [phenyl, chromanyl or benzofuranyl]-2-hydroxypropionic acid derivatives and analogs as hypoglycemic agents
NZ253742A (en) 1992-07-03 1997-06-24 Smithkline Beecham Plc Heterocyclylaminoalkoxy substituted phenyl derivatives and pharmaceutical compositions
GB9225386D0 (en) 1992-12-04 1993-01-27 Smithkline Beecham Plc Novel compounds
US5387613A (en) 1993-07-23 1995-02-07 Ribogene, Inc. Treatment of tachyarrhythmias of supraventricular origin
GB9326171D0 (en) 1993-12-22 1994-02-23 Smithkline Beecham Plc Novel compounds
BR9508468A (pt) 1994-07-29 1997-11-25 Smithkline Beecham Plc Composto processo para a preparação do mesmo composição farmacéutica processos para o tratamento e/ou profilaxia de hiperglicemia em um mamifero humano ou não humano e para o tratamento de hiperlípidemia hipertensão doença cardiovascular alguns distúrbios de alimentação o tratamento e/ou profilaxia de doença renal a prevenção revers o estabilização ou retardo da progressão de microalbuminuria em um mamifero humano ou não humano uso do composto e composto intermediário
WO1996033998A1 (fr) 1995-04-28 1996-10-31 Daiichi Pharmaceutical Co., Ltd. Composes pentacycliques
GB9600464D0 (en) 1996-01-09 1996-03-13 Smithkline Beecham Plc Novel method
GB9606805D0 (en) 1996-03-30 1996-06-05 Glaxo Wellcome Inc Medicaments
AU1198699A (en) 1997-10-27 1999-04-23 Dr. Reddy's Research Foundation Novel heterocyclic compounds and their use in medicine, process for their reparation and pharmaceutical compositions containing them
WO1999019313A1 (fr) 1997-10-27 1999-04-22 Dr. Reddy's Research Foundation Nouveaux composes tricycliques et leur utilisation en medecine, procede de preparation de ces derniers et compositions pharmaceutiques les contenant
WO1999008501A2 (fr) 1998-04-23 1999-02-25 Dr. Reddy's Research Foundation Nouveaux composes heterocycliques, leur utilisation en medecine, leur procede de preparation et compositions pharmaceutiques les contenant
EP1082313A1 (fr) 1998-05-27 2001-03-14 Dr. Reddy's Research Foundation Composes bicycliques, procede de preparation et compositions pharmaceutiques les contenant
EP1123269A1 (fr) 1998-10-21 2001-08-16 Novo Nordisk A/S Nouveaux composes, leur preparation et leur utilisation
AU6325799A (en) 1998-10-21 2000-05-08 Dr. Reddy's Research Foundation New compounds, their preparation and use
AU6325599A (en) 1998-10-21 2000-05-08 Dr. Reddy's Research Foundation New compounds, their preparation and use
CO5150173A1 (es) 1998-12-10 2002-04-29 Novartis Ag Compuestos n-(glicilo sustituido)-2-cianopirrolidinas inhibidores de peptidasa de dipeptidilo-iv (dpp-iv) los cuales son efectivos en el tratamiento de condiciones mediadas por la inhibicion de dpp-iv
ES2449194T3 (es) 2000-01-19 2014-03-18 Cadila Healthcare Limited Compuestos que tienen actividades hipolipidémica e hipocolesterolémica, procedimiento para su preparación y composiciones farmacéuticas que los contienen
US6395767B2 (en) 2000-03-10 2002-05-28 Bristol-Myers Squibb Company Cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV and method
WO2002024625A2 (fr) 2000-09-22 2002-03-28 Dr. Reddy's Research Foundation Procede ameliore pour la preparation de derives d'acide 3-aryl-2-hydroxy propanoique
UA74912C2 (en) 2001-07-06 2006-02-15 Merck & Co Inc Beta-aminotetrahydroimidazo-(1,2-a)-pyrazines and tetratriazolo-(4,3-a)-pyrazines as inhibitors of dipeptylpeptidase for the treatment or prevention of diabetes
US6987123B2 (en) * 2001-07-26 2006-01-17 Cadila Healthcare Limited Heterocyclic compounds, their preparation, pharmaceutical compositions containing them and their use in medicine
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US20070051626A1 (en) 2003-09-26 2007-03-08 Chiho Itou Cataphoresis apparatus cataphoresis method, and detection method for organism-related material using the apparatus and the method
CN102079743B (zh) 2004-03-15 2020-08-25 武田药品工业株式会社 二肽基肽酶抑制剂
EA200800869A1 (ru) * 2005-09-19 2008-10-30 ДЖОНСОН ЭНД ДЖОНСОН ФАРМАСЬЮТИКАЛ РИСЕРЧ ЭНД ДИВЕЛОПМЕНТ, Эл. Эл. Си. Модуляция экспрессии рецептора глюкагона
JP5431940B2 (ja) * 2006-09-18 2014-03-05 アルナイラム ファーマシューティカルズ, インコーポレイテッド SCAPのRNAi調節およびその治療的使用
JP2008184429A (ja) * 2007-01-30 2008-08-14 Japan Health Science Foundation 肝臓トリグリセリド濃度低下剤
CN102647982B (zh) 2009-11-26 2014-10-15 基恩菲特公司 使用1,3-二苯基丙-2-烯-1-酮衍生物治疗肝脏疾患
RU2013121270A (ru) 2010-10-12 2014-11-20 Серекор Инк. Композиции против кашля, содержащие мемантин
EP3009136A1 (fr) * 2011-01-31 2016-04-20 Cadila Healthcare Limited Traitement de la lipodystrophie
UA114360C2 (uk) 2013-04-22 2017-05-25 Каділа Хелткере Лімітед Спосіб лікування та/або зменшення інтенсивності неалкогольної жирової хвороби печінки (нжхп)
US20160107989A1 (en) 2013-05-30 2016-04-21 Cadila Healthcare Limited A process for preparation of pyrroles having hypolipidemic hypocholesteremic activities
TW201636015A (zh) 2013-07-05 2016-10-16 卡地拉保健有限公司 協同性組成物
IN2013MU02470A (fr) 2013-07-25 2015-06-26 Cadila Healthcare Ltd
EP3039011A1 (fr) 2013-08-29 2016-07-06 Cadila Healthcare Limited Forme polymorphe de dérivé du pyrrole et intermédiaire
US10112898B2 (en) 2013-09-06 2018-10-30 Cadila Healthcare Limited Process for the preparation of saroglitazar pharmaceutical salts

Also Published As

Publication number Publication date
IL240183A0 (en) 2015-09-24
WO2014174524A1 (fr) 2014-10-30
AU2013387996B2 (en) 2015-12-10
US9814697B2 (en) 2017-11-14
MX2015010769A (es) 2015-11-26
WO2014174524A8 (fr) 2015-10-01
KR20150118990A (ko) 2015-10-23
EP2988736A1 (fr) 2016-03-02
GEP201706663B (en) 2017-05-10
EA201592020A1 (ru) 2016-05-31
HK1214968A1 (zh) 2016-08-12
CN105377246A (zh) 2016-03-02
UA114360C2 (uk) 2017-05-25
IL240183A (en) 2016-08-31
CN105377246B (zh) 2018-03-20
IL247231A (en) 2017-03-30
PH12015501795A1 (en) 2015-11-09
JP2016515608A (ja) 2016-05-30
US20160166539A1 (en) 2016-06-16
CA2900435A1 (fr) 2014-10-30
MA38385A1 (fr) 2017-09-29
MY180160A (en) 2020-11-23
US20180185330A1 (en) 2018-07-05
BR112015020600A2 (pt) 2017-07-18
SG11201506218UA (en) 2015-09-29
KR101617812B1 (ko) 2016-05-03
AP2015008674A0 (en) 2015-08-31
US20170087127A1 (en) 2017-03-30
CA2900435C (fr) 2017-02-14
MX346943B (es) 2017-04-06
AU2013387996A1 (en) 2015-09-24
JP6246895B2 (ja) 2017-12-13

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