IN2012DE00728A - - Google Patents

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Publication number
IN2012DE00728A
IN2012DE00728A IN728DE2012A IN2012DE00728A IN 2012DE00728 A IN2012DE00728 A IN 2012DE00728A IN 728DE2012 A IN728DE2012 A IN 728DE2012A IN 2012DE00728 A IN2012DE00728 A IN 2012DE00728A
Authority
IN
India
Prior art keywords
solution
organic solvent
heating
imatinib mesylate
clear solution
Prior art date
Application number
Other languages
English (en)
Inventor
Aswini Kumar Sharma
Abhishek Giri
Tapanjyoti Biswal
Govind Singh
Saswata Lahiri
Original Assignee
Fresenius Kabi Oncology Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fresenius Kabi Oncology Ltd filed Critical Fresenius Kabi Oncology Ltd
Priority to PCT/IB2012/054240 priority Critical patent/WO2013136141A1/en
Priority to IN728DE2012 priority patent/IN2012DE00728A/en
Publication of IN2012DE00728A publication Critical patent/IN2012DE00728A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
IN728DE2012 2012-03-13 2012-08-22 IN2012DE00728A (enrdf_load_stackoverflow)

Priority Applications (2)

Application Number Priority Date Filing Date Title
PCT/IB2012/054240 WO2013136141A1 (en) 2012-03-13 2012-08-22 An improved process for the preparation of alpha form of imatinib mesylate
IN728DE2012 IN2012DE00728A (enrdf_load_stackoverflow) 2012-03-13 2012-08-22

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN728DE2012 IN2012DE00728A (enrdf_load_stackoverflow) 2012-03-13 2012-08-22

Publications (1)

Publication Number Publication Date
IN2012DE00728A true IN2012DE00728A (enrdf_load_stackoverflow) 2015-08-21

Family

ID=47010664

Family Applications (1)

Application Number Title Priority Date Filing Date
IN728DE2012 IN2012DE00728A (enrdf_load_stackoverflow) 2012-03-13 2012-08-22

Country Status (2)

Country Link
IN (1) IN2012DE00728A (enrdf_load_stackoverflow)
WO (1) WO2013136141A1 (enrdf_load_stackoverflow)

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW225528B (enrdf_load_stackoverflow) 1992-04-03 1994-06-21 Ciba Geigy Ag
CO4940418A1 (es) 1997-07-18 2000-07-24 Novartis Ag Modificacion de cristal de un derivado de n-fenil-2- pirimidinamina, procesos para su fabricacion y su uso
WO2005077933A1 (en) 2004-02-11 2005-08-25 Natco Pharma Limited Novel polymorphic form of imatinib mesylate and a process for its preparation
UA84462C2 (ru) 2004-04-02 2008-10-27 Институт Фармацевтични Полиморфные модификации кислотно-аддитивных солей иматиниба с метансульфоновой кислотой
KR101348625B1 (ko) * 2004-09-02 2014-01-07 씨아이피엘에이 엘티디. 이매티닙 메실레이트의 안정한 결정형 및 그의 제조방법
WO2006048890A1 (en) 2004-11-04 2006-05-11 Sun Pharmaceutical Industries Limited Imatinib mesylate crystal form and process for preparation thereof
EP1919893A2 (en) 2006-04-27 2008-05-14 Sicor, Inc. Polymorphic forms of imatinib mesylate and processes for their preparation as well as of amorphous imatinib mesylate and form alpha
US20060223816A1 (en) 2006-05-08 2006-10-05 Chemagis Ltd. Imatinib mesylate alpha form and production process therefor
US7550591B2 (en) 2007-05-02 2009-06-23 Chemagis Ltd. Imatinib production process
EP2291366A4 (en) 2008-05-26 2012-06-06 Reddys Lab Ltd Dr PREPARATION OF IMATINIB MESYLATE
PL215042B1 (pl) * 2008-08-01 2013-10-31 Temapharm Spolka Z Ograniczona Odpowiedzialnoscia Sposób wytwarzania imatinibu
US20100330130A1 (en) 2009-05-22 2010-12-30 Actavis Group Ptc Ehf Substantially pure imatinib or a pharmaceutically acceptable salt thereof
US20120309767A1 (en) 2010-02-15 2012-12-06 Sharma Ashwani Process for the preparation of alpha form of imatinib mesylate
PL390611A1 (pl) 2010-03-04 2011-09-12 Tomasz Koźluk Sposób otrzymywania polimorficznej formy alfa i nowa forma polimorficzna mesylanu imatinibu
WO2011158255A1 (en) 2010-06-16 2011-12-22 Aptuit Laurus Private Limited Process for preparation of stable imatintb mesylate alpha form
WO2011157450A1 (en) 2010-06-18 2011-12-22 Krka, D. D., Novo Mesto New polymorphic form of imatinib base and preparation of salts thereof
CN102190649B (zh) * 2011-03-28 2013-01-02 齐鲁天和惠世制药有限公司 一种制备α型甲磺酸伊马替尼的方法

Also Published As

Publication number Publication date
WO2013136141A1 (en) 2013-09-19

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