IN2012DN06061A - - Google Patents
Download PDFInfo
- Publication number
- IN2012DN06061A IN2012DN06061A IN6061DEN2012A IN2012DN06061A IN 2012DN06061 A IN2012DN06061 A IN 2012DN06061A IN 6061DEN2012 A IN6061DEN2012 A IN 6061DEN2012A IN 2012DN06061 A IN2012DN06061 A IN 2012DN06061A
- Authority
- IN
- India
- Prior art keywords
- pyrazol
- thiazole
- disorders
- inhibitors
- diseases
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 2
- 108010089704 Lim Kinases Proteins 0.000 abstract 1
- 102000008020 Lim Kinases Human genes 0.000 abstract 1
- 208000037765 diseases and disorders Diseases 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Ophthalmology & Optometry (AREA)
- Epidemiology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29739710P | 2010-01-22 | 2010-01-22 | |
| PCT/US2011/021970 WO2011091204A1 (en) | 2010-01-22 | 2011-01-21 | 5-(1h-pyrazol-5-yl)thiazole-based compounds for the treatment of diseases and disorders of the eye |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2012DN06061A true IN2012DN06061A (ja) | 2015-09-18 |
Family
ID=43760212
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN6061DEN2012 IN2012DN06061A (ja) | 2010-01-22 | 2011-01-21 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20130059896A1 (ja) |
| EP (1) | EP2525794A1 (ja) |
| JP (1) | JP2013518048A (ja) |
| CN (1) | CN102711758A (ja) |
| AU (1) | AU2011207280A1 (ja) |
| CA (1) | CA2786730A1 (ja) |
| IN (1) | IN2012DN06061A (ja) |
| WO (1) | WO2011091204A1 (ja) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012170951A2 (en) * | 2011-06-10 | 2012-12-13 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| US20120316182A1 (en) | 2011-06-10 | 2012-12-13 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| US9856240B2 (en) | 2011-10-19 | 2018-01-02 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| WO2018055097A1 (en) | 2016-09-23 | 2018-03-29 | Cellipse | Lim kinase inhibitors, pharmaceutical composition and method of use in limk-mediated diseases |
| CN115197166B (zh) * | 2022-07-11 | 2024-07-02 | 安徽英瑞骐生物科技有限公司 | 一种4-甲基-2-肼基苯并噻唑的合成方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4136173A (en) | 1977-01-31 | 1979-01-23 | American Home Products Corp. | Mixed xanthan gum and locust beam gum therapeutic compositions |
| WO1999012910A1 (fr) * | 1997-09-11 | 1999-03-18 | Nissan Chemical Industries, Ltd. | Composes a base de pyrazole et agent de lutte contre les maladies vegetales |
| JP2005501528A (ja) | 2001-06-05 | 2005-01-20 | エクセリクシス・インコーポレイテッド | ｐ５３経路のモディファイヤーとしてのＧＦＡＴｓおよび使用方法 |
| CA2452202A1 (en) | 2001-06-27 | 2003-01-09 | The Walter And Eliza Hall Institute Of Medical Research | Diagnostic methods and agents |
| AU2003302377A1 (en) | 2002-11-27 | 2004-06-18 | Santen Pharmaceutical Co., Ltd. | Remedy for glaucoma containing lim kinase inhibitory compound as active ingredient |
| TWI336257B (en) | 2003-06-13 | 2011-01-21 | Alcon Inc | Ophthalmic compositions containing a synergistic combination of three polymers |
| AU2008236679B2 (en) | 2007-04-03 | 2013-11-28 | Fmc Corporation | Substituted benzene fungicides |
| CA2695857C (en) | 2007-08-08 | 2015-08-04 | Lexicon Pharmaceuticals, Inc. | Kinase inhibitors, compositions comprising them, and methods of their use |
| WO2009131940A1 (en) | 2008-04-21 | 2009-10-29 | Lexicon Pharmaceuticals, Inc. | Limk2 inhibitors, compositions comprising them, and methods of their use |
-
2011
- 2011-01-21 JP JP2012550134A patent/JP2013518048A/ja active Pending
- 2011-01-21 CN CN201180006709.7A patent/CN102711758A/zh active Pending
- 2011-01-21 CA CA2786730A patent/CA2786730A1/en not_active Abandoned
- 2011-01-21 AU AU2011207280A patent/AU2011207280A1/en not_active Abandoned
- 2011-01-21 US US13/574,024 patent/US20130059896A1/en not_active Abandoned
- 2011-01-21 IN IN6061DEN2012 patent/IN2012DN06061A/en unknown
- 2011-01-21 WO PCT/US2011/021970 patent/WO2011091204A1/en active Application Filing
- 2011-01-21 EP EP11702341A patent/EP2525794A1/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| US20130059896A1 (en) | 2013-03-07 |
| CN102711758A (zh) | 2012-10-03 |
| EP2525794A1 (en) | 2012-11-28 |
| AU2011207280A1 (en) | 2012-07-19 |
| CA2786730A1 (en) | 2011-07-28 |
| JP2013518048A (ja) | 2013-05-20 |
| WO2011091204A1 (en) | 2011-07-28 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| WO2014028600A3 (en) | 3-AMINOCYCLOALKYL COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF | |
| TN2013000348A1 (en) | Compounds and compositions as trk inhibitors | |
| PH12014501947A1 (en) | Serine/threonine kinase inhibitors | |
| WO2014028591A3 (en) | N-ALKYLATED INDOLE AND INDAZOLE COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF | |
| MX2015012431A (es) | Pirrol amida como inhibidores. | |
| WO2014031928A3 (en) | Heterocyclic modulators of hif activity for treatment of disease | |
| WO2014179564A8 (en) | Thiazolopyrrolidine inhibitors of ror-gamma | |
| MX2014012695A (es) | Derivados de isoindolona. | |
| MX2013011908A (es) | Composiciones y usos terapeuticos de inhibidores de cinasa epsilon relacionados con cinasa i-kappa b (ikk) y cinasa 1 de union tank. | |
| EA023222B8 (ru) | Пиразолилхиноксалиновые ингибиторы киназы | |
| AU2012214029A8 (en) | Rorgammat inhibitors | |
| MX353806B (es) | Quinolinas como moduladores de cinasas del receptor del factor de crecimiento de fibroblasto (fgfr). | |
| EA024842B9 (ru) | Соединения в качестве модуляторов протеинкиназы pi3k | |
| MX2016008449A (es) | Inhibidores de serina/treonina cinasa. | |
| AU2012258977A8 (en) | Inhibitors of LRRK2 kinase activity | |
| WO2012013282A8 (en) | Bicyclic azaheterocyclic carboxamides as inhibitors of the kinase p70s6k | |
| WO2014031933A3 (en) | Heterocyclic modulators of hif activity for treatment of disease | |
| IN2015DN01151A (ja) | ||
| MY167898A (en) | Co-crystals and salts of ccr3-inhibitors | |
| WO2012048129A3 (en) | Inhibitors of polo-like kinase | |
| WO2014031936A3 (en) | Heterocyclic modulators of hif activity for treatment of disease | |
| MX2012001134A (es) | Composiciones y metodos para inhibicion de la via jak. | |
| MX345127B (es) | Derivados de tiazol. | |
| WO2011150201A3 (en) | Azolyl amide compounds and methods of use thereof | |
| EA032271B9 (ru) | Вещества, фармацевтическая композиция и методы применения при лечении воспалительных заболеваний |